
RGS proteins destroy spare receptors: Effects of GPCR-interacting proteins and signal deamplification on measurements of GPCR agonist potency
Keywords: سازگاری گیرنده; Agonist potency; Receptor conformation; G protein-mediated signaling; GPCR-interacting proteins (GIPs); Regulator of G protein signaling proteins (RGS proteins); Functional selectivity;