Keywords: افزایش ریزش; Nanosuspension; Media milling; Dissolution enhancement; Spray drying; Lyophilization; Saturation solubility;
مقالات ISI افزایش ریزش (ترجمه نشده)
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Keywords: افزایش ریزش; Melt mixing; Solid dispersions; Soluplus; PVP; Poloxamer; Felodipine; Dissolution enhancement;
Keywords: افزایش ریزش; Silk sericin; Poorly soluble drugs; Binary dispersion; Solubility improvement; Dissolution enhancement;
Keywords: افزایش ریزش; AA; glacial acetic acid; APCC; amorphous precipitation in a crystalline carrier; ASD; amorphous solid dispersion; C-DXT; crystal solid dispersion of docetaxel in SA; BCS; biopharmaceutics classification system; CSD; crystal solid dispersion; CSS; crystall
Keywords: افزایش ریزش; Poorly water-soluble drug; Ionic liquids; Antisolvent crystallization; Dissolution enhancement;
Keywords: افزایش ریزش; Solvent-free; Mesoporous silica; Melt-absorption; Amorphous formulation; Dissolution enhancement;
Keywords: افزایش ریزش; Liquisolid; Dissolution enhancement; Leflunomide; SEDDS; BCS class II;
Keywords: افزایش ریزش; Mesoporous silica materials; Physico-chemical properties; Poorly water-soluble drugs; Dissolution enhancement; Oral bioavailability;
Keywords: افزایش ریزش; Nebivolol hydrochloride; Electrospinning; Nanofibers; Positron annihilation lifetime spectroscopy (PALS); Differential scanning calorimetry (DSC); Dissolution enhancement;
Keywords: افزایش ریزش; Centrifugal spinning; Microfiber; Amorphous solid dispersion; Sucrose; Poorly water soluble drug; Dissolution enhancement; Supersaturation;
Keywords: افزایش ریزش; Tadalafil; Soluplus®; High energy ball milling; Supercritical fluids; Glassy molecular alloys; Solid dispersions; Dissolution enhancement;
Keywords: افزایش ریزش; MPC polymer; Wet grinding; Dissolution enhancement; Poorly water-soluble; Ibuprofen;
Keywords: افزایش ریزش; Solid dispersions; Carbamazepin-gluconolactone; Dissolution enhancement; Eutectic mixtures; Mechanistic solid state analysis
Keywords: افزایش ریزش; Carvedilol; Cyclodextrin; Tartaric acid; Ionization process; Water soluble polymer; Dissolution enhancement
Jelly containing composite based on α-glucosyl stevia and polyvinylpyrrolidone: Improved dissolution property of curcumin
Keywords: افزایش ریزش; Curcumin; α-Glucosyl stevia; Polyvinylpyrrolidone K-30; Composite; Dissolution enhancement; Jelly formulation;
The potential of synergism between ultrasonic energy and Soluplus® as a tool for solubilization and dissolution enhancement of a poorly water soluble drug. A statistically based process optimization
Keywords: افزایش ریزش; Sonocrystallization; Soluplus®; Solubilization; Dissolution enhancement;
Stable and Fast-Dissolving Amorphous Drug Composites Preparation via Impregnation of Neusilin® UFL2
Keywords: افزایش ریزش; poorly water-soluble drug; mesoporous Neusilin®; impregnation; high drug-load; amorphous drug; stability; dissolution enhancement;
Study on effect of L-arginine on solubility and dissolution of Zaltoprofen: Preparation and characterization of binary and ternary cyclodextrin inclusion complexes
Keywords: افزایش ریزش; Ternary complex; Cyclodextrin; Dissolution enhancement; Inclusion complex; Solubility enhancement;
Encapsulation of boswellic acid with β- and hydroxypropyl-β-cyclodextrin: Synthesis, characterization, in vitro drug release and molecular modelling studies
Keywords: افزایش ریزش; Boswellic acid; Cyclodextrin; Inclusion complex; Dissolution enhancement;
Dissolution enhancement of griseofulvin from griseofulvin-sodium dodecyl sulfate discs investigated by UV imaging
Keywords: افزایش ریزش; Dissolution enhancement; Dissolution imaging; Griseofulvin; Poorly soluble drugs; Surfactant; UV imaging;
Microwave processed solid dispersions for enhanced dissolution of gemfibrozil using non-ordered mesoporous silica
Keywords: افزایش ریزش; Amorphous; Dissolution enhancement; Gemfibrozil; Microwave heating; Silica; Solid dispersion;
Liquisolid technique and its applications in pharmaceutics
Keywords: افزایش ریزش; Liquisolid technique; Dissolution enhancement; Poorly water-soluble drugs; Sustained release; pH variation; Photostability;
Solid state behavior of progesterone and its release from Neusilin US2 based liquisolid compacts
Keywords: افزایش ریزش; Progesterone; Neusilin US2; Liquisolid compact; Metastable polymorph; Dissolution enhancement; Progesterone (PubChem CID: 5994); Neusilin US2 (PubChem CID: 3084116); Syloid 244 FP (PubChem CID: 24261); Polysorbate 80 (PubChem CID: 5284448); Propylene glyc
AC and DC electrospinning of hydroxypropylmethylcellulose with polyethylene oxides as secondary polymer for improved drug dissolution
Keywords: افزایش ریزش; Electrospinning; Nanofibers; Hypromellose; Dissolution enhancement; Polyethylene oxide
High speed electrospinning for scaled-up production of amorphous solid dispersion of itraconazole
Keywords: افزایش ریزش; Electrospinning; Itraconazole; Amorphous solid dispersion; Scaling-up; Dissolution enhancement; Continuous nanoformulation;
Formulation and optimization of Embelin nanosuspensions using central composite design for dissolution enhancement
Keywords: افزایش ریزش; Embelin; Nanosuspension; Nanocrystal; Dissolution enhancement; Central composite design; Characterization studies
Self nano-emulsifying drug delivery system for Embelin: Design, characterization and in-vitro studies
Keywords: افزایش ریزش; Embelin; SNEDDS; Dissolution enhancement; Box-Behnken design; Characterization
Alternating current electrospinning for preparation of fibrous drug delivery systems
Keywords: افزایش ریزش; Electrospinning; Alternating current electrospinning; Dissolution enhancement; Poorly water-soluble drugs; Solid dispersion;
Tracking of crystalline-amorphous transition of carvedilol in rotary spun microfibers and their formulation to orodispersible tablets for in vitro dissolution enhancement
Keywords: افزایش ریزش; FTIR; X-ray diffractometry (XRD); Positron annihilation spectroscopy (PALS); Differential scanning calorimetry (DSC); Rotary-spun microfiber; Dissolution enhancement;
Amorphous formulations for dissolution and bioavailability enhancement of poorly soluble APIs
Keywords: افزایش ریزش; Amorphous formulation; Solid dispersion; Dissolution enhancement;
Amorphous isradipine nanosuspension by the sonoprecipitation method
Keywords: افزایش ریزش; Nanosuspension; Sonoprecipitation method; Crystallinity; Dissolution enhancement
Preformulation study of fiber formation and formulation of drug-loaded microfiber based orodispersible tablets for in vitro dissolution enhancement
Keywords: افزایش ریزش; High-speed rotary spinning; Microfibers; Hydroxypropyl cellulose; Orodispersible tablet; Dissolution enhancement;
Dissolution enhancement of Deflazacort using hollow crystals prepared by antisolvent crystallization process
Keywords: افزایش ریزش; Deflazacort; Antisolvent crystallization; Hollow crystal; Micronization; Dissolution enhancement;
Application of Plackett–Burman screening design for preparing glibenclamide nanoparticles for dissolution enhancement
Keywords: افزایش ریزش; Glibenclamide; Liquid antisolvent precipitation; Dissolution enhancement; Plackett–Burman screening design
Mesoporous silica based macromolecules for dissolution enhancement of Irbesartan drug using pre-adjusted pH method
Keywords: افزایش ریزش; Irbesartan; Silica-based microcapsules; Dissolution enhancement; Pre-adjusted pH method; Solid dispersion
New formulation approaches to improve solubility and drug release from fixed dose combinations: Case examples pioglitazone/glimepiride and ezetimibe/simvastatin
Keywords: افزایش ریزش; Fixed dose combination; Solubility improvement; Dissolution enhancement; Solid dispersions; Ternary comlexes
NoteNanocomposite formation between alpha-glucosyl stevia and surfactant improves the dissolution profile of poorly water-soluble drug
Keywords: افزایش ریزش; α-glucosyl stevia; Flurbiprofen; Surfactant; Dissolution enhancement; Nanocomposite;
The influence of supercritical carbon dioxide (SC-CO2) processing conditions on drug loading and physicochemical properties
Keywords: افزایش ریزش; Supercritical carbon dioxide; Mesoporous silica; Dissolution enhancement; Fenofibrate; Drug-loading; Poorly-water soluble; SBA-15;
α-Glucosyl hesperidin induced an improvement in the bioavailability of pranlukast hemihydrate using high-pressure homogenization
Keywords: افزایش ریزش; α-Glucosyl hesperidin; Pranlukast hemihydrate; High-pressure homogenization; Dissolution enhancement; Absorption enhancement
Transglycosylated stevia and hesperidin as pharmaceutical excipients: Dramatic improvement in drug dissolution and bioavailability
Keywords: افزایش ریزش; α-glucosyl hesperidin; α-glycosyltransferase treated stevia; Flurbiprofen; Probucol; Dissolution enhancement; Absorption enhancement
Carbamazepine-Loaded Porous Microspheres for Short-Term Sustained Drug Delivery
Keywords: افزایش ریزش; Carbamazepine; microspheres; re-precipitation; sustained release; dissolution enhancement;
Cogrinding as an approach to enhance dissolution rate of a poorly water-soluble drug (gliclazide)
Keywords: افزایش ریزش; Cogrinding; Solid dispersion; Gliclazide; Dissolution enhancement; X-ray diffraction; DSC; Carrier
A one-pot method to enhance dissolution rate of low solubility drug molecules using dispersion polymerization in supercritical carbon dioxide
Keywords: افزایش ریزش; Supercritical fluid; Drug release kinetics; Solid dispersion; Dissolution enhancement; Polymer microspheres
Intraorally fast-dissolving particles of a poorly soluble drug: Preparation and in vitro characterization
Keywords: افزایش ریزش; Solid dispersion; Solid solution; Dissolution enhancement; PVP; PEG; Amorphous
Development and optimization of solid dispersion containing pellets of itraconazole prepared by high shear pelletization
Keywords: افزایش ریزش; Itraconazole; Solid dispersion; Dissolution enhancement; High shear pelletization; Pellet characteristics; Central composite design
Effect of the melt granulation technique on the dissolution characteristics of griseofulvin
Keywords: افزایش ریزش; Griseofulvin; Melt granulation; PEG 3350; Gelucire 44/14; HPMC; Dissolution enhancement
Investigation of the release mechanism of a sparingly water-soluble drug from solid dispersions in hydrophilic carriers based on physical state of drug, particle size distribution and drug–polymer interactions
Keywords: افزایش ریزش; Felodipine; PVP; PEG; Solid dispersion; Sparingly soluble drugs; Dissolution enhancement
Enhancement of dissolution rate of poorly soluble active ingredients by supercritical fluid processes
Keywords: افزایش ریزش; Particle design; Supercritical fluid; Dissolution enhancement; Micronization; Nanoparticles; Microspheres;
Enhancement of dissolution rate of poorly-soluble active ingredients by supercritical fluid processes
Keywords: افزایش ریزش; Particle design; Supercritical fluid; Dissolution enhancement; Micronization; Nanoparticles; Microspheres;