Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; Cape, capecitabine; DFCR, 5′-deoxy-5-fluorocytidine; DFUR, 5′-deoxy-5-fluorouridine; EMA, European Medicines Agency; FDA, Food and Drug Administration; HQC, high quality control; IS, internal standard; LLOQ, lower limit of quantifica
مقالات ISI 5-FU، 5-fluorouracil (ترجمه نشده)
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Keywords: 5-FU، 5-fluorouracil; Oxaliplatin; Chemotherapy; Cognition; Rat; Peripheral neuropathy; Mechanical allodyniaCNS, Central nervous system; OX, Oxaliplatin; NOR, Novel object recognition; NLR, Novel location recognition; 5-FU, 5-fluorouracil
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; ara-C, cytosine arabinoside; AUC, area under the curve, chol, cholesterol; CLA, conjugated linoleic acid; BLI, bioluminescence imaging; dCK, deoxycitydine kinase; dCK, deoxycitydine kinase; dFdU, difluorodeoxyuridine; DNA, deoxyribon
Keywords: 5-FU، 5-fluorouracil; AT, ambient temperature; BSA, bovine serum albumin; CRC, colorectal cancer; DMEM, Dulbecco’s modified Eagle’s medium; EMT, epithelial-mesenchymal transition; FBS, fetal bovine serum; IKK, IκB kinase; 5-FU, 5-Fluorouracil; MMP, matrix metalloproteinase; MT
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; CRC, colorectal cancer; TS, thymidylate synthase; TSER, thymidylate synthase enhancer region; MTHFR, methylenetetrahydrofolate reductase; RFC1, reduced folate carrier 1; OS, overall survival; RFS, relapse-free survival; HR, hazard ra
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; APR, abdominoperineal resection; CA19-9, carbohydrate antigen 19-9; CCK-8, cell counting kit-8; CEA, carcinoembryonic antigen; CI, confidence interval; DCF, 2′, 7′-dichlorofluorescein; DCFH-DA, 2′,7′-dichlorofluorescein diacetate; DF
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; 5-HT, serotonergic; E2, 17β-estradiol; ACTH, adrenocorticotropic hormone; AMY, amygdala; ANS, autonomic nervous system; AP, action potential; AR, androgen receptors; ARC, arcuate nucleus; AVP, arginine vasopressin; AVPV, anterolatera
Keywords: 5-FU، 5-fluorouracil; AKT, protein kinase B; AM, acetoxymethyl ester; ATF6, activating transcription factor 6; CHOP, C/EBP homologous protein; eIF2, eukaryotic initiation factor 2; ER, endoplasmic reticulum; ERK, extracellular signal-regulated kinase; 5-FU, 5-fluorouracil; GRP
Keywords: 5-FU، 5-fluorouracil; CDHP, 5 chloro-2,4-dihydroxypyridine; 5-FU, 5-fluorouracil; %RET, percentage of reticulocytes; FITC, fluorescein isothiocyanate; GEM, gemcitabine; GPI, glycosylphosphatidylinositol; MF, mutant frequency; Oxo, monopotassium 1,2,3,4-tetrahydro-2,4-dioxo-1,3
Wheat bran arabinoxylan supplementation alleviates 5-fluorouracil induced mucositis and myelosuppression in BALB/c mice
Keywords: 5-FU، 5-fluorouracil; AX, rabinoxylan; 5-FU, 5-fluorouracil; PCNA, proliferating cell nuclear antigenArabinoxylan; Mucositis; Myelosuppression; 5-fluorouracil; Chemotherapy5-fluouracil (PubChem CID: 3385); Chloroform (PubChem CID: 6212); Diethylpyrocarbonate (PubChem CID: 3051
Macrophages induce resistance to 5-fluorouracil chemotherapy in colorectal cancer through the release of putrescine
Keywords: 5-FU، 5-fluorouracil; Colorectal cancer; Chemoresistance; Macrophage; Putrescine; ApoptosisTAM, tumor associated macrophage; 5-FU, 5-fluorouracil; CRC, colorectal cancer; ODC, ornithine decarboxylase; DMEM, Dulbecco modified Eagle's medium; FACS, fluorescence-activated cell so
pH and redox-operated nanovalve for size-selective cargo delivery on hollow mesoporous silica spheres
Keywords: 5-FU، 5-fluorouracil; β-CD, β-cyclodextrins; HMSs, hollow mesoporous silica nanoparticles; Fc, ferrocenyl moiety; NHS, N-hydroxysuccinimide; EDC, 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide-HCl; R6G, Rhodamine 6G; DOX, doxorubicin hydrochloride; 5-FU, 5-fluorouracil; MSNs, m
Lipopolysaccharide supports maintaining the stemness of CD133+ hepatoma cells through activation of the NF-κB/HIF-1α pathway
Keywords: 5-FU، 5-fluorouracil; HCC, hepatocellular carcinoma; CSCs, cancer stem cells; TICs, tumor initiating cells; LPS, lipopolysaccharide; EMT, epithelial–mesenchymal transition; FBS, fetal bovine serum; 5-Fu, 5-fluorouracil; TLR4, toll-like receptor 4; PAMPs, pathogen-associated mo
Silencing of CD59 enhanced the sensitivity of HT29 cells to 5-Fluorouracil and Oxaliplatin
Keywords: 5-FU، 5-fluorouracil; CD55; CD59; 5-Fluorouracil; Oxaliplatin; HT-29; Chemotherapy sensitivitymCRPs, membrane complement regulatory proteins; 5-FU, 5-Fluorouracil; SiRNA, small interfering RNA; MCP, membrane cofactor protein (CD46); MAC, membrane attack complex; DAF, decay-acc
Autophagy contributes to the enrichment and survival of colorectal cancer stem cells under oxaliplatin treatment
Keywords: 5-FU، 5-fluorouracil; Colorectal cancer; Autophagy; Cancer stem cells; ChemoresistanceCRC, colorectal cancer; CSCs, cancer stem cells; 5-FU, 5-fluorouracil; OXA, oxaliplatin; H/S, hypoxia/starvation environment; 3-MA, 3-methyladenine; CQ, chloroquine
Anti-proliferative activity of 2,6-dichloro-9- or 7-(ethoxycarbonylmethyl)-9H- or 7H-purines against several human solid tumour cell lines
Keywords: 5-FU، 5-fluorouracil; Anti-tumour compounds; Apoptosis; 5-Fluorouracil; Breast cancer; Colon cancer; Melanoma; PurinesDCA, Dichloroacetate; FACS, Flow cytometry; 5-FU, 5-Fluorouracil; MW, Microwave; SRB, Sulforhodamine-B
Orai1 and STIM1 mediate SOCE and contribute to apoptotic resistance of pancreatic adenocarcinoma
Keywords: 5-FU، 5-fluorouracil; PDAC, pancreatic ductal adenocarcinoma; SOCE, store operated calcium entry; SOCs, store-operated calcium channels; STIM1, stromal interaction molecule 1; 5-FU, 5-Fluorouracil; TG, thapsigargin; SERCA, sarco/endoplasmic reticulum Ca2 + ATPase; siRNA, small
Prognostic advantage of irinotecan dose escalation according to uridine diphosphate glucuronosyltransferase 1A1 (UGT1A1) genotyping in patients with metastatic colorectal cancer treated with bevacizumab combined with 5-fluorouracil/leucovorin with irinote
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; AE, adverse event; CRC, colorectal cancer; FOLFIRI, 5-fluorouracil/leucovorin with irinotecan; IV, intravenous; LV, leucovorin; mCRC, metastatic colorectal cancer; OS, overall survival; PCR, polymerase chain reaction; PFS, progressio
Synthesis and in vitro evaluation of bile acid prodrugs of floxuridine to target the liver
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; Boc2O, di-tert-butyl dicarbonate; CDCA, chenodeoxycholic acid; DCC, N,N′-dicyclohexylcarbodiimide; DCM, dichloromethane; DMAP, 4-dimethylaminopyridine; DMEM, Dulbecco’s modified Eagle medium; DMF, dimethyl formamide; DMSO, dimethyl s
γ-H2AX as a biomarker for DNA double-strand breaks in ecotoxicology
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; 53BP1, p53 binding protein 1; API, aphidicolin; ARA-C, cytarabine; ATM, ataxia telangiectasia mutated; ATR, ataxia telangiectasia related; BLAP, ß-lapachone; BLM, bleomycin; BRCA1, breast cancer type 1 susceptibility protein; cDDP, c
Synthesis of platinum(II) complexes of isatin thiosemicarbazones derivatives: In vitro anti-cancer and deoxyribose nucleic acid binding activities
Keywords: 5-FU، 5-fluorouracil; CT DNA, calf-thymus DNA; DMSO, dimethyl sulfoxide; EB, ethidium bromide; 5-FU, 5-fluorouracil; UV–Vis, UV–visible; ROS, reactive oxygen speciesPlatinum(II) complexes; Isatin moiety; Intercalative activity; Anti-proliferative study
Identification of two novel functional p53 responsive elements in the herpes simplex virus-1 genome
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; ChIP, chromatin immunoprecipitation; EMSA, electrophoretic mobility shift assay; FBS, fetal bovine serum; HSV, herpes simplex virus; IE, immediate early; moi, multiplicity of infection; PBS, phosphate buffered saline; RE, responsive
In vitro combinatorial anticancer effects of 5-fluorouracil and curcumin loaded N,O-carboxymethyl chitosan nanoparticles toward colon cancer and in vivo pharmacokinetic studies
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; CUR, curcumin; N,O-CMC, N,O-carboxymethyl chitosan; FT-IR, Fourier transforms Infrared spectroscopy; DDA, degree of deacetylation; kDa, kilo Dalton; Mw, molecular weight; DLS, dynamic light scattering; PBS, phosphate buffered saline;
Ursolic acid induces cell death and modulates autophagy through JNK pathway in apoptosis-resistant colorectal cancer cells
Keywords: 5-FU، 5-fluorouracil; CRC, colorectal carcinoma; 5-FU, 5-fluorouracil; UA, ursolic acid; MSI, microsatellite instability; JNK, c-jun N-terminal kinase; MAPK, mitogen-activated protein kinase; NAC, N-acetyl-l-cysteine; STS, staurosporine; TUNEL, TdT-mediated dUTP nick end label
Antitumor effect of 5-fluorouracil is enhanced by rosemary extract in both drug sensitive and resistant colon cancer cells
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; CI, combination index; MTT, thiazolyl blue tetrazolium bromide; RT-PCR, real-time polymerase chain reaction; SFRE, supercritical fluid rosemary extract; SW620-5FU-R, human colon cancer SW620 cells resistant to 5-fluorouracil5-Fluorou
Attenuation of nucleoside and anti-cancer nucleoside analog drug uptake in prostate cancer cells by Cimicifuga racemosa extract BNO-1055
Keywords: 5-FU، 5-fluorouracil; BCa, breast cancer; BrdU, 5-bromo-2′-deoxyuridine; CNT, concentrative nucleoside transporter; CR, cimicifuga racemosa; ENT, equilibrative nucleoside transporter; 5-FU, 5-fluorouracil; HPLC, high-pressure liquid chromatography; NBTI, nitrobenzylthioinosine
Interactions between dietary flavonoids apigenin or luteolin and chemotherapeutic drugs to potentiate anti-proliferative effect on human pancreatic cancer cells, in vitro
Keywords: 5-FU، 5-fluorouracil; Api, -apigenin; Cis-, cisplatin; 5-FU, 5-fluorouracil; Gem-, gemcitabine; Oxa, -oxaliplatin; GSK-3β-, glycogen synthase kinase-3β; Lut-, luteolin; MTS, 3-(4,5-dimethylthiazol-2-yl)-5-(3-carboxymethoxyphenyl)-2-(4-sulfophenyl)-2H-tetrazolium; NF-κB, -nucle
Synergistic and individual effects of umbelliferone with 5-fluorouracil on tumor markers and antioxidant status of rat treated with 1,2-dimethylhydrazine
Keywords: 5-FU، 5-fluorouracil; Colon cancer; Complementary medicines; Umbelliferone; 5-fluorouracil; Lipid peroxidationCRC, Colorectal cancer; 5-FU, 5-fluorouracil; UMB, Umbelliferone; CEA, Carcinoembroyonic antigen; CA 19-9, Carbohydrate antigen 19-9; CA 72-4, Carbohydrate antigen 72-
Targeting c-FLIP in cancer
Keywords: 5-FU، 5-fluorouracil; c-FLIP; Death receptors; CancerCDDP, cisplatin; VP16, etoposide; 5-FU, 5-fluorouracil; DISC, death-inducing signaling complex; DcR2, TRAIL-R4 or decoy receptor 2; DR5, TRAIL-R1
Therapeutic Advances in Pancreatic Cancer
Keywords: 5-FU، 5-fluorouracil; Pancreatic Cancer; Chemotherapy; Adjuvant TherapyESPAC, European Study Group for Pancreatic Cancer; 5-FU, 5-fluorouracil; hENT-1, human equilibrative nucleoside transporter 1; LDP, laparoscopic distal pancreatectomy; MDACC, MD Anderson Cancer Center; PDAC
Cancer stem cells: therapeutic implications and perspectives in cancer therapy
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; ABC, ATP-binding cassette; ABCB1, ATP binding cassette superfamily subfamily B member 1; ABCG2, ATP binding cassette superfamily subfamily G member 2; ALDH1, aldehyde dehydrogenase1; AML, acute myeloid leukemia; AMO, anti-miRNA oligo
Overview of the therapeutic potential of piplartine (piperlongumine)
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; AHNAK, neuroblast differentiation-associated protein; ALT, alanine amino transaminase; ANXA5, Annexin A5; AST, aspartate amino transferase; Bcl-2, B-cell leukemia/lymphoma 2; Bim, Bcl-2 interacting mediator of cell death; CBR1, carbo
MBD4 and TDG: Multifaceted DNA glycosylases with ever expanding biological roles
Keywords: 5-FU، 5-fluorouracil; 5-BrU, 5-bromouracil; 5-ClU, 5-chlorouracil; 5-FU, 5-fluorouracil; 5-hmC, 5-hydroxymethylcytosine; 5-hmU, 5-hydroxymethyluracil; 5-IdU, 5-iododeoxyuridine; 5-meC, 5-methylcytosine; A, adenine; AID, activation-induced deaminase; Apc, adenomatous polyposis
Selective sensitization of tumors to chemotherapy by marine-derived lipids: A review
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; CPK, creatine phosphokinase; DHA, docosahexaenoic acid; EPA, eicosapentaenoic acid; FDA, food and drug administration; FEC, 5-fluorouracil epirubicin cyclophosphamide; FOLFIRI, 5-fluorouracil leucovorin irinotecan; FOLFOX, 5-fluorour
Role of the RAD51 G172T polymorphism in the clinical outcome of cervical cancer patients under concomitant chemoradiotherapy
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; RCT, radiochemotherapy; HPV, Human papillomavirus; DSB, double-strand break(s); HR, homologous recombination; NHEJ, non-homologous recombination; kb, kilobase; UTR, untranslated region(s); SNP, single nucleotide polymorphism(s); MAF,
Effects of 5-fluorouracil and gemcitabine on a breast cancer cell line (MCF-7) via the JAK/STAT pathway
Keywords: 5-FU، 5-fluorouracil; ANOVA, analysis of variance; BclxL, B-cell lymphoma-extra large; DSMZ, Deutsche Sammlung von Mikroorganismen und Zellkulturen (German Collection of Microorganisms and Cell Cultures); 5 FdUMP, 5-fluorodeoxyuridine monophosphate; 5-FU, 5-fluorouracil; 5 FUT
Synergistic anticancer effect of rAd/P53 combined with 5-fluorouracil or iodized oil in the early therapeutic response of human colon cancer in vivo
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; wt-p53, wild-type p53; rAd/p53, recombinant adenovirus-mediated p53; IACUC, Institutional Animal Care and Use Committee; HE, hematoxylin and eosin; ECL, enhanced chemiluminescence; KI, Ki-67 index; IOD, integrity optical density; RIO
Development and utilization of a combined LC–UV and LC–MS/MS method for the simultaneous analysis of tegafur and 5-fluorouracil in human plasma to support a phase I clinical study of oral UFT®/leucovorin
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; UFT®, uracil and tegafur; LV, leucovorin (folinic acid); PK, pharmacokinetic; AUC, area under the curve; RT, radiation therapy; HPLC, high performance liquid chromatography; MS/MS, tandem mass spectrometry; UV, ultraviolet spectrosco
Expression and regulation of RAD51 mediate cellular responses to chemotherapeutics
Keywords: 5-FU، 5-fluorouracil; HR, homologous recombination; DSBs, DNA double strand breaks; TS, thymidylate synthase; RTX, raltitrexed (Tomudex™); 5-FU, 5-fluorouracil; FdUrd, fluorodeoxyuridine; UCN-01, 7-Hydroxy-staurosporine; GFP, green fluorescent proteinThymidylate synthase; Homo
EUS or percutaneously guided intratumoral TNFerade biologic with 5-fluorouracil and radiotherapy for first-line treatment of locally advanced pancreatic cancer: a phase I/II study
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; ANC, absolute neutrophil count; CRT, chemoradiation therapy; DLT, dose-limiting toxicity; DVT, deep vein thrombosis; EUS-FNI, EUS-guided fine-needle viral injection; FNI, fine-needle viral injection; LAPC, locally advanced pancreatic
Antitumor activity of Dioscorea bulbifera L. rhizome in vivo
Keywords: 5-FU، 5-fluorouracil; DB, Dioscorea bulbifera L.; fraction A, water extract; fraction B, ethanol extract; fraction C, ethyl acetate extract; fraction D, non-ethyl acetate extract; 5-Fu, 5-Fluorouracil; i.g., intragastric administration; CMC-Na, sodium carboxymethyl cellulose;
Anticancer activity of small amphipathic β2,2-amino acid derivatives
Keywords: 5-FU، 5-fluorouracil; Anticancer peptide; Antimicrobial peptide; Amphipathic scaffold; Beta-amino acid; PeptidomimeticsAMP, cationic antimicrobial peptide; BOC2O, di-tert-butyl dicarbonate; DIPEA, di-isopropyl ethyl amine; 5-FU, 5-fluorouracil; LfcinB, bovine lactoferricin; MB
Up-regulation of FXR isoforms is not required for stimulation of the expression of genes involved in the lack of response of colon cancer to chemotherapy
Keywords: 5-FU، 5-fluorouracil; CDDP, cis-diamminedichloroplatinum(II); CRAC, colorectal adenocarcinoma; 5-FU, 5-fluorouracil; FXR, farnesoid X receptor; MDR, multidrug resistance; MOC, mechanism of chemoresistance; TKI, tyrosine kinase inhibitor; TLDA, Taqman Low-Density ArrayChemoresi
Local control of experimental malignant pancreatic tumors by treatment with a combination of chemotherapy and intratumoral 224Radium-loaded wires releasing alpha-emitting atoms
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; DaRT, diffusing alpha-emitters radiation therapy; DSB, double strand breaks; DMEM, Dulbecco's modified eagle medium; LET, linear energy transfer; OD, optical density; PBS, phosphate-buffered saline; SCC, squamous cell carcinoma; SSB,
Suicide gene therapy in cancer: Where do we stand now?
Keywords: 5-FU، 5-fluorouracil; AMSCs, adipose tissue mesenchymal stromal cells; CD, cytosine deaminase; CSCs, cancer stem cells; DOTAP, 1,2-dioleoyl-3-(trimethylammonium) propane; Chol, cholesterol; 5-FC, 5-fluorocytosine; 5-FU, 5-fluorouracil; GCV, ganciclovir; GvHD, graft-versus-host
ATR–Chk1 signaling pathway and homologous recombinational repair protect cells from 5-fluorouracil cytotoxicity
Keywords: 5-FU، 5-fluorouracil; 5-FU, 5-fluorouracil; FUTP, fluorouridine triphosphate; FdUTP, fluorodeoxyuridine triphosphate; FdUMP, fluorodeoxyuridine monophosphate; TS, thymidylate synthase; BER, base excision repair; MMR, mismatch repair; DSB, double-strand break; HRR, homologous r
Acquisition of chemoresistance in intrahepatic cholangiocarcinoma cells by activation of AKT and extracellular signal-regulated kinase (ERK)1/2
Keywords: 5-FU، 5-fluorouracil; ICC, intrahepatic cholangiocarcinoma; ERK1/2, extracellular signal-regulated kinase 1/2; 5-FU, 5-fluorouracil; MEK, mitogen-activated protein kinase; PI3K, phosphoinocitide 3-kinaseCisplatin; Chemoresistance; Cholangiocarcinoma; AKT; ERK1/2
The achievement of mass balance by simultaneous quantification of floxuridine prodrug, floxuridine, 5-fluorouracil, 5-dihydrouracil, α-fluoro-β-ureidopropionate, α-fluoro-β-alanine using LC–MS
Keywords: 5-FU، 5-fluorouracil; FBAL, α-fluoro-β-alanine; FUPA, α-fluoro-β-ureidopropionate; FUH2, 5-fluorodihydrouracil; 5-FU, 5-fluorouracil; 5-FdUrd, 5-fluoro-2′-deoxyuridineα-Fluoro-β-alanine (FBAL); α-Fluoro-β-ureidopropionate (FUPA); 5-Fluorodihydrouracil (FUH2); 5-Fluorouracil (5
Synthesis and anticancer activity of (RS)-9-(2,3-dihydro-1,4-benzoxaheteroin-2-ylmethyl)-9H-purines
Keywords: 5-FU، 5-fluorouracil; Apoptosis; 1,4-Benzodioxin; 1,4-Benzoxathiin; eIF2α; Purine; Breast cancer cell line MCF-7; Neighboring-group participationMCF-7, Michigan Cancer Foundation; IC50, concentration resulting in 50% inhibition; 5-FU, 5-fluorouracil; SEM, standard error of the
R1 resection for aggressive or advanced colorectal liver metastases is justified in combination with effective prehepatectomy chemotherapy
Keywords: 5-FU، 5-fluorouracil; Colorectal cancer; Liver metastasis; Hepatectomy; R1 resection; SurvivalCA, Carbohydrate antigen; CDDP, Cisplatin; CEA, Carcinoembryonic antigen; CT, Computed tomography; DFR, Disease-free rate; FA, Folinic acid; 5-FU, 5-Fluorouracil; PD, Progressive dise