
Design, synthesis, and biological evaluation of a series of bifunctional ligands of opioids/SSRIs
Keywords: AcOH, acetic acid; Boc, tert-butoxycarbonyl; CHO, Chinese hamster ovary; DALEA, [d-Ala2, Leu5] enkephalin amide; DIEA, diisopropylethylamine; DMF, N,N-dimethyl formamide; hDOR, human δ-opioid receptor; DPDPE, c[d-Pen2, d-Pen5]enkephalin; DAMGO, [d-Ala2, N