Keywords: روابط فعالیت ساختاری; Metallo β-lactamase; Antibiotic resistance; Carbapenemase; Inhibitors; Structure activity relationships;
مقالات ISI روابط فعالیت ساختاری (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: روابط فعالیت ساختاری; AD; Alzheimer's disease; Aβ; amyloid β peptide; APP; amyloid precursor protein; BACE1; β-amyloid cleavage enzyme 1, β-secretase 1; GSM; gamma secretase modulator; LHS; left hand side; NSAID; non-steroidal anti-inflammatory drug; SAR; structure activ
Keywords: روابط فعالیت ساختاری; Flavokawain; Cancer; Cytotoxic; Apoptosis; Structure activity relationships; P53; Akt/mTor;
Keywords: روابط فعالیت ساختاری; Chemokine receptors; CCR5; CCR2; Positive allosteric modulator; 2-Benzazepines; TAK-779; TAK-652; Structure-affinity relationships; Structure activity relationships;
Keywords: روابط فعالیت ساختاری; IRAK4; Kinase; Inflammation; Structure activity relationships; Aminopyrimidine;
Keywords: روابط فعالیت ساختاری; Pactamycin; Nanoparticles; Structure activity relationships; Structural derivatization
Keywords: روابط فعالیت ساختاری; Chalcone; Anti-malarial; Anti-parasitic; Mechanism of actions; Molecular targets; Structure activity relationships;
Keywords: روابط فعالیت ساختاری; GPA; green peach aphid (Myzus persicae); IRM; insecticide resistance management; IRAC; Insecticide Resistance Action Committee; MTH; 2-CH3-thiazole; nAChR; nicotinic acetylcholine receptors; SAR; structure activity relationships; SFI; sulfoximine insectic
Discovery of 1-(4-((3-(4-methylpiperazin-1-yl)propyl)amino)benzyl)-5-(trifluoromethyl)pyridin-2(1H)-one, an orally active multi-target agent for the treatment of diabetic nephropathy
Keywords: روابط فعالیت ساختاری; ACR; albumin-to-creatinine ratio; AUC0-t; area under the curve; BuOH; n-butanol; BUN; blood urea nitrogen; Cmax; peak concentration; C13-NMR; C13-nuclear magnetic resonance; CCr; creatinine clearance rate; CCR2; CCchemkin receptor 2; CDCl3; Deuterotrichlo
Systematic variation of the benzenesulfonamide part of the GluN2A selective NMDA receptor antagonist TCN-201
Keywords: روابط فعالیت ساختاری; NMDA receptor; GluN2A selective antagonists; TCN-201; Synthesis; Electrophysiology; Two electrode voltage clamp; Structure activity relationships; Antagonistic activity;
5-Bromoindirubin 3â²-(O-oxiran-2-ylmethyl)oxime: A long-acting anticancer agent and a suicide inhibitor for epoxide hydrolase
Keywords: روابط فعالیت ساختاری; ATP; adenosine 5â²-triphosphate; C1; methylene; C2; ethylene; C3; propylene; CDK; cyclin-dependent kinase; Cys; cysteine residue; DMF; N,N-dimethylformamide; DMSO; dimethyl sulfoxide; EI; electron impact; Epox/5-Br-Ind; 5-bromoindirubin 3â²-(O-oxiran-2-
Discovery of selective ATP-competitive eIF4A3 inhibitors
Keywords: روابط فعالیت ساختاری; RNA helicase; Eukaryotic initiation factor 4A3 (eIF4A3) inhibitors; Exon junction complex (EJC); ATP-competitive type inhibitors; Isothermal titration calorimetry (ITC); Surface plasmon resonance (SPR); BRR2; bad response to refrigeration 2 (an ATP-depend
Design and synthesis of purine analogues as highly specific ligands for FcyB, a ubiquitous fungal nucleobase transporter
Keywords: روابط فعالیت ساختاری; Aspergillus nidulans; Purine transporters; Structure activity relationships; Combiglide; Imidazo[4,5-c]pyridine; Deazaadenine;
Design, synthesis, characterization, cytotoxic and structure activity relationships of novel Ru(II) complexes
Keywords: روابط فعالیت ساختاری; Cytotoxic; Ligand; Ruthenium compounds; Structure activity relationships
Small molecule Mcl-1 inhibitors for the treatment of cancer
Keywords: روابط فعالیت ساختاری; Mcl-1; Myeloid cell leukemia-1; Inhibitors; Small molecule; BH3-mimetic; Bad; Bcl-2-associated death promoter; Bak; Bcl-2 homologous antagonist/killer; Bax; Bcl-2 associated X; Bcl-2; B-cell lymphoma-2; BH; Bcl-2 homology; BH3; Bcl-2 homology domain 3; Bc
Structural basis for cooperative binding of azoles to CYP2E1 as interpreted through guided molecular dynamics simulations
Keywords: روابط فعالیت ساختاری; Cytochrome P450; Allostery; Azole; Molecular dynamics; Docking; Structure activity relationships
Design and synthesis of marine natural product-based 1H-indole-2,3-dione scaffold as a new antifouling/antibacterial agent against fouling bacteria
Keywords: روابط فعالیت ساختاری; Biofilm; Biofouling; Secondary metabolites; Isatin; Marine natural products; Structure activity relationships
Structure-based efforts to optimize a non-β-lactam inhibitor of AmpC β-lactamase
Keywords: روابط فعالیت ساختاری; DMSO; dimethylsulfoxide; DMF; dimethylformamide; NMP; N-methylpyrrolidone; SAR; structure activity relationships; Antibiotic resistance; Structure-based drug design; X-ray crystallography;
Endothelin-1 and -2: Two amino acids matter
Keywords: روابط فعالیت ساختاری; Endothelin; Rat resistance arteries; Agonist-dependence; Allosteric modulation of receptor function; Structure activity relationships;
Bis-chalcone analogues as potent NO production inhibitors and as cytotoxic agents
Keywords: روابط فعالیت ساختاری; Bis-chalcones; Cytotoxicity; NO production inhibition; Structure activity relationships
First synthesis and anticancer activity of novel naphthoquinone amides
Keywords: روابط فعالیت ساختاری; Anticancer activity; Cancer; Naphthoquinone amides; Structure activity relationships; Topoisomerase II
Anti-diabetic effects of sodium 4-amino-2,6-dipicolinatodioxovanadium(V) dihydrate in streptozotocin-induced diabetic rats
Keywords: روابط فعالیت ساختاری; Vanadium(V); Substituted dipicolinatooxovanadium(V) complex; Anti-diabetic effects; Streptozotocin-induced diabetic rats; Blood glucose lowering; Blood lipid lowering; Structure activity relationships
Synthesis, in vivo and in vitro biological activity of novel azaline B analogs
Keywords: روابط فعالیت ساختاری; GnRH antagonists; Structure activity relationships; Azaline B; Degarelix
An α, β-unsaturated oxime identified as a strong contact allergen
Keywords: روابط فعالیت ساختاری; Allergic contact dermatitis; Guinea pigs; Metabolism; Mice; Sensitization; Structure activity relationships;