Keywords: تیمیدین فسفوریزاس; Anticancer activity; Apoptosis; DNA repair; Glioblastoma; Seaweed compounds; Temozolomide; AIC; 5-aminoimidazole-4-carboxamide; Akt; Protein kinase B (PKB); AP site; apurinic/apyrimidinic site; AP-1; activator protein-1; APE-1; AP endonuclease; Bax; Bcl-2
مقالات ISI تیمیدین فسفوریزاس (ترجمه نشده)
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Keywords: تیمیدین فسفوریزاس; 1,3,4-oxadiazole-2-thione; Anticancer activity; Docking; Thymidine phosphorylase; MCF-7;
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Thymidine catabolism; Angiogenesis; 2-deoxy-d-ribose; ROS; NF-κB; 5-FU; Capecitabine; TFTD; 2-deoxy-d-ribose-5-phosphate aldolase; Glycolytic pathway;
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Platelets; Thrombosis; Cancer;
Keywords: تیمیدین فسفوریزاس; Liposomes; Excimer; Thymidine phosphorylase; Surface charge; Quenching; Langmuir isotherms;
Keywords: تیمیدین فسفوریزاس; Predictive biomarkers; Pathology response; Esophageal cancer; Chemo(radio)therapy; Meta-analysis; ESCC; Esophageal squamous cell carcinoma; AC; Adenocarcinoma; TS; Thymidylate synthase; Bax; Bcl-2-associated X protein; Bcl-2; B-cell lymphoma 2; CYFRA21-1;
Keywords: تیمیدین فسفوریزاس; ACSL; Acyl-CoA synthetases; ANOVA; analysis of variance; CHP; cumene hydroperoxide; CPT1; carnitine palmitoyltransferase 1; CRAT; carnitine acetyltransferase; DHB; 2,5-dihydroxybenzoic acid; FABP; fatty acid binding protein; FCCP; carbonyl cyanide-4-(trif
Keywords: تیمیدین فسفوریزاس; Ab; antibody; ACT; adoptive cell therapy; ANG; angiopoietin; ATP; adenosine triphosphate; BMDC; bone marrow derived cell; CA4P; combretastatin A phosphate; CAF; cancer-associated fibroblast; CCL2; C-C motif ligand 2; CD; cluster differentiation antigen; C
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Angiogenesis; Cancer therapy; Enzyme inhibition; Non-nucleobase inhibitors;
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Oxadiazole-2-thione; Molecular modeling; Anti-cancer
Keywords: تیمیدین فسفوریزاس; TAM; tumor-associated macrophage; HR; hormone receptor; ER; estrogen receptor; PR; progesterone receptor; HER2; human epidermal growth factor receptor 2; VEGF; vascular endothelial growth factor; EGFR; epidermal growth factor receptor; HIF; hypoxia-induci
Synthesis and molecular docking study of piperazine derivatives as potent inhibitor of thymidine phosphorylase
Keywords: تیمیدین فسفوریزاس; Synthesis; Piperazine; Thymidine phosphorylase; Molecular docking; SAR;
Synthesis, molecular docking study and in vitro thymidine phosphorylase inhibitory potential of oxadiazole derivatives
Keywords: تیمیدین فسفوریزاس; Synthesis; Oxadiazole; Thymidine phosphorylase; Molecular docking; SAR;
Fluorescence and computational studies of thymidine phosphorylase affinity toward lipidated 5-FU derivatives
Keywords: تیمیدین فسفوریزاس; Spectroscopy; Fluorescence; Liposomes; Dissociation constants; Thymidine phosphorylase; Binding;
Design, synthesis, in-vitro thymidine phosphorylase inhibition, in-vivo antiangiogenic and in-silico studies of C-6 substituted dihydropyrimidines
Keywords: تیمیدین فسفوریزاس; Dihydropyrimine-2-ones; Thymidine phosphorylase; Chorioallantoic membrane assay; Antiangiogenesis;
Single-nucleotide polymorphisms in the genes of CES2, CDA and enzymatic activity of CDA for prediction of the efficacy of capecitabine-containing chemotherapy in patients with metastatic breast cancer
Keywords: تیمیدین فسفوریزاس; 5â²DFCR; 5â²deoxy-5-fluorocytidine; 5â²DFUR; 5â²-deoxy-5-fluorouridine; 5-FU; 5-fluorouracil; AEs; adverse events; AML; acute promyelocytic leukemia; AU; arbitrary unit; CDA; cytidine deaminase; CES; carboxylesterase; DPD; dihydropyrimidine dehydrogen
A phase II trial of carboplatin plus S-1 for elderly patients with advanced non-small-cell lung cancer with wild-type epidermal growth factor receptor: The Okayama Lung Cancer Study Group Trial 1202
Keywords: تیمیدین فسفوریزاس; Carboplatin; Elderly; Non-small cell lung cancer; S-1; Thymidine phosphorylase;
Capillary electrophoresis with online stacking in combination with AgNPs@MCM-41 reinforced hollow fiber solid-liquid phase microextraction for quantitative analysis of Capecitabine and its main metabolite 5-Fluorouracil in plasma samples isolated from can
Keywords: تیمیدین فسفوریزاس; AgNPs; Ag nanoparticles; CAP; Capecitabine; 5-FU; 5-Fluorouracil; TP; Thymidine phosphorylase; CE; Capillary electrophoresis; 5-FUH2; Dihydro-5-fluorouracil; FBAL; α-Fluoro-β-alanine; FUPA; 5-Fluoro-ureido-propionic acid; FLC; Fluoropyrimidine carbamate
Molecular Biomarker Study in a Randomised Phase III Trial of Irinotecan Plus S-1 versus S-1 for Advanced Gastric Cancer (GC0301/TOP-002)
Keywords: تیمیدین فسفوریزاس; Excision repair cross-complementing gene 1; gastric cancer; irinotecan; predictive factor; thymidine phosphorylase; thymidylate synthase;
Intratumoral gene expression of 5-fluorouracil pharmacokinetics-related enzymes in stage I and II non-small cell lung cancer patients treated with uracil-tegafur after surgery: A prospective multi-institutional study in Japan
Keywords: تیمیدین فسفوریزاس; Uracil-tegafur; Non-small cell lung cancer; Adjuvant chemotherapy; Biomarker; Thymidylate synthase; Dihydropyrimidine dehydrogenase; Orotate phosphoribosyltransferase; Thymidine phosphorylase
Enzymatic synthesis and RNA interference of nucleosides incorporating stable isotopes into a base moiety
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Nucleoside synthesis; Nucleosides incorporating stable isotopes; 13C NMR; RNA interference
How do changes in the mtDNA and mitochondrial dysfunction influence cancer and cancer therapy? Challenges, opportunities and models
Keywords: تیمیدین فسفوریزاس; ATP; adenosine triphosphate; OXPHOS; oxidative phosphorylation system; mtDNA; mitochondrial DNA; ECT; electron transport chain; nDNA; nuclear DNA; ROS; reactive oxygen species; SODs; superoxide dismutases; MnSOD; manganese superoxide dismutase; GSH; gluta
Targeting miR-21 enhances the sensitivity of human colon cancer HT-29 cells to chemoradiotherapy in vitro
Keywords: تیمیدین فسفوریزاس; CRC; colorectal cancer; qRT-PCR; quantitative real time polymerase chain reaction; TS; thymidylate synthase; TP; thymidine phosphorylase; DPD; dihydropyrimidine dehydrogenase; MMR; mismatch repair system; UTR; untranslated regions; NC; nonsense control; m
Validation of a HPLC method for the measurement of erythrocyte encapsulated thymidine phosphorylase (EE-TP) activity
Keywords: تیمیدین فسفوریزاس; HPLC; Thymidine phosphorylase; Erythrocyte encapsulated thymidine phosphorylase; Validation; MNGIE;
Making Capecitabine Targeted Therapy for Breast Cancer: Which is the Role of Thymidine Phosphorylase?
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Capecitabine; Predictive factor; Prognostic marker; Immunohistochemistry
The development and validation of an immunoassay for the measurement of anti-thymidine phosphorylase antibodies in mouse and dog sera
Keywords: تیمیدین فسفوریزاس; Anti-TP; anti-thymidine phosphorylase; CF; correction factor; CV; coefficient of variation; ECL; electrochemiluminescent; EE-TP; erythrocyte encapsulated thymidine phosphorylase; EMA; European Medicines Agency; FDA; Food and Drug Administration; GLP; Good
Synthesis of pyrazolo[1,5-a][1,3,5]triazine derivatives as inhibitors of thymidine phosphorylase
Keywords: تیمیدین فسفوریزاس; Pyrazolo[1,5-a][1,3,5]triazines; Thymidine phosphorylase; Enzyme inhibitor
The effect of chemotherapy or radiotherapy on thymidine phosphorylase and dihydropyrimidine dehydrogenase expression in cancer of the uterine cervix
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Dihydropyrimidine dehydrogenase; Uterine cervical cancer; Chemotherapy; Radiotherapy
Prognostic value of TP/PD-ECGF and thrombocytosis in gastric carcinoma
Keywords: تیمیدین فسفوریزاس; Gastric carcinoma; Thymidine phosphorylase; Platelet-derived endothelial cell growth factor; Thrombocytosis; Prognosis;
CoQ10 deficiencies and MNGIE: Two treatable mitochondrial disorders
Keywords: تیمیدین فسفوریزاس; Coenzyme Q; Mitochondria; Mitochondrial DNA; MNGIE; Thymidine phosphorylase; Ubiquinone
Inhibition of thymidine phosphorylase expression by using an HSP90 inhibitor potentiates the cytotoxic effect of cisplatin in non-small-cell lung cancer cells
Keywords: تیمیدین فسفوریزاس; HSP90; Thymidine phosphorylase; Cytotoxicity; Non-small cell lung cancer;
Mitochondrial neurogastrointestinal encephalopathy in an Indian family with possible manifesting carriers of heterozygous TYMP mutation
Keywords: تیمیدین فسفوریزاس; Mitochondrial neurogastrointestinal encephalomyopathy; MNGIE; Thymidine phosphorylase
Structure-activity relationship of 2,4,5-trioxoimidazolidines as inhibitors of thymidine phosphorylase
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Trioxoimidazolidine; Parabanic acid; Hydantoin; Anti-angiogenic; Molecular modelling;
Opposite effects of HIF-1α and HIF-2α on the regulation of IL-8 expression in endothelial cells
Keywords: تیمیدین فسفوریزاس; AdHIF-1α/AdHIF-2α; adenoviral vectors containing HIF-1α or HIF-2α cDNA, respectively; ARE; antioxidant-response element; ARNT; aryl hydrocarbon receptor nuclear translocator; GFP; green fluorescent protein; HIF; hypoxia-inducible factor; HO-1; heme ox
Modulation of Rad51, ERCC1, and thymidine phosphorylase by emodin result in synergistic cytotoxic effect in combination with capecitabine
Keywords: تیمیدین فسفوریزاس; ERCC1; Rad51; Thymidine phosphorylase; Capecitabine; Emodin; ERK1/2; Cytotoxicity; Non-small cell lung cancer
The cytostatic activity of NUC-3073, a phosphoramidate prodrug of 5-fluoro-2′-deoxyuridine, is independent of activation by thymidine kinase and insensitive to degradation by phosphorolytic enzymes
Keywords: تیمیدین فسفوریزاس; Nucleoside analogues; Cancer; Phosphoramidate prodrugs; Mycoplasma; Thymidine phosphorylase; 5-Fluoro-2′-deoxyuridine (5-FdUrd)
The role of phosphate in the action of thymidine phosphorylase inhibitors: Implications for the catalytic mechanism
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Transition state analog; Enzyme mechanism; Inhibition kinetics
Structural diversity of nucleoside phosphonic acids as a key factor in the discovery of potent inhibitors of rat T-cell lymphoma thymidine phosphorylase
Keywords: تیمیدین فسفوریزاس; Phosphonate; Pyrrolidine; Nucleotide analogues; Thymidine phosphorylase; Rat T-cell lymphomas
In vitro and in vivo evaluations of a radioiodinated thymidine phosphorylase inhibitor as a tumor diagnostic agent for angiogenic enzyme imaging
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Angiogenic enzyme imaging; [125I]IIMU
Amplification of thymidylate synthetase in metastatic colorectal cancer patients pretreated with 5-fluorouracil-based chemotherapy
Keywords: تیمیدین فسفوریزاس; Colorectal neoplasms; Neoplasm metastasis; DNA copy number variation; Fluorouracil; Thymidylate synthase; Thymidine phosphorylase
Regulation by degradation, a cellular defense against deoxyribonucleotide pool imbalances
Keywords: تیمیدین فسفوریزاس; ADA; adenosine deaminase; 5BU; 5-Bromo uracil; AdR; deoxyadenosine; cdN; cytosolic 5â²-deoxynucleotidase; cNI; cytosolic 5â²-nucleotidase I; cNII; cytosolic 5â²-nucleotidase II; cpm; counts per minute; dCK; deoxycytidine kinase; dGK; deoxyguanosine kin
Prognostic impact of thymidine phosphorylase expression in breast cancer - Comparison of microarray and immunohistochemical data
Keywords: تیمیدین فسفوریزاس; Breast cancer; Thymidine phosphorylase; Microarray; Immunohistochemistry; Prognosis;
A novel TYMP mutation in a French Canadian patient with mitochondrial neurogastrointestinal encephalomyopathy
Keywords: تیمیدین فسفوریزاس; Mitochondrial neurogastrointestinal encephalomyopathy; MNGIE; TYMP; Thymidine phosphorylase; Mutation; Intergenomic communication
Characterization of a novel TYMP splice site mutation associated with mitochondrial neurogastrointestinal encephalomyopathy (MNGIE)
Keywords: تیمیدین فسفوریزاس; Mitochondrial neurogastrointestinal encephalomyopathy (MNGIE); Thymidine phosphorylase; TYMP; Mitochondrial DNA
Late-onset MNGIE without peripheral neuropathy due to incomplete loss of thymidine phosphorylase activity
Keywords: تیمیدین فسفوریزاس; MNGIE; Mitochondrial disease; Peripheral neuropathy; Late-onset; Thymidine phosphorylase; TYMP/ECGF1 mutations
Structures of native human thymidine phosphorylase and in complex with 5-iodouracil
Keywords: تیمیدین فسفوریزاس; Thymidine phosphorylase; Crystal structure; Enzyme kinetics; Mutagenesis; 5-Iodouracil;
Use of Pd-catalyzed Suzuki-Miyaura coupling reaction in the rapid synthesis of 5-aryl-6-(phosphonomethoxy)uracils and evaluation of their inhibitory effect towards human thymidine phosphorylase
Keywords: تیمیدین فسفوریزاس; Acyclic nucleoside phosphonates; Suzuki-Miyaura reaction; Thymidine phosphorylase; Human thymidine phosphorylase; SD-lymphoma; Suzuki coupling; Uracil; Pyrimidine;
Radiation-Induced Thymidine Phosphorylase Upregulation in Rectal Cancer Is Mediated by Tumor-Associated Macrophages by Monocyte Chemoattractant Protein-1 From Cancer Cells
Keywords: تیمیدین فسفوریزاس; Radiation; Thymidine phosphorylase; Tumor-associated Macrophages; MCP-1; Rectal cancer;
Syntheses of N3-substituted thymine acyclic nucleoside phosphonates and a comparison of their inhibitory effect towards thymidine phosphorylase
Keywords: تیمیدین فسفوریزاس; Acyclic nucleoside phosphonates; Thymidine phosphorylase; Fluorination; Pyrimidine; Alkylation
Encéphalopathie myoneurogastro-intestinale
Keywords: تیمیدین فسفوریزاس; MNGIE; Substance blanche; IRM; Spectroscopie; Cytopathie mitochondriale; Thymidine phosphorylaseMNGIE; White matter; Magnetic resonance imaging; Spectroscopy; Mitochondrial disease; Thymidine phosphorylase