دانلود مقالات ISI درباره خواص ADME + ترجمه فارسی

توسعه لیگاند های گیرنده آدنوزین مبتنی بر پیریدیداسیون

Development of novel pyridazinone-based adenosine receptor ligands

Keywords: خواص ADME; AB-MECA; (N6-(4-aminobenzyl)-N-methylcarboxamidoadenosine); AC; adenylate cyclase; AR; adenosine receptor; CHO; Chinese Hamster Ovary; DPCPX; 8-cyclopentyl-1,3-dipropylxanthine; MV; molecular volume; NECA; 5′-(N-ethylcarboxamido)adenosine; TPSA; Topolog

دانلود رایگان متن کامل مقاله ISI 22 صفحه سال انتشار : 2018 سفارش ترجمه

Microwave-assisted synthesis of novel 5-substituted benzylidene amino-2-butyl benzofuran-3-yl-4-methoxyphenyl methanones as antileishmanial and antioxidant agents

Keywords: خواص ADME; Benzofuran derivatives; Antileishmanial activity; Antioxidant activity; Docking study; ADME properties;

دانلود رایگان متن کامل مقاله ISI 18 صفحه سال انتشار : 2018 سفارش ترجمه

Microwave assisted synthesis, computational study and biological evaluation of novel quinolin-2(1H)-one based pyrazoline hybrids

Keywords: خواص ADME; Microwave synthesis; 3-acetyl-4-hydroxyquinolin-2(1H)-one; Molecular docking; Anti-tubercular activity; ADME properties;

دانلود رایگان متن کامل مقاله ISI 30 صفحه سال انتشار : 2018 سفارش ترجمه

Synthesis, characterization and theoretical study in gaseous and solid phases of the imine 4-Acetyl-N-(4-methoxybenzylidene)aniline

Keywords: خواص ADME; Schiff's base; Ab initio calculations; Electronic structure; ADME properties;

دانلود رایگان متن کامل مقاله ISI 31 صفحه سال انتشار : 2017 سفارش ترجمه

Expeditious synthesis, antileishmanial and antioxidant activities of novel 3-substituted-4-hydroxycoumarin derivatives

Keywords: خواص ADME; 4-Hydroxycoumarin; Ceric ammonium nitrate; Antileishmanial activity; Antioxidant activity; Molecular docking study; ADME properties

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2016 سفارش ترجمه

Bacterial Peptide deformylase inhibition of cyano substituted biaryl analogs: Synthesis, in vitro biological evaluation, molecular docking study and in silico ADME prediction

Keywords: خواص ADME; Cyano substituted biaryl analogs; PDF inhibition; Antibacterial activity; Molecular docking; ADME properties;

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2016 سفارش ترجمه

Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of replacement of the 3-hydroxyphenyl group with pyridine or thiophene bioisosteres

Keywords: خواص ADME; [35S]GTPγS; sulfur-35 guanosine-5′-O-(3-thio)triphosphate; DAMGO; [D-Ala2,MePhe4,Gly-ol5]enkephalin; DPDPE; [D-Pen2,D-Pen5]enkephalin; U69,593; (5α,7α,8β)-(−)-N-methyl-N-[7-(1-pyrrolidinyl)-1-oxaspiro[4,5]dec-8-yl]benzeneacetamide; JDTic; Opioids;

دانلود رایگان متن کامل مقاله ISI 25 صفحه سال انتشار : 2016 سفارش ترجمه

Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of the 3- and 4-methyl substituents

Keywords: خواص ADME; JDTic; Opioids; Kappa antagonist; ADME properties

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2015 سفارش ترجمه

Biofilm inhibition of linezolid-like Schiff bases: Synthesis, biological activity, molecular docking and in silico ADME prediction

Keywords: خواص ADME; Linezolid-like Schiff bases; Biofilm inhibition; Antibacterial activity; Molecular docking; ADME properties;

دانلود رایگان متن کامل مقاله ISI 25 صفحه سال انتشار : 2015 سفارش ترجمه

Synthesis, antileishmanial activity and docking study of N′-substitutedbenzylidene-2-(6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)acetohydrazides

Keywords: خواص ADME; Thieno[3,2-c]pyridine; Antileishmanial activity; L. donovani promastigotes; Antimicrobial activity; Docking study; ADME properties;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2014 سفارش ترجمه

Novel (coumarin-3-yl)carbamates as selective MAO-B inhibitors: Synthesis, in vitro and in vivo assays, theoretical evaluation of ADME properties and docking study

Keywords: خواص ADME; (Coumarin-3-yl)carbamate scaffold; Monoamine oxidase (MAO); In vitro assays; In vivo assays; ADME properties; Docking studies

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2013 سفارش ترجمه

Novel N-methylsulfonamide and retro-N-methylsulfonamide derivatives as 17β-hydroxysteroid dehydrogenase type 2 (17β-HSD2) inhibitors with good ADME-related physicochemical parameters

Keywords: خواص ADME; 17β-Hydroxysteroid dehydrogenase type 2; Enzyme inhibition; Osteoporosis; N-Methylsulfonamide derivatives; Retro-N-methylsulfonamide derivatives; Structure–activity relationship; Structure–property relationship; ADME properties; pKa; Log P; Aqueous solubi

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2013 سفارش ترجمه

Synthesis, cytostatic activity and ADME properties of C-5 substituted and N-acyclic pyrimidine derivatives

Keywords: خواص ADME; 5-Alkyl pyrimidine derivatives; Cytostatic evaluations; Cell cycle analysis; ADME properties;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2012 سفارش ترجمه

Prediction of drug intestinal absorption by new linear and non-linear QSPR

Keywords: خواص ADME; QSPR theory; Molecular descriptors; Replacement method; Drug intestinal absorption; Model's applicability domain; ADME properties;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2011 سفارش ترجمه

Combinatorial design of nonsymmetrical cyclic urea inhibitors of aspartic protease of HIV-1

Keywords: خواص ADME; Inhibitor design; Aspartic protease of HIV-1; Library of nonsymmetrical cyclic ureas; Structure-based focusing; In silico screening; ADME properties

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2005 سفارش ترجمه