
Homodimerization of adenosine A1 receptors in brain cortex explains the biphasic effects of caffeine
Keywords: G protein-coupled receptor; Binding parameters; cooperativity; Allosteric interaction; Two-state dimer receptor model; Proximity ligation assayADA, adenosine deaminase; A1R, adenosine A1 receptor; A2AR, adenosine A2A receptor; A2BR, adenosine A2B receptor