Keywords: تداخل DNA; Pyrroloquinazolinone; Pyridoquinazolinone; Antiproliferative activity; DNA intercalation; DNA topoisomerases;
مقالات ISI تداخل DNA (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: تداخل DNA; Antimycobacterial; Anticancer; DNA intercalation; Indolizine and phenanthroline; Cycloaddition;
Keywords: تداخل DNA; SEPVRGMCAJYTPX-UHFFFAOYSA-N; GFJQKXIBRXPUOQ-UHFFFAOYSA-NEllipticine derivatives; DNA topoisomerase IIα; Anticancer drugs; Catalytic inhibitor; DNA cleavage; DNA intercalation
Synthesis of DNA interactive C3-trans-cinnamide linked β-carboline conjugates as potential cytotoxic and DNA topoisomerase I inhibitors
Keywords: تداخل DNA; β-Carbolines; Trans-cinnamides; DNA intercalation; Topoisomerase I; Anticancer activity;
A potential food biopreservative, CecXJ-37N, non-covalently intercalates into the nucleotides of bacterial genomic DNA beyond membrane attack
Keywords: تداخل DNA; Antimicrobial peptide; Food preservative; Food-borne pathogen; Amide modification; Cell membrane penetration; DNA intercalation;
Imidazopyridinium cations: A new family of azonia aromatic heterocycles with applications as DNA intercalators
Keywords: تداخل DNA; Imidazopyridinium cations; Azonia aromatic heterocycles; DNA intercalation; Cell staining;
Bioactive pigment production by Pseudomonas spp. MCC 3145: Statistical media optimization, biochemical characterization, fungicidal and DNA intercalation-based cytostatic activity
Keywords: تداخل DNA; Pyocyanin; PBD; CCD; Fungicidal; Cytostatic; DNA intercalation;
Experimental and theoretical studies on Cu(II) complex of N,N′-disalicylidene-2,3-diaminopyridine ligand reveal indirect evidence for DNA intercalation
Keywords: تداخل DNA; DNA intercalation; Schiff base; Salphen; Density functional theory; π–π stacking
Photophysical studies of donor, acceptor substituted tetrahydrodibenzo[a,i]phenanthridines
Keywords: تداخل DNA; Phenanthridines; DNA intercalation; Photophysical studies; Fluorescence spectra; UV spectra;
Antiproliferative and apoptosis-inducing activities of novel naphthalimide-cyclam conjugates through dual topoisomerase (topo) I/II inhibition
Keywords: تداخل DNA; Naphthalimide-cyclam conjugates; Antitumor agents; Topoisomerase I; Topoisomerase II; DNA intercalation; Apoptosis;
Antiproliferative, DNA intercalation and redox cycling activities of dioxonaphtho[2,3-d]imidazolium analogs of YM155: A structure-activity relationship study
Keywords: تداخل DNA; YM155; DNA intercalation; Redox cycling; Cell viability; Survivin suppressant; Apoptosis; p54nrb; nuclear RNA-binding protein; ILF3/NF110; interleukin enhancer binding factor 3/nuclear factor 110; SP1; specificity factor 1; STAT3; signal transducer and ac
Molecular and cellular inflammationNew cyclopentaquinoline derivatives with fluorobenzoic acid induce G1 arrest and apoptosis in human lung adenocarcinoma cells
Keywords: تداخل DNA; Cyclopentaquinoline derivatives; Acridine derivatives; Anticancer drug; Lung cancer; DNA intercalation;
DNA-binding studies of AV-153, an antimutagenic and DNA repair-stimulating derivative of 1,4-dihydropiridine
Keywords: تداخل DNA; 1,4-Dihydropyridines; DNA intercalation; Antimutagenic compounds; UV/VIS spectroscopy; Fluorimetry; FTIR;
Novel tetrahydroacridine derivatives inhibit human lung adenocarcinoma cell growth by inducing G1 phase cell cycle arrest and apoptosis
Keywords: تداخل DNA; Tetrahydroacridine derivatives; Acridine derivatives; Anticancer compounds; Lung cancer; DNA intercalation
Photochemical and photobiological studies on furoquinazolines as new psoralen analogs
Keywords: تداخل DNA; Furocoumarins; Furoquinazolines; DNA intercalation; Photobiological activity; Phototoxic activity
Synthesis, in vitro evaluation and molecular modelling of naphthalimide analogue as anticancer agents
Keywords: تداخل DNA; Naphthalimide analogue; Anticancer activity; DNA intercalation; Molecular modelling; Physicochemical parameters;
Novel isoxazole polycyclic aromatic hydrocarbons as DNA-intercalating agents
Keywords: تداخل DNA; DNA intercalation; Antitumor agent; Docking; Polycyclic aromatic hydrocarbons; Isoxazole; 1,3-Dipolar cycloaddition
Design and synthesis of 4-amino-2-phenylquinazolines as novel topoisomerase I inhibitors with molecular modeling
Keywords: تداخل DNA; 4-Amino-2-phenylquinazolines; Topoisomerase I; Cytotoxicity; Docking study; DNA intercalation;
DNA intercalator korkormicin A preferentially kills tumor cells expressing wild type p53
Keywords: تداخل DNA; RPE; tert-immortalized human retinal pigment epithelial cells; PARP; poly (ADP-ribose) polymerase; Korkormicin A; DNA intercalation; p53; Apoptosis; Antitumor agent;
Isoxazolidinyl polycyclic aromatic hydrocarbons as DNA-intercalating antitumor agents
Keywords: تداخل DNA; DNA intercalation; Antitumor agent; Docking; Polycyclic aromatic hydrocarbon; Isoxazolidine; 1,3-Dipolar cycloaddition;
Design, synthesis, and biological evaluation of novel N-γ-carboline arylsulfonamides as anticancer agents
Keywords: تداخل DNA; N-γ-Carboline arylsulfonamides; Anticancer; Antitubulin; DNA intercalation
Synthesis and characterization of the ligand based on benzoxazole and its transition metal complexes: DNA-binding and antitumor activity
Keywords: تداخل DNA; Antitumor activity; Benzoxazole; Transition metal complexes; DNA intercalation
Novel acridine-based compounds that exhibit an anti-pancreatic cancer activity are catalytic inhibitors of human topoisomerase II
Keywords: تداخل DNA; Acridine derivative; Anticancer drug; Cancer; Catalytic inhibitor; DNA intercalation; Topoisomerase
A [4+2] mixed ligand approach to ruthenium DNA metallointercalators [Ru(tpa)(N–N)](PF6)2 using a tris(2-pyridylmethyl)amine (tpa) capping ligand
Keywords: تداخل DNA; Bioinorganic chemistry; DNA intercalation; N ligands; Ruthenium; Density functional calculations
DNA binding of benzophenanthridine compounds sanguinarine versus ethidium: Comparative binding and thermodynamic profile of intercalation
Keywords: تداخل DNA; Sanguinarine; Ethidium; DNA intercalation; Spectroscopy; Thermodynamics; Drug–DNA interaction
Photochemical electrocyclisation of 3-vinylindoles to pyrido[2,3-a]-, pyrido[4,3-a]- and thieno[2,3-a]-carbazoles: Design, synthesis, DNA binding and antitumor cell cytotoxicity
Keywords: تداخل DNA; DNA ligands; Pyridocarbazoles; DNA intercalation; DNA minor groove binding
Naphthalimide intercalators with chiral amino side chains: Effects of chirality on DNA binding, photodamage and antitumor cytotoxicity
Keywords: تداخل DNA; Antitumor agents; Chirality; Naphthalimide; DNA intercalation; DNA photodamage
Five-coordinated oxovanadium(IV) complexes derived from amino acids and ciprofloxacin: Synthesis, spectral, antimicrobial, and DNA interaction approach
Keywords: تداخل DNA; Oxovanadium; DNA intercalation; Ciprofloxacin; Gel electrophoresis; Viscometric studies; SOD-like activity;
Genotoxicity of non-covalent interactions: DNA intercalators
Keywords: تداخل DNA; Acridines; DNA intercalation; Frameshift mutation; “Petite” mutagenesis; Topoisomerase II inhibition; Covalent DNA binding
Assessment of atypical DNA intercalating agents in biological and in silico systems
Keywords: تداخل DNA; DNA intercalation; In silico; Chinese hamster V79 cells; DNA topoisomerase II
Small molecule intercalation with double stranded DNA: Implications for normal gene regulation and for predicting the biological efficacy and genotoxicity of drugs and other chemicals
Keywords: تداخل DNA; Double stranded DNA; DNA intercalation; Drug discovery; Nuclear receptors; Gene regulation; Genotoxicity
Design, synthesis and biological evaluation of new oligopyrrole carboxamides linked with tricyclic DNA-intercalators as potential DNA ligands or topoisomerase inhibitors
Keywords: تداخل DNA; DNA ligands; Oligopyrrole carboxamides; Hybrid molecules; DNA intercalation; DNA minor groove binding
Cytotoxicity, haematotoxicity and genotoxicity of high molecular mass arborescent polyoxyethylene polymers with polyglycidol-block-containing shells
Keywords: تداخل DNA; Hyperbranched polymers; Polyoxyethylene; Polyglycidol; MTT assay; Haemolysis; DNA intercalation; Ethidium bromide; MTT; 3-[4,5-dimethylthiazole-2-yl]-2,5 diphenyltetrazolium bromide; EB; ethidium bromide;
Point-to-point capture of DNA with the aid of intercalation by immobilized rod-shaped Ru complexes at solid surface towards nanowiring
Keywords: تداخل DNA; DNA nanowiring; Ru complexes; Self-assembly; Naphthalene-1, 4: 5,8-bis(dicarboximide); DNA intercalation
CA224, a non-planar analogue of fascaplysin, inhibits Cdk4 but not Cdk2 and arrests cells at G0/G1 inhibiting pRB phosphorylation
Keywords: تداخل DNA; Cyclin-dependent kinases; G0/G1 arrest; pRB; Cell cycle; Cell growth inhibition; DNA intercalation
DNA intercalative potential of marketed drugs testing positive in in vitro cytogenetics assays
Keywords: تداخل DNA; DNA intercalation; Genotoxicity; Marketed pharmaceuticals
Antimalarial activity of thioacridone compounds related to the acronycine alkaloid
Keywords: تداخل DNA; Thioacridones; Malaria; QSAR; DNA intercalation; Plasmodium; FLEXIDOCK; SYBYL; MOLCAD;
Role of the amino sugar in the DNA binding of disaccharide anthracyclines: crystal structure of the complex MAR70/d(CGATCG)
Keywords: تداخل DNA; Anthracyclines; Drug/DNA complex; X-ray structure; DNA intercalation;
An optical DNA-based biosensor for the analysis of bioactive constituents with application in drug and herbal drug screening
Keywords: تداخل DNA; Biosensors; DNA intercalation; Synthetic and natural bioactive constituents; Drug discovery; Plant extracts; Bioactivity-guided isolation;
Synthesis, biological evaluation, and molecular modeling of novel thioacridone derivatives related to the anticancer alkaloid acronycine
Keywords: تداخل DNA; Thioacridones; Acronycine; DNA intercalation; Docking; QSAR; Bathochromic shift;
Antitumor activity and distribution of pyrroloiminoquinones in the sponge genus Zyzzya
Keywords: تداخل DNA; Antitumor; Pyrroloiminoquinone; Topoisomerase II; DNA intercalation; DNA damage; Zyzzya