
3,4-Diaza-bicyclo[4.1.0]hept-4-en-2-one phenoxypropylamine analogs of irdabisant (CEP-26401) as potent histamine-3 receptor inverse agonists with robust wake-promoting activity
Keywords: Histamine H3 receptor; H3 inverse agonist; Irdabisant; CEP-26401; Pyridazin-3-one; Sleep-wake;