Keywords: جذب داروی خوراکی; Intestinal permeability; Segmental-dependent permeability; Oral drug absorption;
مقالات ISI جذب داروی خوراکی (ترجمه نشده)
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Keywords: جذب داروی خوراکی; BCS; intestinal permeability; oral drug absorption; solubility-enabling formulations; solubility–permeability interplay
Keywords: جذب داروی خوراکی; First in man pharmacokinetics; Oral drug absorption; Drug development;
Evaluation and optimized selection of supersaturating drug delivery systems of posaconazole (BCS class 2b) in the gastrointestinal simulator (GIS): An in vitro-in silico-in vivo approach
Keywords: جذب داروی خوراکی; Supersaturation; Precipitation; Supersaturating drug delivery systems; Differential scanning calorimetry; Microscopy; In vivo; In vitro; In silico; Oral bioavailability; Oral drug absorption; Pharmacometrics; Bioequivalence;
Investigating drug absorption from the colon: Single-pass vs. Doluisio approaches to in-situ rat large-intestinal perfusion
Keywords: جذب داروی خوراکی; colon; intestinal permeability; oral drug absorption; large intestine; perfusion study;
Segmental-dependent permeability throughout the small intestine following oral drug administration: Single-pass vs. Doluisio approach to in-situ rat perfusion
Keywords: جذب داروی خوراکی; Biopharmaceutics classification system; Intestinal permeability; Segmental-dependent permeability; Oral drug absorption;
Few Drugs Display Flip-Flop Pharmacokinetics and These Are Primarily Associated with Classes 3 and 4 of the BDDCS
Keywords: جذب داروی خوراکی; BDDCS; flip-flop pharmacokinetics; half-life; oral drug absorption; transporters; absorption; pharmacokinetics; intestinal absorption; disposition
In-situ intestinal rat perfusions for human Fabs prediction and BCS permeability class determination: Investigation of the single-pass vs. the Doluisio experimental approaches
Keywords: جذب داروی خوراکی; Biopharmaceutics classification system; Intestinal permeability; Bioequivalence; Biowaiver; Oral drug absorption; Perfusion study;
In silico prediction of the solubility advantage for amorphous drugs – Are there property-based rules for drug discovery and early pharmaceutical development?
Keywords: جذب داروی خوراکی; Poorly soluble drugs; Oral drug absorption; Bioavailability; Amorphous; Molecular modeling; In silico
Enhancement of oral drug absorption—Effect of lipid conjugation on the enzymatic stability and intestinal permeability of l-Glu-l-Trp-NH2
Keywords: جذب داروی خوراکی; IM862; Oral drug absorption; Lipid conjugation; Caco-2; Stability; Permeability
Biorelevant dissolution media as a predictive tool for glyburide a class II drug
Keywords: جذب داروی خوراکی; Solubility; Biorelevant dissolution media (BDM); In vitro dissolution; Permeability; IVIVC; Oral drug absorption; Prediction; Computational simulation; In vitro/in silico; Dynamic dissolution
Site of drug absorption after oral administration: Assessment of membrane permeability and luminal concentration of drugs in each segment of gastrointestinal tract
Keywords: جذب داروی خوراکی; Oral drug absorption; Regional difference; Drug permeability; Luminal concentration; Fluid volume; Gastrointestinal tract
Magnesia-zirconia based mimetic biomembrane chromatography for predicting human drug absorption
Keywords: جذب داروی خوراکی; Magnesia-zirconia composite; Oral drug absorption; Mimetic biomembrane stationary phase;