Keywords: دی هیدروپیریمیدین ها; Dihydropyrimidines; Imidazoles; Antitubercular activity; Mycobacterium tuberculosis dihydrofolate reductase inhibitors; Molecular docking; Cytotoxicity
مقالات ISI دی هیدروپیریمیدین ها (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: دی هیدروپیریمیدین ها; Acetylcholinesterase; Butyrylcholinesterase; Dihydropyrimidines; Blood brain barrier; Dual binding site;
Keywords: دی هیدروپیریمیدین ها; Antimycobacterial; Dihydropyrimidines; Heteroaryl aldehyde; Mycobacterium tuberculosis; CIP and H37Rv strain;
Design, synthesis, in vitro Evaluation and docking studies on dihydropyrimidine-based urease inhibitors
Keywords: دی هیدروپیریمیدین ها; Urease inhibitors; Structure-based drug designing; In silico pharmacokinetics; Dihydropyrimidines; Tautomerism;
Synthesis of new N3-substituted dihydropyrimidine derivatives as L-/T- type calcium channel blockers
Keywords: دی هیدروپیریمیدین ها; L-type calcium channel blockers; T-type calcium channel blockers; Whole patch clamp technique; Dihydropyrimidines; Dihydropyridines; Cav1.2; Cav3.2;
Synthesis and biological evaluation of novel N3-substituted dihydropyrimidine derivatives as T-type calcium channel blockers and their efficacy as analgesics in mouse models of inflammatory pain
Keywords: دی هیدروپیریمیدین ها; Pain; Calcium channels; T-type calcium channel blockers; Whole patch clamp technique; Dihydropyrimidines; 1,4-Dihydropyridines;
Preparation of dihydrotetrazolo[1,5-a]pyrimidine derivatives from Biginelli 3,4-dihydropyrimidine-2-thiones
Keywords: دی هیدروپیریمیدین ها; Dihydropyrimidines; Tetrazole; DHPM scaffold; Monastrol; Biological activities;
Synthesis of pyrazolo[3,4-d]-4,5-dihydropyrimidin-6-ones
Keywords: دی هیدروپیریمیدین ها; Aldehydes; Aminopyrazoles; Dihydropyrimidines; Ureas; Chlorotrimethylsilane;
Convenient synthesis of 1-aryl-9H-β-carboline-3-carbaldehydes and their transformation into dihydropyrimidinone derivatives by Biginelli reaction
Keywords: دی هیدروپیریمیدین ها; Nitrogen heterocycles; β-Carbolines; Dihydropyrimidines; Biginelli reaction;
Structure based virtual screening-driven identification of monastrol as a potent urease inhibitor
Keywords: دی هیدروپیریمیدین ها; Urease inhibitors; Structure-based virtual screening; Monastrol; Dihydropyrimidines; Docking
A facile one-pot synthesis of 2-thioxo-dihydropyrimidines and polyfunctionalized pyran derivatives as mimics of novel calcium channel modulators
Keywords: دی هیدروپیریمیدین ها; Piperidinylamide; Dihydropyrimidines; Polyfunctionalized pyrans; Multi-component reaction; Calcium channel modulator;
Synthesis and in vitro anticancer and antitubercular activity of diarylpyrazole ligated dihydropyrimidines possessing lipophilic carbamoyl group
Keywords: دی هیدروپیریمیدین ها; Dihydropyrimidines; 1,3-Diarylpyrazoles; Multicomponent Reaction; Anticancer; Antitubercular
DFT study on mechanism of the classical Biginelli reaction
Keywords: دی هیدروپیریمیدین ها; Biginelli reaction; Dihydropyrimidines; Transition state; DFT study
Integration of high speed microwave chemistry and a statistical 'design of experiment' approach for the synthesis of the mitotic kinesin Eg5 inhibitor monastrol
Keywords: دی هیدروپیریمیدین ها; Dihydropyrimidines; Multicomponent reaction; Design of experiments; Microwave irradiation; Heterocycles;
Synthesis of 2-sulfanyl-6-methyl-1,4-dihydropyrimidines as a new class of antifilarial agents
Keywords: دی هیدروپیریمیدین ها; Dihydropyrimidines; 1,4-Dihydropyrimidines; Antifilarial; Brugia malayi; Tetrabutyl ammonium bromide
Biorenewable and mercaptoacetylating building blocks in the Biginelli reaction: synthesis of thiosugar-annulated dihydropyrimidines
Keywords: دی هیدروپیریمیدین ها; Biginelli reaction; Stereoselective synthesis; Dihydropyrimidines; Microwaves; 1,3-Oxathiolan-5-one; Solvent-free;
Transamidation reactions of 2-(2-sulfonylguanidino)acetamides
Keywords: دی هیدروپیریمیدین ها; Transamidation; Guanidines; Acetamides; Dihydropyrimidines; Imidazolidinones;