
[1,2,4]Triazolo[1,5-c]pyrimidines as adenosine receptor antagonists: Modifications at the 8 position to reach selectivity towards A3 adenosine receptor subtype
Keywords: G protein-coupled receptor; Adenosine receptor; A3 antagonist; [1,2,4]triazolo[1,5-c]pyrimidine; Molecular modeling; Docking; AR; adenosine receptor; cAMP; cyclic adenosine monophosphate; CCPA; 2-chloro-N6-cyclopentyladenosine; CHO; chinese hamster ovary;