Keywords: مهار رشد کل; Oxindole; Knoevenagel reaction; Antiproliferative activity; NADPH oxidase 4; Tubulin assembly; DTP; Developmental Therapeutics Program; NCI; National Cancer Institute; CSA4; combretastatin A-4; Nox; NAD(P)H oxidase enzyme; ROS; reactive oxygen species; EC
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Quinazoline based α1-adrenoreceptor antagonists with potent antiproliferative activity in human prostate cancer cell lines
Keywords: مهار رشد کل; Quinazoline; Quinone; α1-Adrenoreceptor antagonist; DNA fragmentation; Antiproliferative activity; α1-AR; α1-adrenoreceptor; BPH; benign prostatic hyperplasia; CHO; Chinese hamster ovary; Dox; doxazosin; GSH; glutathione; LUTS; lower urinary tract symp
Synthesis and evaluation of 5-(arylthio)-9H-pyrimido[4,5-b]indole-2,4-diamines as receptor tyrosine kinase and thymidylate synthase inhibitors and as antitumor agents
Keywords: مهار رشد کل; Multiple receptor tyrosine kinase inhibitors; Antiangiogenic agents; Pyrimido[4,5-b]indole synthesis; Thymidylate synthase inhibitors; Combination chemotherapeutic potential in single agents; RTK; receptor tyrosine kinases; VEGF; vascular endothelial grow
Synthesis, anti-proliferative activity, SAR study, and preliminary in vivo toxicity study of substituted N,Nâ²-bis(arylmethyl)benzimidazolium salts against a panel of non-small cell lung cancer cell lines
Keywords: مهار رشد کل; NCI; National Cancer Institute; IC50; inhibitory concentration 50%; NSCLC; non-small cell lung cancer; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; SAR; structure-activity relationship; GI50; growth inhibition 50%; TGI; total growth
Synthesis, in vitro antitumor activity, dihydrofolate reductase inhibition, DNA intercalation and structure-activity relationship studies of 1,3,5-triazine analogues
Keywords: مهار رشد کل; DHFR; dihydrofolate reductase; ct-DNA; calf thymus DNA; NADPH; nicotinamide adenine dinucleotide phosphate; TGI; total growth inhibition; LC50; 50% lethal concentration; GI50; 50% growth inhibition; IC50; 50% inhibitory concentration; Ka; binding constant
Different cell death responses induced by eupomatenoid-5 in MCF-7 and 786-0 tumor cell lines
Keywords: مهار رشد کل; 786-0; human kidney cancer cell line; 7-AAD; 7-aminoactinomycin D; ATP; adenosine triphosphate; DCE; dichloromethanic crude extract; DCF; 2,7-dichlorofluorescein; DCFH; 2,7-dichlorodihydrofluorescein; DCFH-DA; dichlorofluorescin diacetate; DMSO; dimethyl
From arrow poison to herbal medicine - The ethnobotanical, phytochemical and pharmacological significance of Cissampelos (Menispermaceae)
Keywords: مهار رشد کل; Ig; immunoglobulin; OVA; ovalbumin; PG; prostaglandin; PHF; polyherbal formulation; TGI; total growth inhibition; MIC; minimum inhibitory concentration; IZD; inhibition zone diameter; MLE; methanolic leaf extract; HLE; hydroalcoholic leaf extract; HRE; hy