Keywords: Endocrine disruptors; Madrid; Tap water; Bioassays; Chemical monitoring; Transactivation assay; ED; Endocrine disruptor; PAH; Polycyclic aromatic hydrocarbon; PCB; Polychlorinated biphenyl; TH; Thyroid hormone; T3; Triiodothyronine; T4; Thyroxine; EDC; En
مقالات ISI (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Importance of 5/6-aryl substitution on the pharmacological profile of 4ʹ-((2-propyl-1H-benzo[d]imidazol-1-yl)methyl)-[1,1ʹ-biphenyl]-2-carboxylic acid derived PPARγ agonists
Keywords: Peroxisome proliferator-activated receptor γ; Pharmacological profile; Coactivator recruitment; Transactivation assay; Molecular modeling; H; helix; LBD; ligand binding domain; PDB; Protein Data Bank; PPAR; peroxisome proliferator-activated receptor; PPR
Synthesis, in vitro evaluation, and molecular modeling investigation of benzenesulfonimide peroxisome proliferator-activated receptors α antagonists
Keywords: PPARs; PPAR antagonist; Transactivation assay; Benzenesulfonimides; CPT1A; Fibrates; Docking; Molecular dynamic
Utility of an appropriate reporter assay: Heliotrine interferes with GAL4/upstream activation sequence-driven reporter gene systems
Keywords: Firefly luciferase inhibition; Nuclear receptor; Transactivation assay; LBD; ligand-binding domain; DBD; DNA-binding domain; UAS; upstream activating sequence; PXR; pregnane X receptor; mRNA; messenger RNA;
Synthesis and structure-activity relationships of fibrate-based analogues inside PPARs
Keywords: PPARs; Transactivation assay; Fibrates; Chalcone; Stilbene; Gene expression;
Fibrate-derived N-(methylsulfonyl)amides with antagonistic properties on PPARα
Keywords: PPARs; PPAR antagonist; Transactivation assay; FRET
Detection of potential (anti)progestagenic endocrine disruptors using a recombinant human progesterone receptor binding and transactivation assay
Keywords: Progesterone receptor; Endocrine disruptor; Competitive binding; Transactivation assay
Identification of the minimal promoter region of the mouse NKX5-3, a transcription factor implicated in eye development
Keywords: EMSA; electrophoretic mobility shift assay; cDNA; DNA complementary to RNA; PCR; polymerase chain reaction; DMEM; Dulbecco's modified Eagle's medium; PBS; phosphate-buffered saline; AP-2; activator protein 2; Sp1; specificity protein 1; SV40; simian virus
Screening for estrogenicity and anti-estrogenicity: a critical evaluation of an MVLN cell-based transactivation assay
Keywords: Screening for (anti)-estrogenicity; Transactivation assay; MVLN cells; Receptor binding;