Keywords: MG; myasthenia gravis; AChR; nicotinic acetylcholine receptor; ECD; extracellular domain; MIR; main immunogenic region; AChBP; acetylcholine binding protein; α-Btx; α-bungarotoxin.; Nicotinic acetylcholine receptor; Extracellular domain; Myasthenia grav
مقالات ISI (ترجمه نشده)
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Keywords: On-line microfluidics; Nano-liquid chromatography-mass spectrometry (nano-LC-MS); Snake venom proteome screening; Venom purification; Lymnaea stagnalis acetylcholine binding protein (Ls-AChBP); Nicotinic acetylcholine receptor; ACN; acetonitrile; AChB
Keywords: On-line microfluidics; Nano-liquid chromatography-mass spectrometry (nano-LC-MS); Snake venom proteome screening; Venomics; Lymnaea stagnalis acetylcholine binding protein (Ls-AChBP); Nicotinic acetylcholine receptor; AChBP; Acetylcholine binding prot
Neurotoxicity fingerprinting of venoms using on-line microfluidic AChBP profiling
Keywords: Microfluidic HRS; Neurotoxicity fingerprinting; AChBP; α7-nAChR; On-line bioaffinity; Nanolc-MS; Elapid venom profiling;
Stoichiometry dependent inhibition of rat α3β4 nicotinic acetylcholine receptor by the ribbon isomer of α-conotoxin AuIB
Keywords: ACh; acetylcholine; AChBP; acetylcholine-binding protein; ECD; extracellular domain; gAuIB; globular AuIB; ICD; intracellular domain; nAChR; nicotinic acetylcholine receptor; rAuIB; ribbon AuIB; SAR; structure-activity relationship; TMD; transmembrane dom
The binding orientation of epibatidine at α7 nACh receptors
Keywords: Cys-loop; Ion channel; Radioligand; Epibatidine; Agonist; α7 nACh; Nicotinic; Receptor; AChBP; 5-HT; 5-hydroxytryptamine; nACh; nicotinic acetylcholine; GABA; gamma-aminobutyric acid; HEK; human embryonic kidney; AChBP; acetylcholine binding protein; 5HT
Characterization of a reproducible rat EAMG model induced with various human acetylcholine receptor domains
Keywords: MG; myasthenia gravis; AChR; nicotinic acetylcholine receptor; ECD; extracellular domain; MIR; main immunogenic region; AChBP; acetylcholine binding protein; α-Btx; α-bungarotoxin; EAMG; experimental autoimmune myasthenia gravis; EMG; electromyography;
Functional characterization of two prokaryotic pentameric ligand-gated ion channel chimeras - role of the GLIC transmembrane domain in proton sensing
Keywords: 5HT3R; serotonin receptor; α-BTX; α-bungarotoxin; AChBP; acetylcholine-binding protein; ECD; extracellular domain; ELIC; Erwinia ligand-gated ion channel; GLIC; Gloebacter ligand-gated ion channel; GlyR; glycine receptor; nAChR; nicotinic acetylcholine
Assessment of the functionality and stability of detergent purified nAChR from Torpedo using lipidic matrixes and macroscopic electrophysiology
Keywords: nAChR-DCs; nicotinic acetylcholine receptors detergent complexes; Tc; Torpedo californica; Tm; Torpedo marmorata; PLB; planar lipid bilayer; TEVC; two electrode voltage clamp; LCP; Lipidic Cubic Phase; FC; foscholine family 12-16 carbon chain; LFC; lyso
Synthesis and biological activities of indolizine derivatives as alpha-7 nAChR agonists
Keywords: α7 nAChR; Indolizine; Agonists; SAR; Schizophrenia; ACh; acetylcholine; THF; tetrahydrofuran; DMSO; dimethylsulfoxide; CNS; central nervous system; HRMS; high resolution mass; DIPEA; diisopropylethylamine; AChBP; acetylcholine binding protein; SAR; struc
Biomolecular recognition of antagonists by α7 nicotinic acetylcholine receptor: Antagonistic mechanism and structure-activity relationships studies
Keywords: AChBP; acetylcholine binding protein; Ala; alanine; Arg; arginine; ATP; adenosine triphosphate; CNS; central nervous system; CoMFA; comparative molecular field analysis; CoMSIA; comparative molecular similarity indices analysis; Cys; cysteine; 3D-QSAR; th
Exploration of the molecular architecture of the orthosteric binding site in the α4β2 nicotinic acetylcholine receptor with analogs of 3-(dimethylamino)butyl dimethylcarbamate (DMABC) and 1-(pyridin-3-yl)-1,4-diazepane
Keywords: nACh receptor agonists; Structure-activity studies; Ls-AChBP; Ac-AChBP; Lobeline; DMABC analogs; Ac; Aplysia californica; ACh; acetylcholine; AChBP; acetylcholine binding protein; CNS; central nervous system; CDI; 1,1â²-carbonyldiimidazole; Ct; Capitel
The binding characteristics and orientation of a novel radioligand with distinct properties at 5-HT3A and 5-HT3AB receptors
Keywords: Antagonist; Cys-loop; Ion channel; Radioligand; 5-HT3; Agonist; 5-HT; 5-hydroxytryptamine; nACh; nicotinic acetylcholine; GABA; gamma-aminobutyric acid; HEK; human embryonic kidney; AChBP; acetylcholine binding protein; 5HTBP; an AChBP mutant modified to
Pharmacological properties and predicted binding mode of arylmethylene quinuclidine-like derivatives at the α3β4 nicotinic acetylcholine receptor (nAChR)
Keywords: ACHBP; acetylcholine-binding protein; Ach; acetylcholine; CNS; central nervous system; MEC; minimum-effective concentration; nAChR; nicotinic acetylcholine receptor; NIC; nicotine; Pdb; protein databank; rmsd; root-mean-squared-deviation; ROC; receiver op
QM-polarized ligand docking accurately predicts the trend in binding affinity of a series of arylmethylene quinuclidine-like derivatives at the α4β2 and α3β4 nicotinic acetylcholine receptors (nAChRs)
Keywords: ACHBP; acetylcholine-binding protein; Ach; acetylcholine; CNS; central nervous system; MEC; minimum-effective concentration; nAChR; nicotinic acetylcholine receptor; NIC; nicotine; Pdb; protein databank; rmsd; root-mean-squared-deviation; ROC; receiver op
Interactions of acetylcholine binding site residues contributing to nicotinic acetylcholine receptor gating: Role of residues Y93, Y190, K145 and D200
Keywords: ACh; acetylcholine; nAChR; nicotinic acetylcholine receptor; AChBP; acetylcholine binding protein; LBD; ligand binding domain; dTC; d-tubocurarine; DC6C; Dansyl C6 Choline; nAChR; Resting state; Desensitized state; αγ interface; αδ interface; Molecula
Structure-based design, synthesis and structure–activity relationships of dibenzosuberyl- and benzoate-substituted tropines as ligands for acetylcholine-binding protein
Keywords: Fragment-merging; Structure-based design; AChBP; nAChR; Hit-optimization
The pharmacological profile of ELIC, a prokaryotic GABA-gated receptor
Keywords: Cys-loop; Erwinia; Ligand-gated; Antagonist; Nicotinic; ELIC; GLIC; GABA; nACh; nicotinic acetylcholine; AChBP; acetylcholine binding protein; GABA; γ-aminobutyric acid; ELIC; Erwinia ligand-gated ion channel; GLIC; Gloeobacter ligand-gated ion channel;
Discovery of novel α7 nicotinic acetylcholine receptor ligands via pharmacophoric and docking studies of benzylidene anabaseine analogs
Keywords: ACHBP; acetylcholine-binding protein; DMXBA; 3-(2,4-dimethoxybenzilidene)-anabaseine; HBD; hydrogen-bond donor; nAChR; nicotinic acetylcholine receptor; Pdb; protein databank; rmsd; root-mean-squared-deviation; ROC; receiver operating characteristic curve
Identification of novel α7 nicotinic receptor ligands by in silico screening against the crystal structure of a chimeric α7 receptor ligand binding domain
Keywords: α7 Receptor; nAChR; AChBP; Virtual screening; In silico screening; Docking; Cys-loop;
The Haemonchus contortus UNC-49B subunit possesses the residues required for GABA sensitivity in homomeric and heteromeric channels
Keywords: 5-HT3; serotonin (5-hydroxytryptamine)-gated ion channel receptor; AChBP; acetylcholine binding protein; cRNA; copy RNA; LGIC; ligand-gated ion channels; MS-222; 3-aminobenzoic acid ethyl ester, methanesulphonate salt; nAChR; nicotinic acetylcholine recep
Allosteric modulators induce distinct movements at the GABA-binding site interface of the GABA-A receptor
Keywords: GABAA receptor; Benzodiazepine efficacy; Oocyte expression; Allosteric modulation; Pentobarbital; GABA; BZD; benzodiazepine; GABAR; GABA-A receptor; MTSEA-Biotin; N-biotinaminoethyl methanethiosulfonate; MTSES; 2-sulfonatoethyl methanethiosulfonate; DMCM;
Docking studies of benzylidene anabaseine interactions with α7 nicotinic acetylcholine receptor (nAChR) and acetylcholine binding proteins (AChBPs): Application to the design of related α7 selective ligands
Keywords: AChBPs; Nicotinic acetylcholine receptor α7; Docking; Benzylidene-anabaseine analogs; Spirodiazepine and spiroimidazoline quinuclidine series; Ac; Aplysia californica; ACHBP; Acetylcholine-binding protein; AD; Alzheimer's disease; ADHD; Attention defic
Aconitum and Delphinium alkaloids of curare-like activity. QSAR analysis and molecular docking of alkaloids into AChBP
Keywords: Alkaloids; QSAR; Molecular docking; Toxicity; Curare-like activity; nAChR-binders; AChBP
Docking to flexible nicotinic acetylcholine receptors: A validation study using the acetylcholine binding protein
Keywords: Protein flexibility; Molecular docking; Ensemble generation; Nicotinic; Acetylcholine receptors; nAChR; Acetylcholine binding protein; AChBP
A computational study of the binding of 3-(arylidene) anabaseines to two major brain nicotinic acetylcholine receptors and to the acetylcholine binding protein
Keywords: Nicotinic acetylcholine receptor; QSAR; AChBP; Docking; Anabaseine; DMBXA; GTS-21; Benzylidene-anabaseine
Effect of homologous serotonin receptor loop substitutions on the heterologous expression in Pichia of a chimeric acetylcholine-binding protein with α-bungarotoxin-binding activity
Keywords: α-Bungarotoxin; AChBP; Acetylcholine-binding protein; Serotonin receptor; Cys-loop; Ligand-gated ion channels
Design and expression of human α7 nicotinic acetylcholine receptor extracellular domain mutants with enhanced solubility and ligand-binding properties
Keywords: α-bgtx; α-bungarotoxin; α7-dm-ECD; double mutant of the α7-ECD; α7-wt-ECD; wild-type of the α7-ECD; ACh; acetylcholine; AChBP; acetylcholine-binding protein; BSA; bovine serum albumin; CCh; carbamylcholine; CD; circular dichroism; DLS; dynamic light
Docking of 6-chloropyridazin-3-yl derivatives active on nicotinic acetylcholine receptors into molluscan Acetylcholine Binding Protein (AChBP)
Keywords: Docking; 6-Chloropyridazin-3-yl derivatives; AChBP;
Activation of ionotropic receptors and thermodynamics of binding
Keywords: AChBP; acetylcholine binding protein; AMPA; α-amino-3-hydroxy-5-methyl-4-isoxazole; ÎCp; heat capacity change; ÎH; change in enthalpy; ÎS; change in entropy; ÎG; change in free energy; GABAA; A-type γ-aminobutyric acid; MPPB; 1-methyl-5-phenyl-5-pro
A chimera encoding the fusion of an acetylcholine-binding protein to an ion channel is stabilized in a state close to the desensitized form of ligand-gated ion channels
Keywords: AChBP; Acetylcholine; Nicotinic; Receptor; Pentameric ligand-gated ion channel; Allosteric transitions; AChBP; Acétylcholine; Nicotinique; Récepteur; Canal ionique liée à un ligand pentamère; Transitions allostériques;
A model for short α-neurotoxin bound to nicotinic acetylcholine receptor from Torpedo californica: Comparison with long-chain α-neurotoxins and α-conotoxins
Keywords: nAChR; nicotinic acetylcholine receptors; AChBP; acetylcholine-binding protein; MD; molecular dynamics; NTII; α-neurotoxin II; Snake three-fingered short α-neurotoxin; Nicotinic acetylcholine receptor; Toxin-receptor complex; Experimental data based m
The role of inflammation in Alzheimer's disease
Keywords: αBTx; α-bungarotoxin; Aβ; beta-amyloid protein; ACh; acetylcholine; AChBP; acetylcholine-binding protein; AChR; nicotinic acetylcholine receptor; AD; Alzheimer's disease; AICD; amyloid precursor protein intracellular domain; AP; amyloid P; APP; amyloid