Keywords: رادیولینگ; Radioligand; Biotoxins; Shellfish; Monitoring; Atlantic coastline;
مقالات ISI رادیولینگ (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: رادیولینگ; Molecular imaging; Radioligand; Serotonin; 5-HT4; SPECT;
Keywords: رادیولینگ; HPFA, high-performance frontal analysis; PET, positron emission tomography; PBS, phosphate buffered saline; MIV, minimum injection volumePlasma protein binding; High-performance frontal analysis (HPFA); Positron emission tomography (PET); Radioligand; Min
Keywords: رادیولینگ; CB1R; Cannabis; Cannabinoid; Marijuana; PET; Rimonabant; Radioligand; Prefrontal cortex; Schizophrenia;
Are dopamine receptor and transporter changes in Rett syndrome reflected in Mecp2-deficient mice?
Keywords: رادیولینگ; Autoradiography; Binding potential; Gene mutation; Intellectual disability; Neurotransmitter; Nigrostriatal pathway; Postmortem; Positron emission tomography; Partial volume correction; Radioligand;
Preclinical comparison study between [18F]fluoromethyl-PBR28 and its deuterated analog in a rat model of neuroinflammation
Keywords: رادیولینگ; Translocator protein; Neuroinflammation; Deuterated methoxy group; PET; Radioligand; PBR28;
[11C]AZ10419096 - a full antagonist PET radioligand for imaging brain 5-HT1B receptors
Keywords: رادیولینگ; 5-HT1B receptor; Antagonist; Radioligand; Carbon-11; PET;
The binding orientation of epibatidine at α7 nACh receptors
Keywords: رادیولینگ; Cys-loop; Ion channel; Radioligand; Epibatidine; Agonist; α7 nACh; Nicotinic; Receptor; AChBP; 5-HT; 5-hydroxytryptamine; nACh; nicotinic acetylcholine; GABA; gamma-aminobutyric acid; HEK; human embryonic kidney; AChBP; acetylcholine binding protein; 5HT
The binding orientations of structurally-related ligands can differ; AÂ cautionary note
Keywords: رادیولینگ; Cys-loop; Ion channel; Receptor; Radioligand; 5-HT3; Agonist; Antagonist; Crystal; Binding; Granisetron; Tropisetron; Ligand; Structure; Synthesis; 5-HT; 5-hydroxytryptamine; nACh; nicotinic acetylcholine; GABA; gamma-aminobutyric acid; HEK; human embryon
Biochemical and behavioral effects of PDE10A inhibitors: Relationship to target site occupancy
Keywords: رادیولینگ; PDE10A; Antipsychotic; Conditioned avoidance response; Catalepsy; Radioligand; Occupancy;
A practical process for the preparation of [32P]S1P and binding assay for S1P receptor ligands
Keywords: رادیولینگ; Competitive binding assay; Phosphorus-32; Radioligand; Sphingosine 1-phosphate; Sphingosine 1-phosphate Receptors; Sphingosine kinase 1;
Radiosynthesis and in vitro validation of 3H-NS14492 as a novel high affinity alpha7 nicotinic receptor radioligand
Keywords: رادیولینگ; Bmax; maximum density; 125I-BTX; 125I-α-bungarotoxin; Kd; dissociation constant; Ki; inhibition constant; NSB; non-specific binding; OD; optical density; PAM; positive allosteric modulator; SB; specific binding; TB; total binding; TE; tissue equivalent;
[carbonyl-11C]4-Fluoro-N-methyl-N-(4-(6-(methylamino)pyrimidin-4-yl)thiazol-2-yl)benzamide ([11C]FIMX) is an effective radioligand for PET imaging of metabotropic glutamate receptor 1 (mGluR1) in monkey brain
Keywords: رادیولینگ; mGluR1; Radioligand; PET; Carbon-11; Monkey; Brain;
In vitro and ex vivo characterization of (−)-TZ659 as a ligand for imaging the vesicular acetylcholine transporter
Keywords: رادیولینگ; Vesicular acetylcholine transporter; Radioligand; Binding assay; Autoradiography
Synthesis, in vitro and in vivo evaluation of 1,3,5-triazines as cannabinoid CB2 receptor agonists
Keywords: رادیولینگ; Cannabinoid receptor; CB2R agonists; Triazines; Radioligand;
Acute repeated intracerebroventricular injections of angiotensin II reduce agonist and antagonist radioligand binding in the paraventricular nucleus of the hypothalamus and median preoptic nucleus in the rat brain
Keywords: رادیولینگ; Angiotensin; Brain; Hypertension; Desensitization; Radioligand; Water intake; Saline intake; AT1 angiotensin receptors; Thirst;
The binding characteristics and orientation of a novel radioligand with distinct properties at 5-HT3A and 5-HT3AB receptors
Keywords: رادیولینگ; Antagonist; Cys-loop; Ion channel; Radioligand; 5-HT3; Agonist; 5-HT; 5-hydroxytryptamine; nACh; nicotinic acetylcholine; GABA; gamma-aminobutyric acid; HEK; human embryonic kidney; AChBP; acetylcholine binding protein; 5HTBP; an AChBP mutant modified to
N-(4-[18F]-fluoropyridin-2-yl)-N-{2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl}carboxamides as analogs of WAY100635. New PET tracers of serotonin 5-HT1A receptors
Keywords: رادیولینگ; 5-HT1A; Positron emission tomography; Fluorine-18; Radioligand; N-(4-[18F]-fluoropyridin-2-yl)-N-{2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl}carboxamidesPET, positron emission tomography; 5-HT1A, receptor 1A of 5-hydroxytryptamine; 5-HT, 5-hydroxytryptami
Synthesis, radiolabeling and in vivo evaluation of [11C](R)-1-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT7 receptor
Keywords: رادیولینگ; 5-HT7 receptor; PET; Radioligand; Arylpiperazine; SB-269970
Characterization of FlipIDAM as a SERT-selective SPECT imaging agent
Keywords: رادیولینگ; DASB; (N,N-dimethyl-2-(2-amino-4-cyanophenylthio)benzylamine); IACUC; Institutional Animal Care and Use Committee; (+)-McN5652; trans-1,2,3,5,6,10- < beta > -hexahydro-6-[4-(methylthio)phenyl-[pyrrolo-[2,1- < alpha >]isoquinoline; FlipIDAM (4); (2-
Synthesis and evaluation of new radioligands [11C]A-833834 and [11C]A-752274 for positron-emission tomography of α7-nicotinic acetylcholine receptors
Keywords: رادیولینگ; Positron emission tomography; PET; Radioligand; Nicotinic acetylcholine receptor; α7-nAChR
[18F]FE@SNAP-A new PET tracer for the melanin concentrating hormone receptor 1 (MCHR1): Microfluidic and vessel-based approaches
Keywords: رادیولینگ; MCHR1; Fluorine-18; PET; Microfluidic; SNAP-7941; Radioligand;
[18F](R)-5-chloro-1-(1-cyclopropyl-2-methoxyethyl)-3-(4-(2-fluoroethoxy)-2,5-dimethyl phenylamino)pyrazin-2(1H)-one: Introduction of N3-phenylpyrazinones as potential CRF-R1 PET imaging agents
Keywords: رادیولینگ; Corticotropin-releasing factor; Positron Emission Tomography; Antidepressants; Anxiolytics; Radioligand;
5-(5-(6-[11C]methyl-3,6-diazabicyclo[3.2.0]heptan-3-yl)pyridin-2-yl)-1H-indole as a potential PET radioligand for imaging cerebral α7-nAChR in mice
Keywords: رادیولینگ; Positron emission tomography; Radioligand; Nicotinic acetylcholine receptors; α7-nAChR;
Characterization of [3H]Lu AE60157 ([3H]8-(4-methylpiperazin-1-yl)-3-phenylsulfonylquinoline) binding to 5-hydroxytryptamine6 (5-HT6) receptors in vivo
Keywords: رادیولینگ; 5-HT6 receptor; Striatum; In vivo binding; Radioligand; Occupancy; Brain
Radiosynthesis of [11C]SNAP-7941-the first PET-tracer for the melanin concentrating hormone receptor 1 (MCHR1)
Keywords: رادیولینگ; MCHR1; SNAP-7941; Carbon-11; Radioligand; PET;
Evolution of microglial activation in ischaemic core and peri-infarct regions after stroke: A PET study with the TSPO molecular imaging biomarker [11C]vinpocetine
Keywords: رادیولینگ; Positron emission tomography (PET); Radioligand; [11C]vipocetine; Peripheral benzodiazepine receptor (PBR); 18 kD translocator protein (TSPO); Stroke; Ischaemic core; Peri-infarct zone; Microglia; Molecular imaging biomarker;
Synthesis of fluorine-18-labelled TSPO ligands for imaging neuroinflammation with Positron Emission Tomography
Keywords: رادیولینگ; Fluorine-18; 18 kDa TSPO; Radioligand; Neuroinflammation
Identifying improved TSPO PET imaging probes through biomathematics: The impact of multiple TSPO binding sites in vivo
Keywords: رادیولینگ; TSPO; PET; Radioligand; Biomathematical modelling; Multiple binding affinities;
Serotonin-1A receptors in major depression quantified using PET: Controversies, confounds, and recommendations
Keywords: رادیولینگ; Major depressive disorder (MDD); Neuroimaging; Permeability-glycoprotein (P-gp); Positron emission tomography (PET); Radioligand; Serotonin-1A (5-HT1A) receptors;
Synthesis of 6-[18F]fluoro-PBR28, a novel radiotracer for imaging the TSPO 18 kDa with PET
Keywords: رادیولینگ; Translocator protein (TSPO); Radioligand; Fluorine-18; PET tracer; Neuroinflammation
Characterization of a novel and selective CB1 antagonist as a radioligand for receptor occupancy studies
Keywords: رادیولینگ; Cannabinoid; Radioligand; Receptor occupancy; Obesity
[125I]YP20: A novel radioligand specific for the extracellular domain of the CRF1 receptor
Keywords: رادیولینگ; CRF; CRF1 receptor; Radioligand; Extracellular domain
Radiosynthesis and ex vivo evaluation of (R)-(−)-2-chloro-N-[1-11C-propyl]n-propylnorapomorphine
Keywords: رادیولینگ; PET; Agonist; D2; D3; Dopamine; Apomorphine; 2-Cl-[11C]-(−)-NPA; [11C]-(−)-NPA; Radioligand; P-glycoprotein; Amphetamine
In vitro binding characteristics of [3H]AZ11637326, a novel α7-selective neuronal nicotinic receptor agonist radioligand
Keywords: رادیولینگ; Nicotinic; Radioligand; Alpha 7
Pharmacological characterization of the cannabinoid CB1 receptor PET ligand ortholog, [3H]MePPEP
Keywords: رادیولینگ; Cannabinoid; CB1; MePPEP; PET; Radioligand; Inverse agonist
In vivo studies of the SERT-selective [18F]FPBM and VMAT2-selective [18F]AV-133 radiotracers in a rat model of Parkinson's disease
Keywords: رادیولینگ; Brain imaging; Radioligand; SERT; VMAT2; Parkinson's disease
Development of radioligands with optimized imaging properties for quantification of nicotinic acetylcholine receptors by positron emission tomography
Keywords: رادیولینگ; PET; Positron emission tomography; nAChR; Radioligand; Nicotine; Nicotinic acetylcholine receptor
Synthesis, radiofluorination and first evaluation of [18F]fluorophenylsulfonyl- and [18F]fluorophenylsulfinyl-piperidines as serotonin 5-HT2A receptor antagonists for PET
Keywords: رادیولینگ; Radiofluorination; 5-HT2A antagonist; PET; Radioligand; Autoradiography
High-resolution imaging of brain 5-HT1B receptors in the rhesus monkey using [11C]P943
Keywords: رادیولینگ; 5-HT1B receptor; Antagonist; PET; Radioligand; C-11; HRRT
Multiple strategies for the preparation of a sulfur-35 labeled NPC1L1 radioligand
Keywords: رادیولینگ; Sulfur-35; NPC1L1; Radioligand; Synthesis
Development of a selective and potent radioactive ligand for histamine H3 receptors: A compound potentially useful for receptor occupancy studies
Keywords: رادیولینگ; Histamine H3 receptors; Inverse agonist; Radioligand; Receptor occupancy;
Synthesis and in vitro autoradiographic evaluation of a novel high-affinity radioiodinated ligand for imaging brain cannabinoid subtype-1 receptors
Keywords: رادیولینگ; SPECT; PET; CB1 receptors; Radioiodination; Radioligand;
Identification and characterization of a selective radioligand for melanin-concentrating hormone 1-receptor (MCH1R)
Keywords: رادیولینگ; Melanin-concentrating hormone 1-receptor; Antagonist; Radioligand; Receptor occupancy
Characterization of two novel tritiated radioligands for labelling Neuropeptide FF (NPFF1 and NPFF2) receptors
Keywords: رادیولینگ; Radioligand; Neuropeptide FF; Receptor; Binding
Examining the binding properties of MK-0974: A CGRP receptor antagonist for the acute treatment of migraine
Keywords: رادیولینگ; Migraine; CGRP; Telcagepant; Radioligand; MK-0974
Synthesis and biological evaluation of novel carbon-11 labeled pyridyl ethers: candidate ligands for in vivo imaging of α4β2 nicotinic acetylcholine receptors (α4β2-nAChRs) in the brain with positron emission tomography
Keywords: رادیولینگ; Nicotinic acetylcholine receptor; nAChR; PET; Radioligand
A change of in vivo characteristics depending on specific activity of radioiodinated (+)-2-[4-(4-iodophenyl)piperidino]cyclohexanol [(+)-pIV] as a ligand for sigma receptor imaging
Keywords: رادیولینگ; (+)-p-Iodovesamicol; Sigma-1 receptor; Radioligand; Biodistribution; High and low specific activity radiolabeled (+)-pIV
Preparation and first evaluation of [18F]FE@SUPPY: a new PET tracer for the adenosine A3 receptor
Keywords: رادیولینگ; Adenosine; PET; Receptor; Fluorine-18; Radioligand
[3H]BMS-599240 — A novel tritiated ligand for the characterization of BACE1 inhibitors
Keywords: رادیولینگ; Alzheimer disease; β-amyloid precursor protein; BACE; BMS-599240; Radioligand; β-Secretase