Keywords: CB2، گیرنده کانابینوئید 2; 2-AG, 2-arachidonoylglycerol; ALI, air–liquid interface; ANOVA, analysis of variance; ATCC, American Type Culture Collection; BALF, bronchioalveolar lavage fluid; CB1 receptor, cannabinoid receptor 1; CB2, cannabinoid receptor 2; COPD, chronic obstructive
مقالات ISI CB2، گیرنده کانابینوئید 2 (ترجمه نشده)
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Keywords: CB2، گیرنده کانابینوئید 2; AEA, anandamide; AG, 2-arachidonoyl glycerol; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CB receptor, cannabinoid receptor; FAAH, fatty acid amide hydrolase; NM, nitrogen mustard; OEA, oleyolethanolamide; PEA, palmitoylethanolamide; PPARα,
Keywords: CB2، گیرنده کانابینوئید 2; AEA, arachidonoyl ethanolamide; 2-AG, 2-arachidonoylglycerol; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; FAAH, fatty acid amide hydrolase; FLS, fibroblastlike synoviocyte; IFN, interferon; IL, interleukin; MMP, matrix metalloproteinase; RA,
Pyrazole antagonists of the CB1 receptor with reduced brain penetration
Keywords: CB2، گیرنده کانابینوئید 2; BBB, blood–brain barrier; BOP, benzotriazol-1-yl-oxytris(dimethylamino)phosphonium hexafluorophosphate; CB, cannabinoid receptors; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CHO-K1, Chinese hamster ovary cells; CMA 80, 80% chloroform, 18% m
Discovery of novel Tetrahydrobenzo[b]thiophene and pyrrole based scaffolds as potent and selective CB2 receptor ligands: The structural elements controlling binding affinity, selectivity and functionality
Keywords: CB2، گیرنده کانابینوئید 2; CB2 selective ligands; CB2 agonist; CB2 inverse agonist; CannabinoidsCB1, Cannabinoid receptor 1; CB2, Cannabinoid receptor 2; DIPEA, N,N-Diisopropylethylamine; EDC, 1-Ethyl-3-(3’-dimethylamino)carbodiimide HCl salt; HATU, 1-[Bis(dimethylamino)methylene]-
Enterocyte fatty acid-binding proteins (FABPs): Different functions of liver and intestinal FABPs in the intestine
Keywords: CB2، گیرنده کانابینوئید 2; Fatty acid-binding protein; Fatty acid; Intestine; Lipid; LFABP; IFABP2-AG, 2-arachidonoylglycerol; AEA, arachidinoylethanolamide; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; FA, fatty acid; FXR, farnesoid X receptor; IFABP, intestinal fatty
Endocannabinoid metabolism by cytochrome P450 monooxygenases
Keywords: CB2، گیرنده کانابینوئید 2; 2-AG, 2-arachidonylglycerol; AEA, anandamide; AA, arachidonic acid; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CNS, central nervous system; COX, cyclooxygenase; CYP, cytochrome P450; DAG, diacylglycerol; DHET, dihydroxyeicosatrienoic acid;
Cannabinoid receptor antagonists and fatty acids alter endocannabinoid system gene expression and COX activity
Keywords: CB2، گیرنده کانابینوئید 2; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; NAPE-PLD, N-acyl phosphatidylethanolamine phospholipase D; FAAH, fatty acid amide hydrolase; DAGL-α, diacylglycerol lipase α; DAGL-ß, diacylglycerol lipase β; NF-κB, nuclear factor kappa-light-chai
Cannabinoids increase lung cancer cell lysis by lymphokine-activated killer cells via upregulation of ICAM-1
Keywords: CB2، گیرنده کانابینوئید 2; AM-251, N-(piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide; AM-630, (6-iodo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl)(4-methoxyphenyl)methanone; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2;
Selective CB2 receptor activation ameliorates EAE by reducing Th17 differentiation and immune cell accumulation in the CNS
Keywords: CB2، گیرنده کانابینوئید 2; APC, antigen-presenting cell; BBB, blood brain barrier; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CNS, central nervous system; DC, dendritic cell; EAE, experimental autoimmune encephalomyelitis; FACS, fluorescence activated cell sorter; LP
Identification of raloxifene as a novel CB2 inverse agonist
Keywords: CB2، گیرنده کانابینوئید 2; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; GPCR, G protein-coupled receptor; FDA, food and drug administration; HTRF, homogenous time-resolved fluorescenceCannabinoid receptor; Inverse agonist; Drug repurposing; Raloxifene; Osteoporosis
The role of CB1 in immune modulation by cannabinoids
Keywords: CB2، گیرنده کانابینوئید 2; 2-AG, 2-arachidonyl-glycerol; ACEA, arachidonyl-2′-chlorethanylamide; ACPA, arachidonylcyclopropylamide; AEA, arachidonylethanolamide; AP-1, activator protein-1; APC, antigen presenting cell; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CD, c
Alterations in endocannabinoid tone following chemotherapy-induced peripheral neuropathy: Effects of endocannabinoid deactivation inhibitors targeting fatty-acid amide hydrolase and monoacylglycerol lipase in comparison to reference analgesics following c
Keywords: CB2، گیرنده کانابینوئید 2; 2-AG, 2-arachidonoyl glycerol; AEA, anandamide; ANOVA, analysis of variance; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CNS, central nervous system; COX-2, cyclooxygenase-2; Δ9-THC, delta 9-tetrahydrocannabinol; DMSO, dimethylsulfoxide; DRG
Mastering tricyclic ring systems for desirable functional cannabinoid activity
Keywords: CB2، گیرنده کانابینوئید 2; Cannabinoid; CB2; GPCR; Neuropathic pain; Carbazole; CB1BSA, bovine serum albumin; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; EC50, half maximal effective concentration; EDTA, ethylenediaminetetraacetic acid; GTP, guanosine-5′-triphosphate;
The CB2-preferring agonist JWH015 also potently and efficaciously activates CB1 in autaptic hippocampal neurons
Keywords: CB2، گیرنده کانابینوئید 2; 2-AG, 2-arachidonoylglycerol; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; JWH015, (2-methyl-1-propyl-1H-indol-3-yl)-1-naphthalenylmethanone; Δ9-THC, tetrahydrocannabinol; SR141716 (aka Rimonabant), 5-(4-chlorophenyl)-1-(2′,4-dichloro-phenyl)
Hind limb suspension and long-chain omega-3 PUFA increase mRNA endocannabinoid system levels in skeletal muscle
Keywords: CB2، گیرنده کانابینوئید 2; 2-AG, 2-arachidonylgycerol; AA, arachidonic acid; AEA, anandamide; AMPK, AMP-activated protein kinase; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; DAGL, diacylglycerol; DHA, docosahexaenoic acid; DXA, dual-energy X-ray absorptiometry; EC, en
Cannabinoid receptors: nomenclature and pharmacological principles
Keywords: CB2، گیرنده کانابینوئید 2; abn-CBD, Abnormal cannabidiol; ACEA, Arachidonyl-2′-chlorethylamide; AEA, N-arachidonoyl ethanolamide, a.k.a. anandamide; 2-AG, 2-arachidonoyl glycerol; CB1, Cannabinoid receptor 1; CB2, Cannabinoid receptor 2; CGRP, Calcitonin gene-related peptide; EC50,
Cytotoxicity of synthetic cannabinoids found in “Spice” products: The role of cannabinoid receptors and the caspase cascade in the NG 108-15 cell line
Keywords: CB2، گیرنده کانابینوئید 2; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; DAPI, 4′,6-diamino-2-phenylindole; DMSO, dimethyl sulfoxide; DMEM, Dulbecco's modified Eagle's medium; FLICA, fluorescent labeled inhibitor of caspases; HAT, hypoxanthine, aminopterin and thymidine
Distribution patterns of cannabinoid CB1 receptors in the hippocampus of APPswe/PS1ΔE9 double transgenic mice
Keywords: CB2، گیرنده کانابینوئید 2; AD, Alzheimer's Disease; Aβ, amyloid beta; APP, amyloid precursor protein; AEA, Arachidonylethanolamide; 2-AG, 2-arachidonylglycerol; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CNS, central nervous system; dtg, double transgenic; GFAP, glia
Cannabinoid receptor stimulation is anti-inflammatory and improves memory in old rats
Keywords: CB2، گیرنده کانابینوئید 2; Δ9-THC, Δ9-tetrahydrocannabinol; aCSF, artificial cerebral spinal fluid; AD, Alzheimer's disease; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CBr, cannabinoid receptors; DG, dentate gyrus; EC, entorhinal cortex; LPS, lipopolysaccharide; NMDA
BfCBR: A cannabinoid receptor ortholog in the cephalochordate Branchiostoma floridae (Amphioxus)
Keywords: CB2، گیرنده کانابینوئید 2; bp, base pair(s); BLAST, Basic Local Alignment Search Tool; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; BfCBR, Branchiostoma floridae cannabinoid receptor; CiCBR, Ciona intestinalis cannabinoid receptor; Mb, megabase(s); PCR, polymerase chai
Anti-inflammatory property of the cannabinoid agonist WIN-55212-2 in a rodent model of chronic brain inflammation
Keywords: CB2، گیرنده کانابینوئید 2; cannabinoid receptors; inflammation; activated microglia; Alzheimer’s disease; LPS; spatial memoryaCSF, artificial cerebrospinal fluid; AD, Alzheimer’s disease; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; CBr, cannabinoid receptors; DG, dent
Coevolution between cannabinoid receptors and endocannabinoid ligands
Keywords: CB2، گیرنده کانابینوئید 2; ABHD4, abhydrolase domain-containing protein 4; AEA, anandamide; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; COX2, cyclooxygenase 2; DAGLα, diacylglycerol lipase alpha; DAGLβ, diacylglycerol lipase beta; FAAH, fatty acid amide hydrolase; ML,
Anandamide inhibits Cdk2 and activates Chk1 leading to cell cycle arrest in human breast cancer cells
Keywords: CB2، گیرنده کانابینوئید 2; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; Met-F-AEA, 2-methyl-arachidonoyl-2′-F-ethylamide; Rb, retinoblastoma; Cdk, cyclin dependent kinase; CKIs, cdk inhibitors; HU, hydroxyureaEndocannabinoids; Chk1; Cyclin dependent kinase 2; Breast ca
The synthetic cannabinoid WIN 55,212-2 increases COX-2 expression and PGE2 release in murine brain-derived endothelial cells following Theiler's virus infection
Keywords: CB2، گیرنده کانابینوئید 2; 2-AG, 2-arachidonoyl glicerol; Abn-CBD, abnormal cannabidiol; AEA, anandamide; CB, cannabinoid; CB1, cannabinoid receptor 1; CB2, cannabinoid receptor 2; COX-2, cyclooxygenase-2; IL-1β, interleukin-1 beta; IL-12, interleukin-12; LDH, lactate dehydrogenase
Cannabinoid CB2 receptors: Immunohistochemical localization in rat brain
Keywords: CB2، گیرنده کانابینوئید 2; CB2, cannabinoid receptor 2; CB1, cannabinoid receptor 1; Cnr, cannabinoid receptor; Cnrs, cannabinoid receptors; EPCS, endocannabinoid physiological control system; eCBs, endocannabinoidsCB2 cannabinoid receptor; Brain; Immunohistochemistry; CB2 polyclon