Keywords: Permeapad®; Lipid based formulations; Lipolysis; Permeability; Cinnarizine; In vitro; SNEDDS; Calcein (PubChem CID 65079); Calcium chloride (PubChem CID 5284359); Cinnarizine (PubChem CID 1547484); Ethanol (PubChem CID 702); Oleic acid (PubChem CID 44563
مقالات ISI (ترجمه نشده)
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Keywords: Lipophilic weak base; Luminal concentration; Re-dissolution; Supersaturation; AUCduodenum; area under the duodenal concentration-time curve; BA; bioavailability; BCS; Biopharmaceutics Classification System; CNZ; cinnarizine; DSC; differential scanning cal
Keywords: SNEDDS; Food effect; Low soluble compounds; Humans; Enabling formulations; Oral absorption; Cinnarizine
Keywords: Cyclodextrins; Danazol; Cinnarizine; In vivo; Rats; Complexation;
Keywords: Cinnarizine; Nanosuspension; Sonoprecipitation; Optimization; Bioavailability
Keywords: Cinnarizine; Dimenhydrinate; Dual wavelength; Ratio difference; Constant center; Mean centering;
Keywords: children; migraine; cinnarizine; placebo; clinical trial
Keywords: Solid solubility; Supercritical carbon dioxide; Cinnarizine; Pentoxifylline; Piracetam
Keywords: Spectrophotometry; Cinnarizine; Domperidone; Area under curve; Dual wavelength; Pharmaceutical formulation;
Keywords: Vestibular evoked myogenic potentials; Scopolamine; Cinnarizine; Dimenhydrinate; Seasickness; Motion sickness
Small molecules bind human mTOR protein and inhibit mTORC1 specifically
Keywords: mTOR; mTORC1; mTORC2; Piperazine; Cinnarizine; Hydroxyzine; Cancer;
Exploring the feasibility of the use of biopolymers as a carrier in the formulation of amorphous solid dispersions - Part I: Gelatin
Keywords: Carbamazepine (2554); Cinnarizine (1547484); Darunavir (Ethanolate: 23725083); Fenofibrate (3339); Griseofulvin (441140); Indomethacin (3715); Itraconazole (55283); Ketoconazole (456201); Naproxen (156391); Nifedipine (4485); Ritonavir (392622); Diazepam
Simultaneous determination of Dimenhydrinate, Cinnarizine and Cinnarizine impurity by TLC and HPLC chromatographic methods
Keywords: Dimenhydrinate; Cinnarizine; 1-(Diphenylmethyl) piperazine); TLC; HPLC;
Research paperSolution or suspension - Does it matter for lipid based systems? In vivo studies of chase dosing lipid vehicles with aqueous suspensions of a poorly soluble drug
Keywords: Lipid based formulation; Suspension; Solution; Labrafil M2125CS; Danazol; Cinnarizine; Halofantrine;
Research paperEudragit® RL as a stabilizer for supersaturation and a substrate for nanocrystal formation
Keywords: Solid dispersions; Eudragit RL; Supersaturation; Nanocrystals; Thermal analysis; X-ray powder diffraction; Spray drying; INDO; indomethacin; NAP; naproxen; CINN; cinnarizine; ERL; Eudragit RL; PVP; polyvinylpyrrolidone; Tg; glass transition temperature; m
Validated HPTLC method for the simultaneous determination of cinnarizine and dimenhydrinate in their combined dosage form
Keywords: Cinnarizine; Dimenhydrinate; HPTLC; Tablets dosage form
Development of normalized spectra manipulating spectrophotometric methods for simultaneous determination of Dimenhydrinate and Cinnarizine binary mixture
Keywords: Dimenhydrinate; Cinnarizine; Normalized spectra; Simultaneous constant center; Simultaneous derivative ratio; Ratio H-point standard addition method
Histamine H1-receptor antagonists against Leishmania (L.) infantum: an in vitro and in vivo evaluation using phosphatidylserine-liposomes
Keywords: Leishmania; Histamine; H1 antagonist; Liposomes; Cinnarizine; Therapy;
Oral bioavailability of cinnarizine in dogs: Relation to SNEDDS droplet size, drug solubility and in vitro precipitation
Keywords: Oral delivery; Lipolysis; Bioavailability; Self-nanoemulsifying drug delivery systems; Cinnarizine
Is the amorphous fraction of a dried nanosuspension caused by milling or by drying? A case study with Naproxen and Cinnarizine
Keywords: Amorphous; Nanocrystal; Media milling; Naproxen; Cinnarizine; HPMC
Quantification of cyclizine and norcyclizine in human plasma by liquid chromatography–tandem mass spectrometry (LC–MS/MS)
Keywords: Cyclizine; Norcyclizine; Cinnarizine; LC–MS/MS; Plasma; Human
Quantitative determination of pimozide in human plasma by liquid chromatography–mass spectrometry and its application in a bioequivalence study
Keywords: Pimozide; Cinnarizine; LC–ESI/MS; Determination; Bioequivalence
Effect of route of administration on the pharmacokinetics and toxicokinetics of cinnarizine in dogs
Keywords: Cinnarizine; Pharmacokinetics; Toxicokinetics; Intravenous injection
Pharmacokinetics, tissue distribution and safety of cinnarizine delivered in lipid emulsion
Keywords: Cinnarizine; Lipid emulsion; Pharmacokinetics; Tissue distribution; Safety
Solution calorimetry as an alternative approach for dissolution testing of nanosuspensions
Keywords: Nanosuspensions; Dissolution rate; Solution calorimetry; Naproxen; Cinnarizine
Precipitation of a Poorly Soluble Model Drug during In Vitro Lipolysis: Characterization and Dissolution of the Precipitate
Keywords: in vitro lipolysis; self-microemulsifying drug delivery system (SMEDDS); cinnarizine; Biopharmaceutics Classification System (BCS) class 2 drugs; precipitation; dissolution rate; triacylglycerides; digestion; X-ray powder diffraction (XRPD); polarized lig
Voltammetric oxidation and determination of cinnarizine at glassy carbon electrode modified with multi-walled carbon nanotubes
Keywords: Cinnarizine; Multi-walled carbon nanotubes; Voltammetry; Modified electrode
Formulation, stability and degradation kinetics of intravenous cinnarizine lipid emulsion
Keywords: Cinnarizine; Formulation; Intravenous lipid emulsion; Stability; Degradation kinetic
Determination of mianserin in human plasma by high performance liquid chromatography–electrospray ionization mass spectrometry (HPLC–ESI/MS): Application to a bioequivalence study in Chinese volunteers
Keywords: Mianserin; Cinnarizine; LC–ESI/MS; Determination; Bioequivalence
Method development and validation for the simultaneous determination of cinnarizine and co-formulated drugs in pharmaceutical preparations by capillary electrophoresis
Keywords: Capillary electrophoresis; Cinnarizine; Domperidone; Nicergoline; Co-formulated tablets
A lipid-based liquid crystalline matrix that provides sustained release and enhanced oral bioavailability for a model poorly water soluble drug in rats
Keywords: Poorly water soluble drug; Lipid formulation; Liquid crystal; Cinnarizine; Bioavailability
The effect of cinnarizine and cocculus indicus on simulator sickness
Keywords: Motion sickness; Simulator sickness; Postural balance; Cinnarizine; Cocculus indicus; Sleepiness