Keywords: Eg5; LSCC; qPCR; IHC
مقالات ISI (ترجمه نشده)
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VPS28, an ESCRT-I protein, regulates mitotic spindle organization via Gβγ, EG5 and TPX2
Keywords: Mitotic spindle; VPS28; Gbetagamma; Gproteins; Eg5; TPX2;
Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors
Keywords: 1,3,4-thiadiazole; K858 enantiomers; Eg5; Antimitotic drugs; Eg5-K858 complex; Rational drug design; KSP; Kinesin spindle protein; MT; Microtubule; PDB; Protein Data Bank; PK; Pyruvate kinase; LDH; Lactate dehydrogenase; ITC; Isothermal titration calorime
CD52, CD22, CD26, EG5 and IGF-1R expression in thymic malignancies
Keywords: CD52; CD22; CD26; EG5; IGF-1R; Thymic;
Alzheimer amyloid beta inhibition of Eg5/kinesin 5 reduces neurotrophin and/or transmitter receptor function
Keywords: Alzheimer's disease; Abeta peptide; Eg5; Kinesin 5; Microtubules; Neurotrophin receptor; Neurotransmitter receptor; p75; NMDA receptor; Neurite outgrowth; Neurodegeneration; Down syndrome;
Synergism between inhibitors of Aurora A and KIF11 overcomes KIF15-dependent drug resistance
Keywords: Drug-resistance; Drug screening; Eg5; Infrared; Kinesin; Mitosis;
Kif11 dependent cell cycle progression in radial glial cells is required for proper neurogenesis in the zebrafish neural tube
Keywords: Kif11; Eg5; Kinesin; Radial glia; Neural stem cell; Mitosis; Zebrafish; Interneuron; Motorneuron; Oligodendrocyte; Mathematical modeling;
Insight into Nek2A activity regulation and its pharmacological prospects
Keywords: Nek2A; CEP135; C-Nap1; Rootelin; Mst1/Mst2; HSav1; Eg5; Cancer; Inhibitor; Activity regulation; Functional domains
Advances in the discovery of kinesin spindle protein (Eg5) inhibitors as antitumor agents
Keywords: Eg5; KSP; Inhibitors; Antimitotic agentsACAT, acyl-CoA:cholesterol acyltransferase; ADP, adenosine diphosphate; AML, acute myeloid leukemia cell; AS-2, adociasulfate-2; ATP, adenosine triphosphate; bimC, blocked in mitosis; CHK1, checkpoint 1; CR, complet
Doing the methylene shuffle - Further insights into the inhibition of mitotic kinesin Eg5 with S-trityl l-cysteine
Keywords: Mitotic kinesins; Eg5; Antimitotic agents; STLC; Molecular dynamics; KSP; cLogD7.4; calculated LogD7.4; cLogS; calculated Log S, where S is the solubility in mol/L; DMEM; Dulbecco's Modified Eagle Medium; Et2O; diethyl ether; EtOAc; ethyl acetate; GI50
The discovery of tetrahydro-β-carbolines as inhibitors of the kinesin Eg5
Keywords: Eg5; KSP; Kinesin
Mitotic functions of kinesin-5
Keywords: Eg5; Mitosis; Spindle; Kinesin; Dynein
Kinesin passing permanent blockages along its protofilament track
Keywords: KIF5A; Eg5; Motility; Bypassing; Non-exchangeable blockages
Mutations in the human kinesin Eg5 that confer resistance to monastrol and S-trityl-l-cysteine in tumor derived cell lines
Keywords: Eg5; Mitosis; Monastrol; STLC; Drug; Resistance
Cryo-electron tomography of microtubule-kinesin motor complexes
Keywords: Cryo-electron microscopy; Cryo-electron tomography; Kinesin; Microtubules; Helical 3-D reconstruction; Eg5; Kar3Vik1;
Assessing compound binding to the Eg5 motor domain using a thermal shift assay
Keywords: Eg5; Kinesin; Kinesin spindle protein; KSP; Thermal shift assay; Cancer
Synthesis and biological evaluation of l-cysteine derivatives as mitotic kinesin Eg5 inhibitors
Keywords: S-Trityl-l-cysteine; Mitotic kinesin; Eg5; Inhibitor; Anticancer
The kinesin related motor protein, Eg5, is essential for maintenance of pre-implantation embryogenesis
Keywords: Eg5; Kinesin related protein; Mitotic spindle; Cell cycle arrest; Embryonic lethal; Gene knock out; Genetrap; Proliferation defect; Preimplantation embryo
Synthesis and SAR of thiophene containing kinesin spindle protein (KSP) inhibitors
Keywords: Eg5; KSP; Kinesin spindle protein; Anti-mitotics; Thiophenes
New chemical tools for investigating human mitotic kinesin Eg5
Keywords: Antitumor agent; Inhibitor; Molecular motor; Eg5; Monastrol; Structure–activity relationships
Mitotic drug targets and the development of novel anti-mitotic anticancer drugs
Keywords: Mitosis; Chemotherapy; Spindle checkpoint; Aurora kinase; Polo-like kinase; KSP; Eg5; Microtubules; Taxanes; Vinca alkaloids; UCN-01; G2 checkpoint; Anticancer drug resistance
Synthesis and SAR of pyrrolotriazine-4-one based Eg5 inhibitors
Keywords: Eg5; Pyrrolotraizine; Microtubule; Kinesin; Anti-tumor; Cytotoxic
Inhibitors of human mitotic kinesin Eg5: Characterization of the 4-phenyl-tetrahydroisoquinoline lead series
Keywords: Eg5 inhibitor; Kinesin inhibitor; Kinesin spindle protein; KSP; Eg5
Phenothiazine and carbazole-related compounds inhibit mitotic kinesin Eg5 and trigger apoptosis in transformed culture cells
Keywords: Phenothiazine; Mitotic arrest; Apoptosis; Eg5