دانلود مقالات ISI درباره Spirocyclic Piperidines + ترجمه فارسی

Oxa-Pictet–Spengler reaction as key step in the synthesis of novel σ receptor ligands with 2-benzopyran structure

Keywords: σ ligands; Oxa-Pictet–Spengler reaction; Intramolecular Oxa-Pictet–Spengler reaction; 2-Benzopyrans; Spirocyclic piperidines; Tricyclic systems; Aryl-N-distance

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

One-pot synthesis and sigma receptor binding studies of novel spirocyclic-2,6-diketopiperazine derivatives

Keywords: BWOLKJFUETYFAF-UHFFFAOYSA-N; DQMQUKUXAXPUCX-UHFFFAOYSA-N; DSMDWLOPPRGRFN-UHFFFAOYSA-N; YOVRBAYQBRCCLG-UHFFFAOYSA-N; LPOFDRFGEPRFCF-UHFFFAOYSA-N; KEFONRLCIUIPSX-UHFFFAOYSA-N; VLTOBCXOBHNDDX-UHFFFAOYSA-N; QVHSKMHZXNZQNN-UHFFFAOYSA-N; HVRYHFQLCLCWSE-UHFFFAOY

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis and biological evaluation of spirocyclic antagonists of CCR2 (chemokine CC receptor subtype 2)

Keywords: Chemokine CC receptor subtype 2 (CCR2) antagonists; Oxa-Pictet–Spengler reaction; Ethylene sulfate; Appel reaction; Polymer-bound triphenylphosphine; Spirocyclic piperidines; Receptor binding studies; Ca2+ flux; β-Arrestin recruitment; Structure–activity-

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2015 سفارش ترجمه

Pyridine analogues of spirocyclic σ1 receptor ligands

Keywords: σ1 Receptor ligands; Spirocyclic piperidines; Electron density; Pyranopyridines; Structure affinity relationships

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2014 سفارش ترجمه

Synthesis and σ receptor affinity of regioisomeric spirocyclic furopyridines

Keywords: σ1 receptor ligands; Spirocyclic piperidines; Furopyridines; Regioisomers; Structure affinity relationships

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2014 سفارش ترجمه

Synthesis, radiofluorination and pharmacological evaluation of a fluoromethyl spirocyclic PET tracer for central σ1 receptors and comparison with fluoroalkyl homologs

Keywords: DMT; N,N-dimethyltryptamine; MAM; mitochondrion-associated ER membrane; ER; endoplasmatic reticulum; BiP; binding immunoglobulin protein; IP3R; inositol 1,4,5-triphosphate receptor; PET; positron emission tomography; EMP; emopamil-binding protein; VAChT;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2012 سفارش ترجمه

Divergent approach to the polymaxenolide and pinnaic acid cores

Keywords: Pinnaic acid; Polymaxenolide; Spirocyclic pyrans; Spirocyclic piperidines;

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2011 سفارش ترجمه

Synthesis, pharmacological activity and structure affinity relationships of spirocyclic σ1 receptor ligands with a (2-fluoroethyl) residue in 3-position

Keywords: σ1 Receptor ligands; Spirocyclic piperidines; [18F] Radiotracer; Neuroimaging; Structure affinity relationships; Ring contraction;

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2011 سفارش ترجمه

5D-QSAR for spirocyclic σ1 receptor ligands by Quasar receptor surface modeling

Keywords: σ1 Receptor ligands; Spirocyclic piperidines; 5D-QSAR; σ1 Receptor surface

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2010 سفارش ترجمه

Synthesis of σ receptor ligands with unsymmetrical spiro connection of the piperidine moiety

Keywords: σ Receptor ligands; Spirocyclic piperidines; Structure–affinity relationships; Receptor binding studies; Halogen–metal exchange; Transmetallation

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis of spirocyclic σ1 receptor ligands as potential PET radiotracers, structure–affinity relationships and in vitro metabolic stability

Keywords: σ1 Receptor antagonists; Spirocyclic piperidines; Metabolism; 18F Radiotracer; Neuroimaging; Structure–affinity-relationships

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2009 سفارش ترجمه

Synthesis and structure–affinity relationships of novel spirocyclic σ receptor ligands with furopyrazole structure

Keywords: Spirocyclic piperidines; Pharmacophore model; Molecular modeling experiments; Theoretical considerations

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2008 سفارش ترجمه