Keywords: خواص دارویی; crystallinity; crystallization; drug-like properties; nonlinear regression; physical characterization; physicochemical properties; physicochemical; preformulation; structure-property relationship (SPR);
مقالات ISI خواص دارویی (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: خواص دارویی; blood-brain barrier; permeability; in vitro models; CNS; drug-like properties; drug design;
Keywords: خواص دارویی; Tuberculosis; Cell wall permeability; Drug-like properties; In silico; ADME; Physiochemical parameters;
Keywords: خواص دارویی; antiinfectives; drug resistance; drug-like properties; formulation; global health;
Keywords: خواص دارویی; drug-like properties; operating models in discovery; physicochemical properties; Drug Design; ADMET properties; insilico modeling; in-vitro models;target therapeutic profile (TPP); developability risk assessment; MAD; rule of five;
Keywords: خواص دارویی; Computer-aided drug design; QSPR; crystals; drug design; drug-like properties; molecular modeling; physical characterization; physicochemical properties
Keywords: خواص دارویی; omega-3 fatty acids; antidepressants; fluoxetine; forced swimming test; depression; drug effects; drug-like properties; pharmacodynamic; preclinical pharmacokinetic; physiological model;
MF-8, a novel promising arylpiperazine-hydantoin based 5-HT7 receptor antagonist: In vitro drug-likeness studies and in vivo pharmacological evaluation
Keywords: خواص دارویی; 5-HT7 receptor antagonist; Drug-like properties; Antidepressant-like activity; Anxiolytic-like activity; Arylpiperazines;
Estimating the Physicochemical Properties of Polysubstituted Aromatic Compounds Using UPPER
Keywords: خواص دارویی; physicochemical properties; QSPR; structure-property relationship (SPR); thermodynamics; drug-like properties; log p; molecular modeling;
Synthesis and biological activity of novel tert-amylphenoxyalkyl (homo)piperidine derivatives as histamine H3R ligands
Keywords: خواص دارویی; Histamine H3 receptor; Histamine H3 receptor ligands; Non-imidazole histamine H3R ligands; Piperidine derivatives; Anticonvulsants; Molecular docking; Drug-like properties; NLVYWCRLGFDESU-UHFFFAOYSA-N; CUKJWVHEMLBESD-UHFFFAOYSA-N; POQQPNLUXGVXQL-UHFFFAOYS
Chlorophenoxy aminoalkyl derivatives as histamine H3R ligands and antiseizure agents
Keywords: خواص دارویی; KCDBGISMCSMDRJ-UHFFFAOYSA-N; GPTIYOZHRGPQPV-UHFFFAOYSA-NHistamine H3 receptor; Histamine H3R ligands; Anticonvulsant; Ethers; Piperidine derivatives; Drug-like properties
Zanamivir Amidoxime- and N-Hydroxyguanidine-Based Prodrug Approaches to Tackle Poor Oral Bioavailability
Keywords: خواص دارویی; influenza A; neuraminidase inhibitor; synthesis; drug-like properties; prodrug; pharmacokinetics; bioavailability; guanidine bioisoster; amidine
Blood-brain barrier permeable anticholinesterase aurones: Synthesis, structure-activity relationship, and drug-like properties
Keywords: خواص دارویی; Aurones; Acetylcholinesterase inhibitors; Structure-activity relationship; Blood-brain barrier permeability; Metabolic stability; Drug-like properties;
Quality by design (QbD) of amide isosteres: 5,5-Disubstituted isoxazolines as potent CRTh2 antagonists with favorable pharmacokinetic and drug-like properties
Keywords: خواص دارویی; CRTh2 antagonists; Agonism/antagonism switch; Quality by design (QbD); Amide isostere; Isoxazolines; Drug-like properties;
Unified Physicochemical Property Estimation Relationships (UPPER)
Keywords: خواص دارویی; physicochemical properties; QSPR; thermodynamics; molecular modeling; drug-like properties; solubility; log P; multivariate analysis
Exploring nature profits: Development of novel and potent lipophilic antioxidants based on galloyl–cinnamic hybrids
Keywords: خواص دارویی; Cinnamic acid; Gallic acid; Hybrid antioxidants; Antioxidant activity; Redox potential; SPAR; Drug-like properties
Synthesis, Characterization, and Liposome Partition of a Novel Tetracycline Derivative Using the Ionic Liquids Framework
Keywords: خواص دارویی; Tetracycline; Docusate; Ionic Liquids; Synthesis; Drug-like properties; Solubility; Partition Coefficient; Liposomes; UV-VIS spectroscopy;
Functionalized indoleamines as potent, drug-like inhibitors of isoprenylcysteine carboxyl methyltransferase (Icmt)
Keywords: خواص دارویی; Isoprenylcysteine carboxyl methyltransferase (Icmt) inhibitors; Indoleamines; Antiproliferative activity; Solubility; PAMPA permeability; Drug-like properties; Metabolic stability
On Quantitative Relationships Between Drug-Like Compound Lipophilicity and Plasma Free Fraction in Monkey and Human
Keywords: خواص دارویی; Protein binding; drug-like properties; physicochemical properties; logP; structure-property relationship; lipophilicity; drug; radiotracer; logD; plasma free fraction;
Biomolecular Chemistry of Isopropyl Fibrates
Keywords: خواص دارویی; fibrates; polymorph; puckered; surface area; packing energy; drug-like properties; biophysical models; prodrugs; crystal engineering;
In Vitro Measurement of Drug Efficiency Index to Aid Early Lead Optimization
Keywords: خواص دارویی; ADME; biomimetics; HPLC (high-performance/pressure liquid chromatography); log P; protein binding; phospholipids; tissue partition; drug-like properties;
Early phase drug discovery: Cheminformatics and computational techniques in identifying lead series
Keywords: خواص دارویی; Hit-to-lead; Cheminformatics; Chemical databases; Lead-like properties; Drug-like properties; High throughput screening analysis;
In vitro Conversion of Model Sulfenamide Prodrugs in the Presence of Small Molecule Thiols
Keywords: خواص دارویی; chemical stability; drug-like properties; kinetics; prodrugs; stability;
Anti-prion activities and drug-like potential of functionalized quinacrine analogs with basic phenyl residues at the 9-amino position
Keywords: خواص دارویی; Cell-based anti-prion activity; Quinacrine analogs; Drug-like properties; Binding to human prion protein fragment; PAMPA-BBB permeability; Pgp substrate
Novel 2-imidazoles as potent and selective α1A adrenoceptor partial agonists
Keywords: خواص دارویی; α1A Adrenoceptor; Partial agonist; Selectivity; 2-Imidazole; Drug-like properties
Pharmacophore identification and virtual screening for methionyl-tRNA synthetase inhibitors
Keywords: خواص دارویی; MetRS; Pharmacophore model development; Cat-scramble; Database screening; GOLD molecular docking; Drug-like properties
Preclinical characterization of anticancer gallium(III) complexes: Solubility, stability, lipophilicity and binding to serum proteins
Keywords: خواص دارویی; Anticancer drugs; Gallium(III) complexes; Drug-like properties; Serum protein-binding; Capillary electrophoresis;
An efficient approach for the rapid assessment of oral rat exposures for new chemical entities in drug discovery
Keywords: خواص دارویی; preclinical pharmacokinetics; ADME; high throughput technologies; oral absorption; mass spectrometry; physicochemical properties; drug-like properties; drug design; sampling pooling;