Third generation of matrix metalloprotease inhibitors: Gain in selectivity by targeting the depth of the S1â² cavity
Keywords: روی پروتئاز; MMPs; Zinc protease; Selective inhibitors; S1â² loop conformational variability; P1, P2, P3 and P1â², P2â², P3â²; designate inhibitor (or substrate) residues amino-terminal and carboxy-terminal of the scissile bond respectively; S1, S2, S3 and S1â²,