Keywords: فعال سازی بیولوژیک; Endocrine disruption; Reporter gene assay; Metabolism; Bioactivation;
مقالات ISI فعال سازی بیولوژیک (ترجمه نشده)
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Keywords: فعال سازی بیولوژیک; Earthworms; Biochar; Extracellular enzymes; Bioactivation; Soil pollution;
Keywords: فعال سازی بیولوژیک; Bioactivation; Drug discovery and development; Drug metabolism; Metabolite; Pharmacokinetics; Pharmacodynamics; Safety; Toxicity;
Keywords: فعال سازی بیولوژیک; Terbinafine; Reactivity; Liver toxicity; Bioactivation; TBF-A;
Keywords: فعال سازی بیولوژیک; Masked mycotoxins; Regulation; Deconjugation; Bioactivation;
Keywords: فعال سازی بیولوژیک; Bioactivation; Titanium disc; Octacalcium phosphate (OCP); Induction time ((τin)); Nucleation; Supersaturated solution
Keywords: فعال سازی بیولوژیک; Bioactivation; Biotransformation; Cytochrome P450; Drug development; Drug discovery; Drug metabolism; Electrochemical generation; Electrochemistry; Metabolite synthesis; Reactive metabolite
Keywords: فعال سازی بیولوژیک; Toremifene; Tamoxifen; Metabolite kinetics; Bioactivation; CYP2D6; CYP3A4; CYP2C9; Pharmacogenomics; PolymorphismsTOR, toremifene; TAM, tamoxifen; SERM, selective estrogen receptor modulator; SSRI, selective serotonin reuptake inhibitor; 4OH, 4-hydroxy; N
Keywords: فعال سازی بیولوژیک; Bioactivation; Glutathione trapping assay; Idiosyncratic toxicity; Reactive intermediate; Stable isotope
Keywords: فعال سازی بیولوژیک; Orexin; Antagonist; Sleep; Bioactivation; Pyrimidine;
Effect of UGT2B7*2 and CYP2C8*4 polymorphisms on diclofenac metabolism
Keywords: فعال سازی بیولوژیک; CYP; cytochrome P450; CYP-reductase; NADPH cytochrome P450 reductase; DCF-AG; diclofenac acyl glucuronide; DCF-SG; diclofenac glutathione conjugate; DILI; drug-induced liver injury; ESI; electrospray ionization; GST; glutathione S-transferase; GWAS; genom
Formation and biological targets of botanical o-quinones
Keywords: فعال سازی بیولوژیک; Quinones; P450; Bioactivation; Botanicals; Chemoprevention; Carcinogen; ARE; antioxidant response element; BiP; binding immunoglobin protein; COX-2; cyclooxygenase-2; JNK; c-Jun N-terminal kinase; EGCG; (â)-epigallocatechin gallate; GST; glutathione-S-t
In vitro ocular metabolism and bioactivation of ketoconazole in rat, rabbit and human
Keywords: فعال سازی بیولوژیک; Ocular metabolism; Ocular S9 fractions; Liver S9 fractions; Bioactivation; Potassium cyanide; [M+H]+; protonated molecular ion; KT; ketoconazole; RT; retention time; DAK; N-deacetylated ketoconazole; FMO; Flavin monooxygenase; LC; liquid chromatography; M
Is there a human health risk associated with indirect exposure to perfluoroalkyl carboxylates (PFCAs)?
Keywords: فعال سازی بیولوژیک; Fluorotelomer-based substances; Perfluorinated carboxylates; Exposure; Toxicity; Bioactivation; Covalent binding;
Difluorocyclobutylacetylenes as positive allosteric modulators of mGluR5 with reduced bioactivation potential
Keywords: فعال سازی بیولوژیک; mGluR5; PAMs; Cognition; Schizophrenia; Bioactivation;
Hepato-protective effects of six schisandra lignans on acetaminophen-induced liver injury are partially associated with the inhibition of CYP-mediated bioactivation
Keywords: فعال سازی بیولوژیک; ALT; alanine aminotransferase; APAP; acetaminophen; AST; aspartate aminotransferase; CYP; cytochrome P450; GSH; glutathione; NAPQI; N-acetyl-p-benzoquinone imine; SinA; Schisandrin A; SinB; Schisandrin B; SinC; Schisandrin C; SolA; Schisandrol A; SolB; Sc
Novel adducts from the reaction of 1-chloro-3-buten-2-one with 2â²-deoxyguanosine. Structural characterization and potential as tools to investigate 1,3-butadiene carcinogenicity
Keywords: فعال سازی بیولوژیک; ADH; alcohol dehydrogenase; BD; 1,3-butadiene; CBO; 1-chloro-3-buten-2-one; CHB; 1-chloro-2-hydroxy-butene; COSY; correlation spectroscopy; dG; 2â²-deoxyguanosine; DMSO-d6; hexadeuterodimethyl sulfoxide; ESI; electrospray ionization; HMBC; heteronuclear
Nicotine, cotinine, and β-nicotyrine inhibit NNK-induced DNA-strand break in the hepatic cell line HepaRG
Keywords: فعال سازی بیولوژیک; 8-MOP; 8-methoxypsoralen; dH2O; deionosed water; HBECS; human bronchial epithelial cells; HPB; 4-oxo-4-(3-pyridyl) 1-butanol; HPLC; high pressure liquid chromatography; IARC; International Agency for the Research on Cancer; NNK; 4-(methylnitrosamino)-1-(3
N-(Pyridin-2-yl) arylsulfonamide inhibitors of 11β-hydroxysteroid dehydrogenase type 1: Strategies to eliminate reactive metabolites
Keywords: فعال سازی بیولوژیک; 11β-Hydroxysteroid dehydrogenase; 11β-HSD; PF-915275; Reactive metabolite; Bioactivation; Glutathione adduct; Diabetes; Inhibitor;
Inhibition of methyleugenol bioactivation by the herb-based constituent nevadensin and prediction of possible in vivo consequences using physiologically based kinetic modeling
Keywords: فعال سازی بیولوژیک; Methyleugenol; PBK; Nevadensin; Inhibition; Bioactivation; In vivo; NTP; National Toxicology Program; SCF; Scientific Committee on Food; FEMA; Flavor and Extract Manufacturers Association; PBK; physiologically based kinetic; NEV; nevadensin; DMSO; dimethy
Scrambled and fried: Cigarette smoke exposure causes antral follicle destruction and oocyte dysfunction through oxidative stress
Keywords: فعال سازی بیولوژیک; Cigarette; Ovotoxicity; Oxidative stress; Bioactivation; Atresia; Infertility
Structural modifications of a 3-methoxy-2-aminopyridine compound to reduce potential for mutagenicity and time-dependent drug-drug interaction
Keywords: فعال سازی بیولوژیک; Bioactivation; AMES positive; TDI; Toxicity; Electron rich heteroaryls; Kinase inhibitor; Reactive metabolite; Mutagenicity; Time dependent drug-drug interaction;
Structure-toxicity relationship study of para-halogenated styrene analogues in CYP2E1 transgenic cells
Keywords: فعال سازی بیولوژیک; Styrene; Styrene oxide; Bioactivation; Protein adduct
Bovine liver slices: A multifunctional in vitro model to study the prohormone dehydroepiandrosterone (DHEA)
Keywords: فعال سازی بیولوژیک; Bioactivation; Prohormone; Liver slice; Bioassay; Mass spectrometry; Genomics;
A new class of bioactivable self-immolative N,O-ligands
Keywords: فعال سازی بیولوژیک; Amino-phenol ligand; N,O-ligand; Bioactivation; β-Galactosidase; Self-immolativeKJBYBRFWTKPYPH-UHFFFAOYSA-N; VVRBMHPNQBIASX-UHFFFAOYSA-N; CKUJUWPSSMSMGC-UHFFFAOYSA-N; DNSURQOAHPWGTC-UHFFFAOYSA-N; POLIMGHWFJBGIY-UHFFFAOYSA-N; HOGRZCLXGFXORR-UHFFFAOYSA-N; P
Stimulation of Human Monocytic THP-1 Cells by Metabolic Activation of Hepatotoxic Drugs
Keywords: فعال سازی بیولوژیک; adverse drug reactions; bioactivation; monocytes/macrophages; CYP3A4; drug-induced hepatotoxicity; inflammation;
Establishing a total allowable concentration of o-toluidine in drinking water incorporating early lifestage exposure and susceptibility
Keywords: فعال سازی بیولوژیک; Risk assessment; o-Toluidine; Drinking water; Susceptibility; Childhood; Lifestage; Bioactivation; Mutagenic; Mode of action; Cancer
Nanoengineered polymeric S-layers based capsules with targeting activity
Keywords: فعال سازی بیولوژیک; Polyelectrolyte capsules; Bacterial S-layer proteins; Bioactivation; Cytotoxicity
Drug bioactivation and protein adduct formation in the pathogenesis of drug-induced toxicity
Keywords: فعال سازی بیولوژیک; Bioactivation; Innate immunity; Adaptive immunity; Protein adduct; Drug hypersensitivity; Toxicity
d-Isomer of gly-tyr-pro-cys-pro-his-pro peptide: A novel and sensitive in vitro trapping agent to detect reactive metabolites by electrospray mass spectrometry
Keywords: فعال سازی بیولوژیک; Bioactivation; LC/MS liquid chromatography mass spectrometry; Reactive metabolites; Covalent binding; Peptide d-isomer and peptide adducts
Aflatoxin B1 in poultry: Toxicology, metabolism and prevention
Keywords: فعال سازی بیولوژیک; Aflatoxin B1; Aflatoxicosis; P450s; Metabolism; Bioactivation; Liver cancer; Cytochrome P450; Glutathione S-transferase; Chemoprevention
Quantitative assessment of the metabolic activation of alicyclic amines via aldehyde
Keywords: فعال سازی بیولوژیک; Aldehyde; Alicyclic amines; Bioactivation; In vitro method; Post-incubation; Quantitative; Radiolabeled trapping reagent
Evidence for cellular protein covalent binding derived from styrene metabolite
Keywords: فعال سازی بیولوژیک; PBST, 200 mM phosphate-buffered saline solution containing 0.02% Tween-20 at pH 7.4; TBS-Tween, 100 mM Tris-base buffer containing 154 mM NaCl and 0.5% Tween-20 at pH 7.4; TRI, trichloroethyleneStyrene; Styrene oxide; Bioactivation; Protein adduction
A framework for using structural, reactivity, metabolic and physicochemical similarity to evaluate the suitability of analogs for SAR-based toxicological assessments
Keywords: فعال سازی بیولوژیک; Structural-similarity; Reactive-similarity; Metabolic-similarity; Bioactivation; Chemical analogs identification; Structure activity relationship (SAR); Toxicological assessments
Mitochondrial aldehyde dehydrogenase (ALDH-2)—Maker of and marker for nitrate tolerance in response to nitroglycerin treatment
Keywords: فعال سازی بیولوژیک; Organic nitrate; Bioactivation; Superoxide; Peroxynitrite; Mitochondrial aldehyde dehydrogenase; Mitochondrial oxidative stress; Vascular function
Bioactivation of fluorotelomer alcohols in isolated rat hepatocytes
Keywords: فعال سازی بیولوژیک; Perfluorinated acid; Telomer alcohol; Bioactivation; Cytotoxicity; Protein carbonylation; Alkenal toxicity
Effect of local, long-term delivery of platelet-derived growth factor (PDGF) on injected fat graft survival in severe combined immunodeficient (SCID) mice
Keywords: فعال سازی بیولوژیک; Fat graft; PDGF; Bioactivation
Bioactivation of coumarin in rat olfactory mucosal microsomes: Detection of protein covalent binding and identification of reactive intermediates through analysis of glutathione adducts
Keywords: فعال سازی بیولوژیک; Coumarin; Olfactory mucosa; Bioactivation; Glutathione adduct; Protein covalent binding
Phase I to II cross-induction of xenobiotic metabolizing enzymes: A feedforward control mechanism for potential hormetic responses
Keywords: فعال سازی بیولوژیک; Hormesis; Bioactivation; Feedforward; Feedback; Overcompensation; Reactive metabolite; Xenobiotics; Nrf2
Comparative preclinical drug metabolism and pharmacokinetic evaluation of novel 4-aminoquinoline anti-malarials
Keywords: فعال سازی بیولوژیک; preclinical pharmacokinetics; drug design; pro-drugs; ADME; cytochrome P450; MDCK cells; protein binding; blood partitioning; anti-malarials; bioactivation;
Drug metabolism
Keywords: فعال سازی بیولوژیک; bioactivation; cytochrome P450 enzymes; enzyme induction; enzyme inhibition; genetic polymorphisms; interactions; metabolism
Trifluoromethylpyrimidine-based inhibitors of proline-rich tyrosine kinase 2 (PYK2): Structure–activity relationships and strategies for the elimination of reactive metabolite formation
Keywords: فعال سازی بیولوژیک; PYK2; FAK; Kinase; Osteoporosis; Bioactivation; Reactive metabolite
Bioactivation of the tricyclic antidepressant amitriptyline and its metabolite nortriptyline to arene oxide intermediates in human liver microsomes and recombinant P450s
Keywords: فعال سازی بیولوژیک; P450, cytochrome P450; TCAs, tricyclic antidepressants; PI, precursor ion; EPI, enhanced product ion; HLM, human liver microsomes; GSH, glutathioneAmitriptyline; Nortriptyline; Bioactivation; P450; Hepatotoxicity; Arene oxide
High potency of bioactivation of 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine (PhIP) in mouse colon epithelial cells with ApcMin mutation
Keywords: فعال سازی بیولوژیک; Bioactivation; Heterocyclic aromatic amines; PhIP; Apc gene; Min Mutation; Colorectal carcinogenesis; Ah receptor; CYP1A
β-Glucosidases as detonators of plant chemical defense
Keywords: فعال سازی بیولوژیک; BGAF; β-glucosidase aggregating factor; DIBOA; 2,4-dihydroxy-1,4-benzoxazin-3-one; DIMBOA; 2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one; ESM; epithiospecifier modifying protein; ESP; epithiospecifier protein; BxGlc; benzoxazinoid glucoside; MBP; myrosina
Human cytosolic sulfotransferase SULT1A1
Keywords: فعال سازی بیولوژیک; Human cytosolic sulfotransferase; SULT1A1; Phase II metabolism; Bioactivation; PAPS; p-Nitrophenol;
Structure–activity relationship study of novel NR2B-selective antagonists with arylamides to avoid reactive metabolites formation
Keywords: فعال سازی بیولوژیک; Reactive metabolite; Bioactivation; NR2B; NMDA; Metabolic stability
Regulating biological activity in plants with carboxylesterases
Keywords: فعال سازی بیولوژیک; Bioactivation; Detoxification; Herbicides; Secondary metabolism; Serine hydrolase; Signalling;
Toxicokinetics and toxicity of thioacetamide sulfoxide: a metabolite of thioacetamide
Keywords: فعال سازی بیولوژیک; Thioacetamide; Thioacetamide sulfoxide; Liver injury; Bioactivation; Saturation
Human glutathione transferases catalyzing the bioactivation of anticancer thiopurine prodrugs
Keywords: فعال سازی بیولوژیک; Thiopurine prodrugs; Glutathione transferase; cis-6-(2-Acetylvinylthio)purine; trans-6-(2-Acetylvinylthio)guanine; Bioactivation; Chemotherapy