Keywords: فعالیت ضد انعکاس; Leishmaniasis; Medicinal plants; Antileishmanial activity; Ouezzane;
مقالات ISI فعالیت ضد انعکاس (ترجمه نشده)
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Keywords: فعالیت ضد انعکاس; Amino acid hydrazides; Quinazolinones; Antileishmanial activity;
Keywords: فعالیت ضد انعکاس; Ecuadorian propolis; Flavonoids; Triterpenoid; NMR; GC-MS; Antileishmanial activity;
Keywords: فعالیت ضد انعکاس; 4-amino-1,2,4-triazole; DFT calculations; NMR chemical shifts; FT-IR vibrational frequencies; Antileishmanial activity;
Keywords: فعالیت ضد انعکاس; Quinoline; Chalcones; 2-pyrazolines; Anticancer activity; Antifungal activity; Antibacterial activity; Antimalarial activity; Antitrypanosomal activity; Antileishmanial activity;
Keywords: فعالیت ضد انعکاس; Phenoxazines; Phenothiazines; Antileishmanial activity; Chloroacetamides; Trypanothione reductaseL. major, Leishmania major; MDR, multiple drug resistance; ND, not determined; Px, nonselenium glutathione peroxidase type tryparedoxin peroxidase; SAR, struc
Keywords: فعالیت ضد انعکاس; Quinolizidinyl-alkyliminophenazine derivatives; Pyrrolizidinyl-alkyliminophenazine derivatives; Clofazimine; Clofazimine analogs; Antiplasmodial activity; Antileishmanial activity;
Keywords: فعالیت ضد انعکاس; Antileishmanial activity; Leishmania braziliensis; Leishmania amazonensis; Tetrazole;
Promising antileishmanial activity of novel imidazole antifungal drug luliconazole against Leishmania major: In vitro and in silico studies
Keywords: فعالیت ضد انعکاس; Leishmania major; Luliconazole; Antileishmanial activity; In silico study;
In vitro activity of new N-benzyl-1H-benzimidazol-2-amine derivatives against cutaneous, mucocutaneous and visceral Leishmania species
Keywords: فعالیت ضد انعکاس; Benzimidazole derivatives; Antileishmanial activity; Selectivity Index; Arginase;
Microwave-assisted synthesis of novel 5-substituted benzylidene amino-2-butyl benzofuran-3-yl-4-methoxyphenyl methanones as antileishmanial and antioxidant agents
Keywords: فعالیت ضد انعکاس; Benzofuran derivatives; Antileishmanial activity; Antioxidant activity; Docking study; ADME properties;
Fruticulosin: A novel type 2 ribosome-inactivating protein from Abrus fruticulosus seeds that exhibits toxic and antileishmanial activity
Keywords: فعالیت ضد انعکاس; Type 2 RIP; Abrus fruticulosus; Toxin; Antileishmanial activity; SDS-PAGE; dodecyl sulphate-polyacrylamide gel electrophoresis; BSA; bovine serum albumin; CD; Circular dichroism; PBS; phosphate-buffered saline; FITC; fluorescein isothiocyanate; MTS; 3-(4,
Physicochemical and in vitro biological evaluations of furazolidone-based β-cyclodextrin complexes in Leishmania amazonensis
Keywords: فعالیت ضد انعکاس; Inclusion complex; Antileishmanial activity; Cutaneous canine leishmaniasis;
Novel organic salts based on quinoline derivatives: The in vitro activity trigger apoptosis inhibiting autophagy in Leishmania spp.
Keywords: فعالیت ضد انعکاس; Antileishmanial activity; Quinolines; Organic salts; Oxidative stress; Mitochondria dysfunction; Apoptosis;
Antileishmanial potential of fused 5-(pyrazin-2-yl)-4H-1,2,4-triazole-3-thiols: Synthesis, biological evaluations and computational studies
Keywords: فعالیت ضد انعکاس; Pyrazine; 1,2,4-Triazole; Antioxidant activity; Antileishmanial activity; Cytotoxicity activity; Molecular docking; ADMET analysis;
Antileishmanial evaluation of clubbed bis(indolyl)-pyridine derivatives: One-pot synthesis, in vitro biological evaluations and in silico ADME prediction
Keywords: فعالیت ضد انعکاس; Bis(indolyl)-pyridines; Camphor-10-sulfonic acid; Antileishmanial activity; Antibacterial activity; In silico studies;
Correlation between phenological changes, chemical composition and biological activities of the essential oil from Moroccan endemic Oregano (Origanum compactum Benth)
Keywords: فعالیت ضد انعکاس; Origanum compactum; Essential oil; Phenological stages; Antioxidant activity; Antibacterial activity; Antileishmanial activity;
Ag- and B-TiO2 nanostructures: Preparation, characterization and their antileishmanial activity
Keywords: فعالیت ضد انعکاس; TiO2; Ag-/B-TiO2; Nanotube; Hydrothermal synthesis; Amorphous boron; Antileishmanial activity;
Antioxidant antileishmanial cytotoxic and antimicrobial activities of a local plant Myrtus nivellei from Algeria Sahara
Keywords: فعالیت ضد انعکاس; Phenolic compounds; Flavonoids; Antioxidant activity; Antimicrobial activity; Antileishmanial activity; Myrtus nivellei;
1,2,4-triazole derivative with Schiff base; thiol-thione tautomerism, DFT study and antileishmanial activity
Keywords: فعالیت ضد انعکاس; NMR; FTIR and UV-vis spectroscopy; 1,2,4-Triazole derivative with Schiff base; Thiol-thione tautomerism; DFT calculations; Antileishmanial activity;
Effect of 1,2,3-triazole salts, non-classical bioisosteres of miltefosine, on Leishmania amazonensis
Keywords: فعالیت ضد انعکاس; 1/2/3-Triazoles; Leishmania; Miltefosine; Antileishmanial activity; Apoptosis; Necrosis;
Chemical composition of Mentha pulegium and Rosmarinus officinalis essential oils and their antileishmanial, antibacterial and antioxidant activities
Keywords: فعالیت ضد انعکاس; Essential oil; Mentha pulegium; Rosmarinus officinalis; Antileishmanial activity; Antibacterial activity; Antioxidant activity; Ouezzane;
Design, synthesis, structure-activity relationship and mechanism of action studies of a series of 4-chloro-1-phthalazinyl hydrazones as a potent agent against Leishmania braziliensis
Keywords: فعالیت ضد انعکاس; Leishmania braziliensis; Antileishmanial activity; Superoxide dismutase; Promastigotes; Phthalazine; Nitroheterocycle;
In silico molecular docking studies of new potential 4-phthalazinyl-hydrazones on selected Trypanosoma cruzi and Leishmania enzyme targets
Keywords: فعالیت ضد انعکاس; Trypanosoma cruzi; Leishmania; Molecular docking; Phthalazines; Antichagasic activity; Antileishmanial activity;
Ring-closing metathesis based total synthesis of ciliatamides A and B and their structural confirmation
Keywords: فعالیت ضد انعکاس; Ciliatamides; Antileishmanial activity; Caprolactam; Amide bond formation; Ring-closing metathesis;
In vitro studies of the antileishmanial activity of the newer 2-(substitutedphenoxy)-N-[(aryl)methylidene]acetohydrazide analogues
Keywords: فعالیت ضد انعکاس; Acetohydrazide analogues; Antileishmanial activity; Leishmania donovani
New platinum(II) complexes of CCC-pincer N-heterocyclic carbene ligand: Synthesis, characterization, cytotoxicity and antileishmanial activity
Keywords: فعالیت ضد انعکاس; Carbene ligand; Pt(II) complex; Antileishmanial activity; Cytotoxicity; Lipophilicity
Physalis angulata induces death of promastigotes and amastigotes of Leishmania (Leishmania) amazonensis via the generation of reactive oxygen species
Keywords: فعالیت ضد انعکاس; Physalis angulata; L. (L.) amazonensis; Antileishmanial activity; Macrophage activation; ROS production
Expeditious synthesis, antileishmanial and antioxidant activities of novel 3-substituted-4-hydroxycoumarin derivatives
Keywords: فعالیت ضد انعکاس; 4-Hydroxycoumarin; Ceric ammonium nitrate; Antileishmanial activity; Antioxidant activity; Molecular docking study; ADME properties
An effective in vitro and in vivo antileishmanial activity and mechanism of action of 8-hydroxyquinoline against Leishmania species causing visceral and tegumentary leishmaniasis
Keywords: فعالیت ضد انعکاس; Leishmania; 8-Hydroxyquinoline; Antileishmanial activity; Leishmaniasis; Treatment; Toxicity
Synthesis and evaluation against Leishmania amazonensis of novel pyrazolo[3,4-d]pyridazinone-N-acylhydrazone-(bi)thiophene hybrids
Keywords: فعالیت ضد انعکاس; Antileishmanial activity; Pyrazolo-pyridazinone; N-acylhydrazone; Thiophene; Trypanothione reductase;
Antileishmanial activity and mechanism of action from a purified fraction of Zingiber officinalis Roscoe against Leishmania amazonensis
Keywords: فعالیت ضد انعکاس; Antileishmanial activity; Zingiber officinalis Roscoe; Leishmania amazonensis; Treatment; Nitric oxide; Purified compounds;
Synthesis and biological evaluation of 2-arylbenzimidazoles targeting Leishmania donovani
Keywords: فعالیت ضد انعکاس; 2-Arylbenzimidazoles; Leishmania donovani; Antileishmanial activity; Biological activity; Medicinal chemistry
Chemical constituents from Sidastrum paniculatum and evaluation of their leishmanicidal activity
Keywords: فعالیت ضد انعکاس; Sidastrum paniculatum; Malvaceae; Leishmania braziliensis; Antileishmanial activity
Synthesis of 5-isoxazol-3-yl-pyrimidine nucleosides as potential antileishmanial agents
Keywords: فعالیت ضد انعکاس; Isoxazole; Pyrimidine nucleoside; Hybrid; 1,3-Dipolar cycloaddition; Antileishmanial activity;
Nanoemulsions loaded with amphotericin B: A new approach for the treatment of leishmaniasis
Keywords: فعالیت ضد انعکاس; Amphotericin B; Nanoemulsion; Stearylamine; Cholesterol; Cytotoxicity; Antileishmanial activity
Antileishmanial and cytotoxic potential of essential oils from medicinal plants in Northern Tunisia
Keywords: فعالیت ضد انعکاس; Leishmaniasis; L. major; L. infantum; Essential oils; Antileishmanial activity; Cytotoxicity
Antimony(III) complexes with 2-amino-4,6-dimethoxypyrimidines: Synthesis, characterization and biological evaluation
Keywords: فعالیت ضد انعکاس; Antimony(III) complexes; Antileishmanial activity; Glutathione reductase inhibition
Synthesis, spectroscopic characterization and in vitro antimicrobial, anticancer and antileishmanial activities as well interaction with Salmon sperm DNA of newly synthesized carboxylic acid derivative, 4-(4-methoxy-2-nitrophenylamino)-4-oxobutanoic acid
Keywords: فعالیت ضد انعکاس; Carboxylic acid derivative; Antimicrobial activity; Anticancer activity; Antileishmanial activity; DNA interaction; Petra/Osiris/Molinspiration (POM) analyses
Design, structural and spectroscopic elucidation and in vitro antimicrobial, anticancer, antileishmanial, urease inhibition activities and interaction with SS-DNA of newly synthesized amide based carboxylic acid
Keywords: فعالیت ضد انعکاس; Crystal structure; Antimicrobial activity; Anticancer activity; Antileishmanial activity; DNA interaction
Synthesis, spectroscopic characterization, biological screenings, DNA binding study and POM analyses of transition metal carboxylates
Keywords: فعالیت ضد انعکاس; Metal carboxylate; Antifungal activity; Antileishmanial activity; DNA-interaction; POM analysis
Synthesis, antileishmanial activity and cytotoxicity of 2,3-diaryl- and 2,3,8-trisubstituted imidazo[1,2-a]pyrazines
Keywords: فعالیت ضد انعکاس; Antileishmanial activity; Imidazo[1,2-a]pyrazines; Direct arylation; Casein kinase 1;
Synthesis, characterization, and antileishmanial activities of gold(I) complexes involving quinoline functionalized N-heterocyclic carbenes
Keywords: فعالیت ضد انعکاس; Gold; N-heterocyclic carbene; Quinoline; Leishmania infantum; J774A.1; Antileishmanial activity;
The effect of the phytol-rich fraction from Lacistema pubescens against Leishmania amazonensis is mediated by mitochondrial dysfunction
Keywords: فعالیت ضد انعکاس; Lacistema pubescens; Phytol; Leishmania amazonensis; Antileishmanial activity; Mitochondrial dysfunction;
Antileishmanial activity of Opuntia ficus-indica fractions
Keywords: فعالیت ضد انعکاس; Opuntia ficus-indica; Antileishmanial activity; Trypanocidal activity; Bioguided fractionation
Antileishmanial metabolites from Trixis antimenorrhoea
Keywords: فعالیت ضد انعکاس; Trixis antimenorrhoea; Nortrixane; Trixanolide; Antileishmanial activity; Structural elucidation;
Synthesis, antileishmanial activity and docking study of Nâ²-substitutedbenzylidene-2-(6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)acetohydrazides
Keywords: فعالیت ضد انعکاس; Thieno[3,2-c]pyridine; Antileishmanial activity; L. donovani promastigotes; Antimicrobial activity; Docking study; ADME properties;
Bioactive indole alkaloids isolated from Alstonia angustifolia
Keywords: فعالیت ضد انعکاس; Alstonia angustifolia (Apocynaceae); Stem bark; Sarpagine-type alkaloid; Macroline-type alkaloid; Macroline-pleiocarpamine bisindole alkaloid; Cytotoxicity; NF-κB (p65) inhibitory activity; Antileishmanial activity;
Binary classification of chalcone derivatives with LDA or KNN based on their antileishmanial activity and molecular descriptors selected using the Successive Projections Algorithm feature-selection technique
Keywords: فعالیت ضد انعکاس; Antileishmanial activity; Successive Projections Algorithm; Linear Discriminant Analysis; Genetic Algorithm; One Nearest Neighbour
Synthesis and evaluation of the antiparasitic activity of bis-(arylmethylidene) cycloalkanones
Keywords: فعالیت ضد انعکاس; Bis-(arylmethylidene)-cycloalkanones; Antileishmanial activity; Leishmania amazonensis; Trypanocidal; Trypanosoma cruziQBJZDRXWVFLWLM-AYKLPDECSA-N; MOGZMXKHFUIRHE-RYQLWAFASA-N; CETXDHNPPYXEOF-OZNQKUEASA-N; CYVVJSKZRBZHAV-UNZYHPAISA-N; VJTIKIQJUZWNSW-JOBJL