
The dual modulatory effects of efavirenz on GABAA receptors are mediated via two distinct sites
Keywords: Recombinant GABAA receptors; Adverse CNS side effects; Picrotoxin; AIDS; Antiretroviral; BDZ; benzodiazepine; CNS; central nervous system; DMSO; dimethyl sulfoxide; DZ; diazepam; EFAV; efavirenz; FLU; flumazenil; LGICs; ligand-gated ion channels; HEK293;