Keywords: CB1، گیرنده کانابینوئید 1; AEA, anandamide; AG, 2-arachidonoyl glycerol; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CB receptor, cannabinoid receptor; FAAH, fatty acid amide hydrolase; NM, nitrogen mustard; OEA, oleyolethanolamide; PEA, palmitoylethanolamide; PPARα,
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Keywords: CB1، گیرنده کانابینوئید 1; AEA, arachidonoyl ethanolamide; 2-AG, 2-arachidonoylglycerol; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; FAAH, fatty acid amide hydrolase; FLS, fibroblastlike synoviocyte; IFN, interferon; IL, interleukin; MMP, matrix metalloproteinase; RA,
Keywords: CB1، گیرنده کانابینوئید 1; PND, post natal day; PPI, pre-pulse inhibition; THC, delta9-tetrahydrocannabinol; PCP, phencyclidine; COMT, catechol-O-methyltransferase; CB1, cannabinoid receptor 1; 5-HT2A serotonin 2A receptor, NMDA N-methyl-D-aspartate receptor; mGluR5, metabotropic g
Keywords: CB1، گیرنده کانابینوئید 1; 5 HT, serotonin; 5NC, 5 individual NC tests; ASIC3, acid-sensing ion channel 3; BDNF, brain-derived neurotrophic factor; BR2, bradykinin receptor; CB1, cannabinoid receptor 1; CGRP, calcitonin gene-related peptide; CI, confidence interval; CMAP, compound
Keywords: CB1، گیرنده کانابینوئید 1; SCBs, synthetic cannabinoids; CB1, cannabinoid receptor 1; QSAR, quantitative structure-activity relationship; Ki, binding constant; CATS, chemically advance template search; PPP, potential pharmacophore points; FPDSim, feature-pair distribution similarit
Pyrazole antagonists of the CB1 receptor with reduced brain penetration
Keywords: CB1، گیرنده کانابینوئید 1; BBB, blood–brain barrier; BOP, benzotriazol-1-yl-oxytris(dimethylamino)phosphonium hexafluorophosphate; CB, cannabinoid receptors; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CHO-K1, Chinese hamster ovary cells; CMA 80, 80% chloroform, 18% m
Anti-inflammatory and antioxidant effects of a combination of cannabidiol and moringin in LPS-stimulated macrophages
Keywords: CB1، گیرنده کانابینوئید 1; LPS, lipopolysaccharide; TNF-α, tumor necrosis factor-α; IL-1β, interleukin-1β; IFN-γ, interferon-γ; IL-6, interleukin-6; NO, nitric oxide; iNOS, nitric oxide synthase; CBD, cannabidiol; THC, tetrahydrocannabinol; CB1, cannabinoid receptor 1; CB2, cannabi
Angiotensin II and taste sensitivity
Keywords: CB1، گیرنده کانابینوئید 1; ALDO, aldosterone; ANG II, angiotensin II; AT1 (AT2), angiotensin II receptor type 1 (type 2); CB1, cannabinoid receptor 1; CT, chorda tympani; ENaC, epithelial sodium channel; GFP, green fluorescent protein; HCl, hydrochloric acid; i.p, intraperitoneal;
Enterocyte fatty acid-binding proteins (FABPs): Different functions of liver and intestinal FABPs in the intestine
Keywords: CB1، گیرنده کانابینوئید 1; Fatty acid-binding protein; Fatty acid; Intestine; Lipid; LFABP; IFABP2-AG, 2-arachidonoylglycerol; AEA, arachidinoylethanolamide; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; FA, fatty acid; FXR, farnesoid X receptor; IFABP, intestinal fatty
Endocannabinoid metabolism by cytochrome P450 monooxygenases
Keywords: CB1، گیرنده کانابینوئید 1; 2-AG, 2-arachidonylglycerol; AEA, anandamide; AA, arachidonic acid; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CNS, central nervous system; COX, cyclooxygenase; CYP, cytochrome P450; DAG, diacylglycerol; DHET, dihydroxyeicosatrienoic acid;
5-HT receptor-mediated modulation of granule cell inhibition after juvenile stress recovers after a second exposure to adult stress
Keywords: CB1، گیرنده کانابینوئید 1; ACSF, artificial cerebrospinal fluid; ampl, amplitude; ANOVA, analysis of variance; as, adult stress; CB1, cannabinoid receptor 1; CCK, cholecystokinin; CNQX, 6-cyano-7-nitroquinoxaline-2,3-dione; CT, cycle threshold; ctrl, control; D-APV, D-2-amino-5-pho
Cannabinoid receptor antagonists and fatty acids alter endocannabinoid system gene expression and COX activity
Keywords: CB1، گیرنده کانابینوئید 1; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; NAPE-PLD, N-acyl phosphatidylethanolamine phospholipase D; FAAH, fatty acid amide hydrolase; DAGL-α, diacylglycerol lipase α; DAGL-ß, diacylglycerol lipase β; NF-κB, nuclear factor kappa-light-chai
Cannabinoids increase lung cancer cell lysis by lymphokine-activated killer cells via upregulation of ICAM-1
Keywords: CB1، گیرنده کانابینوئید 1; AM-251, N-(piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide; AM-630, (6-iodo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl)(4-methoxyphenyl)methanone; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2;
Selective CB2 receptor activation ameliorates EAE by reducing Th17 differentiation and immune cell accumulation in the CNS
Keywords: CB1، گیرنده کانابینوئید 1; APC, antigen-presenting cell; BBB, blood brain barrier; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CNS, central nervous system; DC, dendritic cell; EAE, experimental autoimmune encephalomyelitis; FACS, fluorescence activated cell sorter; LP
Identification of raloxifene as a novel CB2 inverse agonist
Keywords: CB1، گیرنده کانابینوئید 1; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; GPCR, G protein-coupled receptor; FDA, food and drug administration; HTRF, homogenous time-resolved fluorescenceCannabinoid receptor; Inverse agonist; Drug repurposing; Raloxifene; Osteoporosis
The role of CB1 in immune modulation by cannabinoids
Keywords: CB1، گیرنده کانابینوئید 1; 2-AG, 2-arachidonyl-glycerol; ACEA, arachidonyl-2′-chlorethanylamide; ACPA, arachidonylcyclopropylamide; AEA, arachidonylethanolamide; AP-1, activator protein-1; APC, antigen presenting cell; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CD, c
Alterations in endocannabinoid tone following chemotherapy-induced peripheral neuropathy: Effects of endocannabinoid deactivation inhibitors targeting fatty-acid amide hydrolase and monoacylglycerol lipase in comparison to reference analgesics following c
Keywords: CB1، گیرنده کانابینوئید 1; 2-AG, 2-arachidonoyl glycerol; AEA, anandamide; ANOVA, analysis of variance; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CNS, central nervous system; COX-2, cyclooxygenase-2; Δ9-THC, delta 9-tetrahydrocannabinol; DMSO, dimethylsulfoxide; DRG
Mastering tricyclic ring systems for desirable functional cannabinoid activity
Keywords: CB1، گیرنده کانابینوئید 1; Cannabinoid; CB2; GPCR; Neuropathic pain; Carbazole; CB1BSA, bovine serum albumin; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; EC50, half maximal effective concentration; EDTA, ethylenediaminetetraacetic acid; GTP, guanosine-5′-triphosphate;
The CB2-preferring agonist JWH015 also potently and efficaciously activates CB1 in autaptic hippocampal neurons
Keywords: CB1، گیرنده کانابینوئید 1; 2-AG, 2-arachidonoylglycerol; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; JWH015, (2-methyl-1-propyl-1H-indol-3-yl)-1-naphthalenylmethanone; Δ9-THC, tetrahydrocannabinol; SR141716 (aka Rimonabant), 5-(4-chlorophenyl)-1-(2′,4-dichloro-phenyl)
Hind limb suspension and long-chain omega-3 PUFA increase mRNA endocannabinoid system levels in skeletal muscle
Keywords: CB1، گیرنده کانابینوئید 1; 2-AG, 2-arachidonylgycerol; AA, arachidonic acid; AEA, anandamide; AMPK, AMP-activated protein kinase; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; DAGL, diacylglycerol; DHA, docosahexaenoic acid; DXA, dual-energy X-ray absorptiometry; EC, en
Cannabinoid receptors: nomenclature and pharmacological principles
Keywords: CB1، گیرنده کانابینوئید 1; abn-CBD, Abnormal cannabidiol; ACEA, Arachidonyl-2′-chlorethylamide; AEA, N-arachidonoyl ethanolamide, a.k.a. anandamide; 2-AG, 2-arachidonoyl glycerol; CB1, Cannabinoid receptor 1; CB2, Cannabinoid receptor 2; CGRP, Calcitonin gene-related peptide; EC50,
Altered calcium regulation by thermosensitive transient receptor potential channels in etoposide-resistant WERI-Rb1 retinoblastoma cells
Keywords: CB1، گیرنده کانابینوئید 1; human retinoblastoma; etoposide; transient receptor potential channels; calcium; cannabinoid receptor; planar patch-clamp techniqueRB, retinoblastmoma; TRPV, transient receptor potential vanilloid; CB1, cannabinoid receptor 1; RuR, ruthenium-red; 2-APB, 2
Cytotoxicity of synthetic cannabinoids found in “Spice” products: The role of cannabinoid receptors and the caspase cascade in the NG 108-15 cell line
Keywords: CB1، گیرنده کانابینوئید 1; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; DAPI, 4′,6-diamino-2-phenylindole; DMSO, dimethyl sulfoxide; DMEM, Dulbecco's modified Eagle's medium; FLICA, fluorescent labeled inhibitor of caspases; HAT, hypoxanthine, aminopterin and thymidine
Distribution patterns of cannabinoid CB1 receptors in the hippocampus of APPswe/PS1ΔE9 double transgenic mice
Keywords: CB1، گیرنده کانابینوئید 1; AD, Alzheimer's Disease; Aβ, amyloid beta; APP, amyloid precursor protein; AEA, Arachidonylethanolamide; 2-AG, 2-arachidonylglycerol; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CNS, central nervous system; dtg, double transgenic; GFAP, glia
The environment and susceptibility to schizophrenia
Keywords: CB1، گیرنده کانابینوئید 1; BMI, body mass index; CB1, cannabinoid receptor 1; CHDS, Child Health and Development Study; CMV, cytomegalovirus; CNS, central nervous system; CNVs, copy number variants; COMT, catechol-O-methyl transferase; CPP, Collaborative Perinatal Project; CRH, cor
Altered regulation of glutamate release and decreased functional activity and expression of GLT1 and GLAST glutamate transporters in the hippocampus of adolescent rats perinatally exposed to Δ9-THC
Keywords: CB1، گیرنده کانابینوئید 1; CB1, cannabinoid receptor 1; Δ9-THC, Δ9-tetrahydrocannabinol; Δ9-THC rats, 40-day-old rats perinatally exposed to Δ9-THC; EAAC1, excitatory amino acid carrier 1; GD, gestation day; GFAP, glial fibrillary acidic protein; GLAST, glutamate/aspartate transpor
Cannabinoid receptor activation reduces TNFα-Induced surface localization of AMPAR-type glutamate receptors and excitotoxicity
Keywords: CB1، گیرنده کانابینوئید 1; AMPA receptor; Cannabinoid receptor; Excitotoxicity; Glutamate receptor; Neuroprotection2AG, 2-Arachidonoylglycerol; AMPARs, α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptors; ANA, anandamide; CB1, cannabinoid receptor 1; END, Excitotoxic Neu
Cannabinoid Receptor 1 trafficking and the role of the intracellular pool: Implications for therapeutics
Keywords: CB1، گیرنده کانابینوئید 1; AM, AM 251; CB1, Cannabinoid Receptor 1; CHO, Chinese hamster ovary-K1; CHX, cycloheximide; Con A, Concanavalin A; D1, Dopamine Receptor 1; DMEM, Dulbecco's Modified Eagle Medium; eCB, endocannabinoid; ER, endoplasmic reticulum; FBS, fetal bovine serum; G
The paradoxical role of the transient receptor potential vanilloid 1 receptor in inflammation
Keywords: CB1، گیرنده کانابینوئید 1; TRPV1; Sensory nerves; Pain; Inflammation; NeuropeptidesACD, allergic contact dermatitis; AEA, anandamide, N-arachidonyl-ethanolamine; BrdU, Bromodeoxyridine; C-terminus, carboxy-terminus; CaM, calmodulin; CB1, cannabinoid receptor 1; CCI, chronic constri
Tuberoinfundibular peptide of 39 residues (TIP39) signaling modulates acute and tonic nociception
Keywords: CB1، گیرنده کانابینوئید 1; BLA, basolateral amygdaloid nucleus; CB1, cannabinoid receptor 1; FAAH, fatty acid amide hydrolase; HYWH, Histidine3-Tyrosine4-Tryptophan5-Histidine6-TIP39; icv, intracerebroventricular; ip, intraperitoneal; MPL, medial paralemniscal nucleus; PAG, periaqu
The discovery of central monoamine neurons gave volume transmission to the wired brain
Keywords: CB1، گیرنده کانابینوئید 1; A1, adenosine receptor 1; A2A, adenosine receptor 2A; 2-AG, sn-2-arachidonoylglycerol; CA, catecholamine; CB1, cannabinoid receptor 1; CNS, central nervous system; CSF, cerebrospinal fluid; cGMP, cyclic guanosine monophosphate; DA, dopamine; D1, dopamine
Cannabinoids inhibit insulin secretion and cytosolic Ca2+ oscillation in islet β-cells via CB1 receptors
Keywords: CB1، گیرنده کانابینوئید 1; AEA, arachidonylethanolamide (anandamide); CB1, cannabinoid receptor 1; ACPA, arachidonylcyclopropylamide; ACEA, arachidonyl-2-chloroethylamide (ACEA); [Ca2+]i, cytosolic Ca2+ concentrationCannabinoids; CB1 receptor; Insulin; Pancreatic β-cell; Calcium os
Cannabinoid receptor stimulation is anti-inflammatory and improves memory in old rats
Keywords: CB1، گیرنده کانابینوئید 1; Δ9-THC, Δ9-tetrahydrocannabinol; aCSF, artificial cerebral spinal fluid; AD, Alzheimer's disease; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CBr, cannabinoid receptors; DG, dentate gyrus; EC, entorhinal cortex; LPS, lipopolysaccharide; NMDA
Localization of CB1 cannabinoid receptor mRNA in the brain of the chick (Gallus domesticus)
Keywords: CB1، گیرنده کانابینوئید 1; CB, Cannabinoid; CB1, Cannabinoid Receptor 1; IHC, immunohistochemistry; ISH, in situ hybridization; ROI, region of interestAvian; Comparative anatomy; Tectum; Striatum; Sensory system
BfCBR: A cannabinoid receptor ortholog in the cephalochordate Branchiostoma floridae (Amphioxus)
Keywords: CB1، گیرنده کانابینوئید 1; bp, base pair(s); BLAST, Basic Local Alignment Search Tool; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; BfCBR, Branchiostoma floridae cannabinoid receptor; CiCBR, Ciona intestinalis cannabinoid receptor; Mb, megabase(s); PCR, polymerase chai
Anti-inflammatory property of the cannabinoid agonist WIN-55212-2 in a rodent model of chronic brain inflammation
Keywords: CB1، گیرنده کانابینوئید 1; cannabinoid receptors; inflammation; activated microglia; Alzheimer’s disease; LPS; spatial memoryaCSF, artificial cerebrospinal fluid; AD, Alzheimer’s disease; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CBr, cannabinoid receptors; DG, dent
Coevolution between cannabinoid receptors and endocannabinoid ligands
Keywords: CB1، گیرنده کانابینوئید 1; ABHD4, abhydrolase domain-containing protein 4; AEA, anandamide; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; COX2, cyclooxygenase 2; DAGLα, diacylglycerol lipase alpha; DAGLβ, diacylglycerol lipase beta; FAAH, fatty acid amide hydrolase; ML,
Anandamide inhibits Cdk2 and activates Chk1 leading to cell cycle arrest in human breast cancer cells
Keywords: CB1، گیرنده کانابینوئید 1; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; Met-F-AEA, 2-methyl-arachidonoyl-2′-F-ethylamide; Rb, retinoblastoma; Cdk, cyclin dependent kinase; CKIs, cdk inhibitors; HU, hydroxyureaEndocannabinoids; Chk1; Cyclin dependent kinase 2; Breast ca
The synthetic cannabinoid WIN 55,212-2 increases COX-2 expression and PGE2 release in murine brain-derived endothelial cells following Theiler's virus infection
Keywords: CB1، گیرنده کانابینوئید 1; 2-AG, 2-arachidonoyl glicerol; Abn-CBD, abnormal cannabidiol; AEA, anandamide; CB, cannabinoid; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; COX-2, cyclooxygenase-2; IL-1β, interleukin-1 beta; IL-12, interleukin-12; LDH, lactate dehydrogenase
Cannabinoid CB2 receptors: Immunohistochemical localization in rat brain
Keywords: CB1، گیرنده کانابینوئید 1; CB2, cannabinoid receptor 2; CB1, cannabinoid receptor 1; Cnr, cannabinoid receptor; Cnrs, cannabinoid receptors; EPCS, endocannabinoid physiological control system; eCBs, endocannabinoidsCB2 cannabinoid receptor; Brain; Immunohistochemistry; CB2 polyclon