Keywords: مهارکننده Topoisomerase I; Hydrazones; Cytotoxicity; Topoisomerase I inhibitor; Copper(II) complexes
مقالات ISI مهارکننده Topoisomerase I (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Etirinotecan Pegol (NKTR-102) in Third-line Treatment of Patients With Metastatic or Recurrent Non-Small-cell Lung Cancer: Results of a Phase II Study
Keywords: مهارکننده Topoisomerase I; Pegylation; Refractory NSCLC; Third-line therapy; Topoisomerase I inhibitor;
Formyl phloroglucinol meroterpenoids from Eucalyptus tereticornis and their bioactivities
Keywords: مهارکننده Topoisomerase I; Eucalyptus tereticornis; Formyl phloroglucinol meroterpenoids; Cytotoxicity; Topoisomerase I inhibitor;
Allosteric inhibition of topoisomerase I by pinostrobin: Molecular docking, spectroscopic and topoisomerase I activity studies
Keywords: مهارکننده Topoisomerase I; Topoisomerase I inhibitor; DNA binding; Molecular docking;
The combination of A-966492 and Topotecan for effective radiosensitization on glioblastoma spheroids
Keywords: مهارکننده Topoisomerase I; Glioblastoma; PARP inhibitor; Topoisomerase I inhibitor; Topotecan; Radiosensitivity;
Wide application of a novel topoisomerase I inhibitor-based drug conjugation technology
Keywords: مهارکننده Topoisomerase I; Drug-delivery system; Antibody-drug conjugate; Topoisomerase I inhibitor; Exatecan; Membrane permeability; B7-H3; Oncology; Cancer therapy;
Nanoparticle-mediated delivery of a rapidly activatable prodrug of SN-38 for neuroblastoma therapy
Keywords: مهارکننده Topoisomerase I; Drug delivery; Nanoparticle; Prodrug; Topoisomerase I inhibitor; Neuroblastoma
Novel synthetic acridine derivatives as potent DNA-binding and apoptosis-inducing antitumor agents
Keywords: مهارکننده Topoisomerase I; Acridine derivatives; Antiproliferative activity; DNA-binding; Topoisomerase I inhibitor; Apoptosis;
Synthesis and antitumor activity of 10-arylcamptothecin derivatives
Keywords: مهارکننده Topoisomerase I; Antitumor activity; Camptothecin derivative; Lactone stability; Synthesis; Topoisomerase I inhibitor
Induction of apoptosis in colon cancer cells by a novel topoisomerase I inhibitor TopIn
Keywords: مهارکننده Topoisomerase I; Topoisomerase I inhibitor; p53; Colon cancer; Apoptosis;
Synthesis and biological evaluation of novel 7-acyl homocamptothecins as Topoisomerase I inhibitors
Keywords: مهارکننده Topoisomerase I; Homocamptothecin; Camptothecin; Antitumor activity; Topoisomerase I inhibitor;
3-Arylisoquinolines as novel topoisomerase I inhibitors
Keywords: مهارکننده Topoisomerase I; 3-Arylisoquinoline; Benz[b]oxepine; Camptothecin; Indeno[1,2-c]isoquinoline; Isoindolo[2,1-b]isoquinoline; 12-Oxobenzo[c]phenanthridine; Topoisomerase I inhibitor
Belotecan for relapsing small-cell lung cancer patients initially treated with an irinotecan-containing chemotherapy: A phase II trial
Keywords: مهارکننده Topoisomerase I; Belotecan; SCLC; Topoisomerase I inhibitor;
Downregulated ABCG2 Enhances Sensitivity to Topoisomerase I Inhibitor in Epidermal Growth Factor Receptor Tyrosine Kinase Inhibitor-Resistant Non-small Cell Lung Cancer
Keywords: مهارکننده Topoisomerase I; Non-small cell lung cancer (NSCLC); Epidermal growth factor receptor tyrosine kinase inhibitor (EGFR TKI); Drug resistance; ABCG2; Topoisomerase I inhibitor
Altered phospholipid transfer protein gene expression and serum lipid profile by topotecan
Keywords: مهارکننده Topoisomerase I; Topoisomerase I inhibitor; Camptothecin; Topotecan; Phospholipid transfer protein; High-density lipoprotein; Pancreatitis; Hyperlipidemia; Hypertriglyceridemia;
Review role of topotecan in gynaecological cancers: Current indications and perspectives
Keywords: مهارکننده Topoisomerase I; Chemotherapy; Cervical cancer; Ovarian cancer; Topotecan; Topoisomerase I inhibitor
Synthesis of new camptothecin analogs with improved antitumor activities
Keywords: مهارکننده Topoisomerase I; Anticancer agent; Camptothecin analog; Topoisomerase I inhibitor; BCRP
Oxiranylmethyloxy or thiiranylmethyloxy-azaxanthones and -acridone analogues as potential topoisomerase I inhibitors
Keywords: مهارکننده Topoisomerase I; Azaxanthone; Acridone; Topoisomerase I inhibitor; Anticancer agents
Synthesis and biological activities of a pH-dependently activated water-soluble prodrug of a novel hexacyclic camptothecin analog
Keywords: مهارکننده Topoisomerase I; Camptothecin analog; Topoisomerase I inhibitor; TP300, Antitumor agent; Water-soluble; Prodrug; Drug resistance; BCRP
Apoptotic effect of CKD-602 (Camtobell®) on oral squamous cell carcinoma cell lines
Keywords: مهارکننده Topoisomerase I; Oral squamous cell carcinoma; CKD-602; Topoisomerase I inhibitor; Apoptosis; Camptothecin;
XMT-1001, a novel polymeric camptothecin pro-drug in clinical development for patients with advanced cancer
Keywords: مهارکننده Topoisomerase I; Polymer; Camptothecin; Topoisomerase I inhibitor; Drug delivery; Dual phase release; Nanotechnology
The contribution of plukenetione A to the anti-tumoral activity of Cuban propolis
Keywords: مهارکننده Topoisomerase I; Propolis; Plukenetione A; Anti-tumoral activity; Topoisomerase I inhibitor; DNA polymerase inhibitor
In vitro cytotoxicity against different human cancer cell lines of laticifer proteins of Calotropis procera (Ait.) R. Br
Keywords: مهارکننده Topoisomerase I; LP, (laticifer proteins); PBMC, (peripheral blood mononuclear cells)Apoptosis; Cytotoxic activity; Latex; Topoisomerase I inhibitor
Synthesis of benz[d]indeno[1,2-b]pyran-5,11-diones: Versatile intermediates for the design and synthesis of topoisomerase I inhibitors
Keywords: مهارکننده Topoisomerase I; Indenoisoquinoline; Topoisomerase I inhibitor; Synthesis; Anticancer
Evaluation of indenoisoquinoline topoisomerase I inhibitors using a hollow fiber assay
Keywords: مهارکننده Topoisomerase I; Indenoisoquinoline; Topoisomerase I inhibitor; Anticancer; Hollow fiber assay
A phase II trial with RFS2000 (rubitecan) in patients with advanced non-small cell lung cancer
Keywords: مهارکننده Topoisomerase I; Rubitecan; RFS2000; Non-small cell lung cancer; Topoisomerase I inhibitor;
Single-Agent Topotecan as First-Line Chemotherapy in Women with Metastatic Breast Cancer: Final Results of Eastern Cooperative Oncology Group Trial E8193
Keywords: مهارکننده Topoisomerase I; Camptothecin analogues; Hematopoietic toxicity; Topoisomerase I inhibitor;