Keywords: مطالعه SAR; Chromene conjugates; Quinoline conjugates; Anti-proliferative activity; Molecular docking; SAR study;
مقالات ISI مطالعه SAR (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: مطالعه SAR; Oxadiazole-benzohydrazone hybrids; Leishmaniasis; SAR study; Molecular docking studies; DFT; Selectivity index;
Keywords: مطالعه SAR; Opiorphin analogs; SAR study; Neutral endopeptidase; AP-N; Glycopeptides pain;
Keywords: مطالعه SAR; KBXWOBGGKRASMV-UUWRZZSWSA-N; SJCIADFNBNFHIX-WJOKGBTCSA-N; JMSLKPFDIUWLEK-WJOKGBTCSA-N; QRCPXBRMOBALAS-WJOKGBTCSA-N; HHZGNTLQYHMRTI-WJOKGBTCSA-N; SXBFQBBEMSDWMW-SSEXGKCCSA-N; LRGQQQITIJMVGU-SSEXGKCCSA-N; GHFUEMFRBNDQCW-SSEXGKCCSA-N; OBTFKDIQADGXQP-SSEXGKCC
Synthesis and antibacterial studies of teixobactin analogues with non-isostere substitution of enduracididine
Keywords: مطالعه SAR; Teixobactin analogues; Ser ligation; SAR study;
Synthesis and SAR study of new hydroxy and chloro-substituted 2,4-diphenyl 5H-chromeno[4,3-b]pyridines as selective topoisomerase IIα-targeting anticancer agents
Keywords: مطالعه SAR; Anticancer agents; 5H-Chromeno[4,3-b]pyridines; Hydroxyl and chlorine-substitution; Selective topoisomerase IIα inhibition; SAR study;
SAR studies on truxillic acid mono esters as a new class of antinociceptive agents targeting fatty acid binding proteins
Keywords: مطالعه SAR; Fatty acid binding protein; FABP inhibitor; Anti-nociceptive agent; Anti-inflammatory agent; SAR study; Computer-aided design; Molecular docking;
Synthesis and SAR study of novel sarsasapogenin derivatives as potent neuroprotective agents and NO production inhibitors
Keywords: مطالعه SAR; Sarsasapogenin; Natural product; Neuroprotective activity; SAR study;
Synthesis and structure-activity relationship of teixobactin analogues via convergent Ser ligation
Keywords: مطالعه SAR; Teixobactin analogues; SAR study; Ser/Thr ligation;
Structure-activity relationship study of small molecule inhibitors of the DEPTOR-mTOR interaction
Keywords: مطالعه SAR; mTOR; DEPTOR; Multiple myeloma; Cytotoxicity; SAR study;
Inhibition of LPS-stimulated ROS production by fluorinated and hydroxylated chalcones in RAW 264.7 macrophages with structure-activity relationship study
Keywords: مطالعه SAR; Fluorinated and hydroxylated chalcones; Inhibition of LPS-stimulated ROS production; SAR study;
Glycine-replaced derivatives of [Pro3,DLeu9]TL, a temporin L analogue: Evaluation of antimicrobial, cytotoxic and hemolytic activities
Keywords: مطالعه SAR; Antimicrobial peptides; Temporin L analogues; SAR study; Spectroscopy studies;
An overview of benzo[b]thiophene-based medicinal chemistry
Keywords: مطالعه SAR; Heterocyclic compound; Benzothiophene; Synthesis; Anti-microbial; Anti-cancer; SAR study;
Synthesis and biological evaluation of analogues of the potent ADAM8 inhibitor cyclo(RLsKDK) for the treatment of inflammatory diseases and cancer metastasis
Keywords: مطالعه SAR; ADAM8 inhibitors; Cancer metastasis; Cyclic peptides; Peptidomimetics; SAR study
Synthesis and SAR of 4-methyl-5-pentylbenzene-1,3-diol (MPBD), produced by Dictyostelium discoideum
Keywords: مطالعه SAR; 4-Methyl-5-pentylbenzene-1,3-diol; Dictyostelium discoideum; SAR study; Antimicrobial activity
Hydrophobic substituents increase the potency of salacinol, a potent α-glucosidase inhibitor from Ayurvedic traditional medicine 'Salacia'
Keywords: مطالعه SAR; α-Glucosidase inhibitor; In silico docking study; Salacinol; Salacia; SAR study;
Structure-activity relationship studies on acremomannolipin A, the potent calcium signal modulator with a novel glycolipid structure 4: Role of acyl side chains on d-mannose
Keywords: مطالعه SAR; Acremomannolipin A; Glycolipid; Calcium signal modulator; Acremonium strictum; SAR study;
Design, synthesis and docking study of novel tetracyclic oxindole derivatives as α-glucosidase inhibitors
Keywords: مطالعه SAR; Tetracyclic isatins; α-Glucosidase inhibitors; Docking study; Phenanthridine derivatives; SAR study
Isolation, ECD assisted structural analyses, biosynthetic discussions, and biological activities of epi-cochlioquinones D and its derivatives
Keywords: مطالعه SAR; Absolute configuration; Calculations of ECD spectra; Difference ECD spectra; Biological properties; Biosynthetic discussions; SAR study;
Isolation, structure identification and SAR studies on thiosugar sulfonium salts, neosalaprinol and neoponkoranol, as potent α-glucosidase inhibitors
Keywords: مطالعه SAR; Neoponkoranol; Neosalaprinol; α-Glucosidase inhibitor; Salacia; SAR study;
Discovery and SAR study of 3-(tert-butyl)-4-hydroxyphenyl benzoate and benzamide derivatives as novel farnesoid X receptor (FXR) antagonists
Keywords: مطالعه SAR; FXR; FXR antagonist; SAR study; Non-steroidal
Multicomponent assembly of 4-aza-podophyllotoxins: A fast entry to highly selective and potent anti-leukemic agents
Keywords: مطالعه SAR; Multicomponent reactions; Aza-podophyllotoxins; Anti-leukemic agents; AML; SAR study; Etoposide; APT; 4-aza-2,3-didehydropodophyllotoxins; MCR; multicomponent reaction;
Structure-activity relationship studies on acremomannolipin A, the potent calcium signal modulator with a novel glycolipid structure 3: Role of the length of alditol side chain
Keywords: مطالعه SAR; Acremomannolipin A; Glycolipid; Calcium signal modulator; Acremonium strictum; SAR study;
Structure activity relationship (SAR) study of benzimidazole scaffold for different biological activities: A mini-review
Keywords: مطالعه SAR; Anthelmintics; Benzimidazole; Heterocyclic ring systems; Pharmacological activities; SAR study; NPY; neuropeptide; CYP450; cytochrome P450; HBV; hepatitis B virus; HCV; hepatitis C virus; RSV; respiratory syncytial virus; VV; varicella virus; BVDV; bovine
Design, synthesis, and SAR of embelin analogues as the inhibitors of PAI-1 (plasminogen activator inhibitor-1)
Keywords: مطالعه SAR; Embelin; Natural product; PAI-1; Inhibitory activity; SAR study
Discovery and SAR study of hydroxyacetophenone derivatives as potent, non-steroidal farnesoid X receptor (FXR) antagonists
Keywords: مطالعه SAR; FXR antagonist; SAR study; Hydroxyacetophenone derivatives; Non-steroidal;
Structure-activity relationship studies on acremomannolipin A, the potent calcium signal modulator with a novel glycolipid structure 2: Role of the alditol side chain stereochemistry
Keywords: مطالعه SAR; Acremomannolipin A; Glycolipid; Calcium signal modulator; Acremonium strictum; SAR study;
Synthesis, biological evaluation and SAR studies of novel bicyclic antitumor platinum(IV) complexes
Keywords: مطالعه SAR; Cisplatin; Platinum(IV) complexes; SAR study; Cancer; Biological evaluation; Malonatoplatinum complexes
A novel necroptosis inhibitor-necrostatin-21 and its SAR study
Keywords: مطالعه SAR; Necroptosis; Nec-21; Inhibitor; SAR study; RIP1; JNK3;
N-cholesteryl amino acid conjugates and their antimicrobial activities
Keywords: مطالعه SAR; N-Cholesteryl amino acid conjugates; Antimicrobial agents; Methicillin-resistant Staphylococcus aureus; SAR study;
Novel complex crystal structure of prolyl hydroxylase domain-containing protein 2 (PHD2): 2,8-Diazaspiro[4.5]decan-1-ones as potent, orally bioavailable PHD2 inhibitors
Keywords: مطالعه SAR; 2,8-Diazaspiro[4.5]decan-1-one; Prolyl hydroxylase domain-containing protein 2 (PHD2); PHD inhibitors; Hypoxia inducible factor (HIF); PHD2 crystal structure; SAR study;
Synthesis and evaluation of N-substituted nipecotic acid derivatives with an unsymmetrical bis-aromatic residue attached to a vinyl ether spacer as potential GABA uptake inhibitors
Keywords: مطالعه SAR; GABA uptake; Chelation-controlled Heck reaction; Fries rearrangment; Aromatic fluoro-compounds; SAR study;
In vitro inhibition of translation initiation by N,Nâ²-diarylureas-potential anti-cancer agents
Keywords: مطالعه SAR; SAR study; N,Nâ²-Diarylureas; Inhibition of translation initiation; Ternary complex; Phosphorylation of eIF2α; Anti-cancer drugs;
Synthesis and biological activity of new homolupanes and homolupane saponins
Keywords: مطالعه SAR; Homobetulin; Homobetulinic acid; Glycosylation; Lupane saponins; Homolupane saponins; SAR study;
Weight loss effects of quaternary salts of 5-amino-1-(chloromethyl)-1,2-dihydro-3H-benz[e]indoles; structure-activity relationships
Keywords: مطالعه SAR; AIBN; 2,2â²-azobis[isobutyronitrile]; CBI; seco-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one; CSA; camphorsulfonic acid; DIPEA; diisopropylethylamine; DMA; dimethylacetamide; DMAP; 4-dimethylaminopyridine; EDCI·HCl; N-ethyl-Nâ²-(3-dimethylaminopr
Discovery of a series of potent arylthiadiazole H3 antagonists
Keywords: مطالعه SAR; H3 antagonists; SAR study
Synthesis and SAR study of diphenylbutylpiperidines as cell autophagy inducers
Keywords: مطالعه SAR; Autophagy; Diphenylbutylpiperidines; Synthesis; SAR study; Inducers;
Discovery of highly potent agents against influenza A virus
Keywords: مطالعه SAR; Hit-to-lead optimization; Influenza A virus; SAR study; M2; matrix-2 protein; SAR; structure-activity relationship;
Role of the side chain stereochemistry in the α-glucosidase inhibitory activity of kotalanol, a potent natural α-glucosidase inhibitor
Keywords: مطالعه SAR; Kotalanol; α-Glucosidase inhibitor; Salacia; SAR study; Selective inhibition
Structural modification of a specific antimicrobial lead against Helicobacter pylori discovered from traditional Chinese medicine and a structure–activity relationship study
Keywords: مطالعه SAR; Anti-Helicobacter pylori lead; Structural modification; SAR study
Potent agonists of the Hedgehog signaling pathway
Keywords: مطالعه SAR; Hedgehog signaling pathway; Agonist; SAR study; Small molecule;
Exploration of novel thiobarbituric acid-, rhodanine- and thiohydantoin-based HIV-1 integrase inhibitors
Keywords: مطالعه SAR; HIV-1; Integrase inhibitors; SAR study; Thiobarbituric acid; Rhodanine; Thiohydantoin
Discovery of N-aryl-9-oxo-9H-fluorene-1-carboxamides as a new series of apoptosis inducers using a cell- and caspase-based high-throughput screening assay. 1. Structure–activity relationships of the carboxamide group
Keywords: مطالعه SAR; Apoptosis inducers; HTS; Anticancer agents; SAR study
Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones
Keywords: مطالعه SAR; Tuberculosis; Pyrazolones; Pyrazole; SAR study
Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis
Keywords: مطالعه SAR; Tuberculosis; 5-Hydroxy-pyrazole; Pyrazolone; SAR study
Design, synthesis, inhibitory activity, and SAR studies of hydrophobic p-aminosalicylic acid derivatives as neuraminidase inhibitors
Keywords: مطالعه SAR; Influenza; Neuraminidase inhibitor; p-Aminosalicylic acid derivatives; SAR study
Synthesis, antimalarial activity, structure-activity relationship analysis of thieno-[3,2-b]benzothiazine S,S-dioxide analogs
Keywords: مطالعه SAR; Thieno; 1,4-Benzothiazines; Cyclization; Antimalarial; SAR study;
Design, synthesis and biological evaluation of piperazine analogues as CB1 cannabinoid receptor ligands
Keywords: مطالعه SAR; CB1 receptor antagonists; 1-Benzhydrylpiperazine; SAR study; Rimonabant; Piperazine; Cannabinoid receptor; Anti-obesity
Antibacterial activity of a novel series of 3-bromo-4-(1H-3-indolyl)-2,5-dihydro-1H-2,5-pyrroledione derivatives – An extended structure–activity relationship study
Keywords: مطالعه SAR; SAR study; Antibacterial compounds; Indole derivatives; Resistance of Staphylococcus aureus
Parallel synthesis and SAR study of novel oxa-steroids as potent and selective progesterone receptor antagonists
Keywords: مطالعه SAR; Progesterone; Receptor; Antagonist; oxa-Steroid; Glucocorticoid; Parallel synthesis; SAR study; In vitro; In vivo