Keywords: مدولاتور آلومینیومی; Acetylcholinesterase inhibitors; Allosteric modulators; Alzheimer's disease;
مقالات ISI مدولاتور آلومینیومی (ترجمه نشده)
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Keywords: مدولاتور آلومینیومی; GPCRs; Opioid binding; Receptor; Molecular dynamics; Allosteric modulators; Virtual screening; Functional selectivity; Dimerization;
Keywords: مدولاتور آلومینیومی; Tetrahydroquinolines; Nicotinic Acetylcholine Receptors; Microwave-assisted synthesis; Allosteric Modulators; Povarov reaction;
Keywords: مدولاتور آلومینیومی; Agonist; allosteric modulators; convulsions; glutamate; mGlu5; schizophrenia; seizure;
Keywords: مدولاتور آلومینیومی; Nicotinic receptors; Chronic pain; Inflammation; Mice; Allosteric modulators; nAChR; nicotinic acetylcholine receptor(s); s.c.; subcutaneous injection; i.p.; intraperitoneally; CNS; central nervous system; ACh; acetylcholine; PAMs; positive allosteric mod
Profiling of orthosteric and allosteric group-III metabotropic glutamate receptor ligands on various G protein-coupled receptors with Tag-lite® assays
Keywords: مدولاتور آلومینیومی; Allosteric modulators; Screening technologies; Metabotropic glutamate receptors; GPCR; FRET;
Discovery of dual positive allosteric modulators (PAMs) of the metabotropic glutamate 2 receptor and CysLT1 antagonists for treating migraine headache
Keywords: مدولاتور آلومینیومی; Allosteric modulators; mGlu2; PAMs; Metabotropic glutamate receptor; CysLT1; Migraine;
Monastrol, a 3,4-dihydropyrimidin-2(1H)-thione, as structural scaffold for the development of modulators for GHB high-affinity binding sites and α1β2δ GABAA receptors
Keywords: مدولاتور آلومینیومی; GHB high-affinity binding sites; GABAA receptor; Allosteric modulators; Monastrol analogues; Biginelli cyclocondensation;
Structure–activity relationships of substituted 1H-indole-2-carboxamides as CB1 receptor allosteric modulators
Keywords: مدولاتور آلومینیومی; LQPOKCOXYJXERM-UHFFFAOYSA-N; UUUUKDIKVIQJQX-UHFFFAOYSA-NCB1 receptor; Allosteric modulators; Org compounds; Structure–activity relationship
Identification of novel allosteric modulator binding sites in NMDA receptors: A molecular modeling study
Keywords: مدولاتور آلومینیومی; N-methyl-d-aspartate receptors (NMDARs); Allosteric modulators; Molecular modeling; Docking; Modulator binding sites (MBSs)
Toward understanding the molecular basis for chemical allosteric modulator design
Keywords: مدولاتور آلومینیومی; Allosteric regulation; Allosteric modulators; Structural rigidity; “Allosteric-like” rule
Design and synthesis of substituted N-(1,3-diphenyl-1H-pyrazol-5-yl)benzamides as positive allosteric modulators of the metabotropic glutamate receptor subtype 5
Keywords: مدولاتور آلومینیومی; mGluR5; MPEP; CDPPB; Allosteric modulators
Broad-spectrum amino acid-sensing class C G-protein coupled receptors: Molecular mechanisms, physiological significance and options for drug development
Keywords: مدولاتور آلومینیومی; Allosteric modulators; Amino acid-sensing; Calcium-sensing receptor; Dimerisation; GPRC6A; G-protein coupled receptor; Molecular modelling; Taste receptors; Transgenic mouse; Venus FlyTrapAMPA, alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid; CaS
Structure-Activity Relationship of novel phenylacetic CXCR1 inhibitors
Keywords: مدولاتور آلومینیومی; GPCRs; Allosteric modulators; SAR; Conformational analysis;
GABAA receptors: Subtypes provide diversity of function and pharmacology
Keywords: مدولاتور آلومینیومی; GABA; Allosteric modulators; Heteropentamers; Inhibitory neurotransmission; Chloride channels;
Molecular determinants of non-competitive antagonist binding to the mouse GPRC6A receptor
Keywords: مدولاتور آلومینیومی; GPCR; Calcium; Allosteric modulators; Parathyroid
Benzodiazepine ligands can act as allosteric modulators of the Type 1 cholecystokinin receptor
Keywords: مدولاتور آلومینیومی; Allosteric modulators; Cholecystokinin receptor; Cooperativity; G protein-coupled receptors
Receptor activation involving positive allosteric modulation, unlike full agonism, does not result in GABAB receptor desensitization
Keywords: مدولاتور آلومینیومی; GABAB receptor; Allosteric modulators; Desensitization; GS39783GABA, γ-aminobutyric acid; GPCR, G-protein-coupled receptor; CHO, Chinese hamster ovary; CPA, N6-cyclopentyladenosine; GTPγS, guanosine 5′-O-(3-thiotriphosphate); DIV, day in vitro; HBSS, Hank
N6-1,3-Diphenylurea derivatives of 2-phenyl-9-benzyladenines and 8-azaadenines: Synthesis and biological evaluation as allosteric modulators of A2A adenosine receptors
Keywords: مدولاتور آلومینیومی; 2-Phenyl-9-benzyladenines; 2-Phenyl-9-benzyl-8-azaadenines; Adenosine receptor ligands; Allosteric modulators; 1,3-Diphenylureas
Prediction of the binding mode of biarylpropylsulfonamide allosteric AMPA receptor modulators based on docking, GRID molecular interaction fields and 3D-QSAR analysis
Keywords: مدولاتور آلومینیومی; Biarylpropylsulfonamides; AMPA receptor; Allosteric modulators; Binding mode; Docking; Glide; GRID; 3D-QSAR; GOLPE
Metabotropic glutamate receptors: Beyond the regulation of synaptic transmission
Keywords: مدولاتور آلومینیومی; Metabotropic glutamate receptors; Brain tumors; Stem cells; Immunological synapse; Antigen presenting cells; Allosteric modulators
Synthesis of desformylflustrabromine and its evaluation as an α4β2 and α7 nACh receptor modulator
Keywords: مدولاتور آلومینیومی; Nicotinic cholinergic receptors; Allosteric modulators
Pharmacological and computational analysis of alpha-subunit preferential GABAA positive allosteric modulators on the rat septo-hippocampal activity
Keywords: مدولاتور آلومینیومی; Hippocampus; Medial septum; Anxiety; Theta; Allosteric modulators; EEGEEG, electroencephalogram; INa, sodium current; IK, delayed rectifier potassium current; IK(A), A-type potassium current; IK(M), muscarinic potassium current; IK(C), C-type potassium cu
Allosteric modulation of GABAB receptor function in human frontal cortex
Keywords: مدولاتور آلومینیومی; Human frontal cortex; GABAB receptors; Allosteric modulators; [35S]-GTPγS binding; Adenylyl cyclase;
Metabotropic glutamate receptor 2 modulates excitatory synaptic transmission in the rat globus pallidus
Keywords: مدولاتور آلومینیومی; Metabotropic glutamate receptors; Group II; Globus pallidus; Excitatory transmission; Allosteric modulators; Parkinson's disease;