Keywords: Whey protein; In vitro digestion; Bioactive peptide; Glucagon-like peptide-1; Dipeptidyl peptidase IV inhibitor; Antioxidant activity; α-LA; α-lactalbumin; β-LG; β-lactoglobulin; ABAP; 2,2â²-azobis(2-methylpropionamidine) dihydrochloride; AMC; H-Gly-
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Dipeptidyl peptidase IV (DPP-IV) inhibition prevents fibrosis in adipose tissue of obese mice
Keywords: Obesity; Fibrosis; Extracellular matrix; Dipeptidyl peptidase IV inhibitor; Vildagliptin; Neuropeptide Y;
Anagliptin inhibits neointimal hyperplasia after balloon injury via endothelial cell-specific modulation of SOD-1/RhoA/JNK signaling in the arterial wall
Keywords: Intimal hyperplasia; Dipeptidyl peptidase IV inhibitor; Oxidant species; Superoxide dismutase; Cell migration;
A study to evaluate the potential of an in silico approach for predicting dipeptidyl peptidase-IV inhibitory activity in vitro of protein hydrolysates
Keywords: In silico analysis; Dipeptidyl peptidase IV inhibitor; Dietary protein; Correlation analysis;
Synthesis and potent inhibitory activities of carboxybenzyl-substituted 8-(3-(R)-aminopiperidin-1-yl)-7-(2-chloro/cyanobenzyl)-3-methyl-3,7-dihydro-purine-2,6-diones as dipeptidyl peptidase IV (DPP-IV) inhibitors
Keywords: Diabetes; Dipeptidyl peptidase IV inhibitor; 3-Methyl-3,7-dihydro-purine-2,6-dione; Synthesis; Inhibitory activity
Dipeptidyl peptidase IV inhibitory peptides generated in Spanish dry-cured ham
Keywords: Dry-cured ham; Bioactive peptides; Dipeptidyl peptidase IV inhibitor; Type 2 diabetes;
A comparative study of the binding modes of recently launched dipeptidyl peptidase IV inhibitors in the active site
Keywords: Type 2 diabetes; Dipeptidyl peptidase IV inhibitor; X-ray co-crystal structure; Binding subsite;
Substituted piperidinyl glycinyl 2-cyano-4,5-methano pyrrolidines as potent and stable dipeptidyl peptidase IV inhibitors
Keywords: Piperidine; Pyrrolidine; Dipeptidyl peptidase IV inhibitor; Type 2 diabetes
Design, synthesis and primary activity of thiomorpholine derivatives as DPP-IV inhibitors
Keywords: Thiomorpholine; Dipeptidyl peptidase IV inhibitor; Synthesis; Structure–activity relationship; Oral glucose tolerance test
Synthesis, biological assay in vitro and molecular docking studies of new imidazopyrazinone derivatives as potential dipeptidyl peptidase IV inhibitors
Keywords: Dipeptidyl peptidase IV inhibitor; Imidazopyrazinone; Anti-diabetic agent; Molecular docking