Keywords: Antileishmanial; Antimicrobial; Antiplasmodial; Antitrypanosomal; Drug discovery; Eleusine indica; Macaranga barteri;
مقالات ISI (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: Azole; Antitrypanosomal; Antiplasmodial; Antileishmanial; Antifungal; CYP51; In vivo studies; NTDs; neglected tropical diseases; CYP51; sterol 14α-demethylase; Ph; phenyl; Py; 1-pyrrolyl; Tb; Trypanosoma brucei rhodesiense; Tc; Trypanosoma cruzi; Ld; Le
Keywords: Antitrypanosomal; Antileishmanial; Tyrosol; Hydroxytyrosol;
Keywords: Synthesis; Ent-kaurane; Caracasine acid; Cytotoxic activity; Antileishmanial; Antitrypanosomal; Antibacterial;
Keywords: FCQZEZCNARMPGO-UHFFFAOYSA-N; CWGVNUWQWUADFX-BQYQJAHWSA-N; HVBSAKJJOYLTQU-UHFFFAOYSA-N; BPICBUSOMSTKRF-UHFFFAOYSA-N; In silico study; TOMOCOMD-CARDD software; Non-stochastic and stochastic linear indices; Classification model; Machine learning-based QSAR
Biological activities of plant extracts from Ficus elastica and Selaginella vogelli: An antimalarial, antitrypanosomal and cytotoxity evaluation
Keywords: Antiplasmodial; Antitrypanosomal; Cytotoxicity; Ficus elastica; Selaginella vogelii;
Antitrypanosomal activity and evaluation of the mechanism of action of dehydrodieugenol isolated from Nectandra leucantha (Lauraceae) and its methylated derivative against Trypanosoma cruzi
Keywords: Neolignans; Nectandra leucantha; Antitrypanosomal; Plasma membrane permeabilization; ADMET; absorption, distribution, metabolism, excretion, and toxicity; ANOVA; analysis of variance; ASE; accelerated solvent extractor; AU; arbitrary fluorescent unity; BA
Synthesis and evaluation of analogs of 5â²-(((Z)-4-amino-2-butenyl)methylamino)-5â²-deoxyadenosine (MDL 73811, or AbeAdo) - An inhibitor of S-adenosylmethionine decarboxylase with antitrypanosomal activity
Keywords: AdoMet; S-adenosyl-l-methionine; AdoMetDC; S-adenosylmethionine decarboxylase; BBB; bloodbrain barrier; Boc; tert-butoxycarbonyl; BSA; N,O-bis(trimethylsilyl)acetamide; CNS; central nervous system; DEAD; diethyl azodicarboxylate; DIAD; diisopropyl azodica
In vivo ameliorative effects of methanol leaf extract of Lawsonia inermis Linn on experimental Trypanosoma congolense infection in Wistar rats
Keywords: ANOVA; analysis of variance; EOF; erythrocyte osmotic fragility; IP; intraperitoneal; kDNA; kinetoplast deoxyribonucleic acid; L; lawsonia; MDA; malondialdehyde; PCV; packed cell volume; PSS; physiological buffered saline; SEM; standard error of mean; T;
Synthesis of novel amide and urea derivatives of thiazol-2-ethylamines and their activity against Trypanosoma brucei rhodesiense
Keywords: Thiazole; Amide; Urea; Antitrypanosomal; Metabolic stability;
New cycloartane saponin and monoterpenoid glucoindole alkaloids from Mussaenda luteola
Keywords: Mussaenda luteola; Rubiaceae; Antitrypanosomal; Cycloartane-type saponin; Monoterpenoid glucoindole alkaloid;
Potent antitrypanosomal triterpenoid saponins from Mussaenda luteola
Keywords: Mussaenda luteola; Rubiaceae; Triterpenoid saponins; Antitrypanosomal; μ-Opioid receptor binding
Synthesis, antileishmanial and antitrypanosomal activities of N-substituted tetrahydro-β-carbolines
Keywords: Tetrahydro-β-carbolines; Antileishmanial; Antitrypanosomal; Leishmania donovani; Leishmaniasis; African trypanosomiasis;
New metal complexes of NNO tridentate ligands: Effect of metal center and co-ligand on biological activity
Keywords: Oxidovanadium(IV) and dioxidovanadium(V) complexes; Gallium(III); N,N,O ligands; Antitrypanosomal; Antitumoral
Antiprotozoal activity of dicationic 3,5-diphenylisoxazoles, their prodrugs and aza-analogues
Keywords: Diarylisoxazole; Diamidine; Prodrug; Antiprotozoal; Antitrypanosomal;
Oxidovanadium(IV) and dioxidovanadium(V) complexes of tridentate salicylaldehyde semicarbazones: Searching for prospective antitrypanosomal agents
Keywords: Oxidovanadium(IV) complexes; Dioxidovanadium(V) complexes; Salicylaldehyde semicarbazones; Antitrypanosomal; 2,2â²-bipyridine; dipyrido[3,2-a: 2â²,3â²-c]phenazine;
Synthesis and antiprotozoal activities of benzyl phenyl ether diamidine derivatives
Keywords: Diamidines; Prodrugs; Benzyl phenyl ether derivatives; Antiprotozoal; Antitrypanosomal; Antiplasmodial; AntileishmanialATMS, artemisinin; BPE, benzyl phenyl ether; CQ, chloroquine; FMD, furamidine; HAT, human African trypanosomiasis; IC50, 50% inhibition
Synthesis of antitrypanosomal 1,2-dioxane derivatives based on a natural product scaffold
Keywords: Natural product scaffold; Ene reaction; 1,2-Dioxane; Antitrypanosomal; HAT
Convolutamines I and J, antitrypanosomal alkaloids from the bryozoan Amathia tortusa
Keywords: Marine bryozoan; Convolutamines; Antitrypanosomal; Trypanosoma brucei brucei;
In vitro antitrypanosomal activity of plant terpenes against Trypanosoma brucei
Keywords: In vitro; Antitrypanosomal; Terpenes; Plant products;
Antiparasitic activity of alkaloids from plant species of Papua New Guinea and Australia
Keywords: Antimalarial; Antitrypanosomal; Alkaloid; Plant; Flindersia; Stage specificity
Phytochemical and biological investigations of Elaeodendron schlechteranum
Keywords: Elaeodendron schlechteranum; Celastraceae; Antibacterial; Antitrypanosomal; Antileishmanial; Antiplasmodial; Anti-HIV; Cytotoxicity; Triterpenes; Tingenin B; Prodelphinidin
Synthesis, in vitro antitrypanosomal and antibacterial activity of phenoxy, phenylthio or benzyloxy substituted quinolones
Keywords: Chagas’ disease; Trypanosoma cruzi; Quinolones; Antitrypanosomal; Antibacterial activity
Synthesis and antiprotozoal activities of dicationic bis(phenoxymethyl)benzenes, bis(phenoxymethyl)naphthalenes, and bis(benzyloxy)naphthalenes
Keywords: Diamidines; Xylene derivatives; Naphthalene derivatives; Antiprotozoal; Antitrypanosomal; Antiplasmodial; Antileishmanial
In vitro antitrypanosomal activities of quassinoid compounds from the fruits of a medicinal plant, Brucea javanica
Keywords: Brucea javanica; Quassinoids; Trypanosoma evansi; Antitrypanosomal; Medicinal plant