Keywords: ABC; ATP-binding cassette; BCRP/ABCG2; breast cancer resistance protein; Bz; benzoyl; FTC; fumitremorgin C; mBu; methyl isobutyl; LBE; lowest binding energies; MDR; multidrug resistance; MRP1; multidrug-resistance-associated protein 1; POP; polyoxypregnan
مقالات ISI (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: FTM-C; fumitremordin C; BCRP; breast cancer resistance protein; PKS; polyketide synthase; NRPS; nonribosomal peptide synthetase; α-KG; α-ketoglutarate; SAR; structure-activity relationship; KSP; kinesin spindle protein; TAS1; tenuazonic acid synthetase
Olmutinib (HM61713) reversed multidrug resistance by inhibiting the activity of ATP-binding cassette subfamily G member 2 in vitro and in vivo
Keywords: ABC; adenosine triphosphate (ATP)-binding cassette; ABCG2; ABC transporter subfamily G member 2; DDP; cisplatin; DMEM; Dulbecco׳s modified Eagle׳s medium; DMSO; dimethyl sulfoxide; DOX; doxorubicin; FTC; fumitremorgin C; IAAP; iodoarylazidoprazosin; MDR
Halogenated naphthochalcones and structurally related naphthopyrazolines with antitumor activity
Keywords: ABC; adenosine triphosphate binding cassette; BCRP; breast cancer resistance protein; FTC; fumitremorgin C; MDR; multidrug resistance; P-gp; P-glycoptotein; SD; standard deviation; TdT; Terminal deoxyribonucleotide Transferase; Topo; topotecan; TUNEL; Ter
Assessment of ABCG2-mediated transport of pesticides across the rabbit placenta barrier using a novel MDCKII in vitro model
Keywords: ABCG2; ATP-binding cassette sub-family G member 2; CPF; chlorpyrifos; DAPI; 4â²-6-diamidino-2-phenylindole; FTC; fumitremorgin C; MDCKII; Madin-Darby canine kidney type II cells; MRL; maximum residue limits; Papp; apparent permeability coefficient; TEER;
Phenyltetrazolyl-phenylamides: Substituent impact on modulation capability and selectivity toward the efflux protein ABCG2 and investigation of interaction with the transporter
Keywords: ABC-transporter; ABCG2; BCRP inhibitor; Synthesis; Structure-activity relationship; Enzyme kinetics; ABC; ATP-binding cassette; BCRP; breast cancer resistance protein (ABCG2); CsA; cyclosporine A; FTC; fumitremorgin C; Imax; maximal inhibition; i-Pr; isop
The enriched fraction of Vernonia cinerea L. induces apoptosis and inhibits multi-drug resistance transporters in human epithelial cancer cells
Keywords: ATP; Adenosine triphosphate; ABC; ATP binding cassette; DMSO; Dimethyl Sulfoxide; DMEM; Dulbecco׳s modified eagle medium; Dox; Doxorubicin; DNR; Daunorubicin; FBS; Fetal bovine serum; FITC; Fluorescein Isothiocyanate; FTC; Fumitremorgin C; HBSS; Hank׳s
CEP-33779 antagonizes ATP-binding cassette subfamily B member 1 mediated multidrug resistance by inhibiting its transport function
Keywords: ABC; ATP-binding cassette; ABCC1; multidrug resistance-associated protein 1; ABCG2; breast cancer resistance protein; CSCs; Cancer stem cell; DOX; doxorubicin; FTC; fumitremorgin C; GAPDH; glyceraldehyde-3-phosphate dehydrogenase; Rho123; Rhodamine 123; M
Human ABCB1 (P-glycoprotein) and ABCG2 mediate resistance to BI 2536, a potent and selective inhibitor of Polo-like kinase 1
Keywords: MDR; multidrug resistance; ABC; ATP-binding cassette; Plk-1; Polo-like kinase 1; PhA; pheophorbide A; FTC; Fumitremorgin C; MTT; 3-(4,5-dimethylthiazol-yl)-2,5-diphenyllapatinibrazolium bromide; Vi; sodium orthovanadate; ABC transporter; Multidrug resista
Sensitive method for plasma and tumor Ko143 quantification using reversed-phase high-performance liquid chromatography and fluorescence detection
Keywords: Ko143; Fumitremorgin C; Roquefortine C; Topotecan; ABCG2; Drug resistance
Constitutive androstane receptor upregulates Abcb1 and Abcg2 at the blood-brain barrier after CITCO activation
Keywords: ABC-transporter; ATP-binding cassette transporter; BBB; blood-brain barrier; BCRP; breast cancer resistance protein; BMDP; brain multidrug resistance protein; CAR; constitutive androstane receptor; CYP; cytochrome P450; pgCAR; porcine CAR; CITCO; 6-(4-c
OSI-930 analogues as novel reversal agents for ABCG2-mediated multidrug resistance
Keywords: OSI-930; {N-(4-trifluoromethoxyphenyl)3-((quinolin-4-ylmethyl) amino) thiophene-2-carboxamide}; ABC; ATP binding cassette; ABCG2 (BCRP/MXR/ABCP); ABC subfamily G member 2; MDR; multidrug resistance; P-gp; P-glycoprotein; ABCCs (MRPs); ABC subfamily C memb
Breast cancer resistance protein BCRP/ABCG2 regulatory microRNAs (hsa-miR-328, -519c and -520h) and their differential expression in stem-like ABCG2+ cancer cells
Keywords: miRNA; microRNA; BCRP/ABCG2; breast cancer resistance protein/ATP-binding cassette, subfamily G (white), member 2; hsa-miR-328; human microRNA-328; miR-519c; microRNA-519c; miR-520 h; microRNA-520h; MRE; microRNA response element; 3â²UTR; 3â²-untranslat
Differential inhibition of murine Bcrp1/Abcg2 and human BCRP/ABCG2 by the mycotoxin fumitremorgin C
Keywords: Fumitremorgin C; BCRP/ABCG2; Transport; Inhibition; Cytotoxicity;
Chemotherapeutic Drug-Induced ABCG2 Promoter Demethylation as a Novel Mechanism of Acquired Multidrug Resistance
Keywords: ABC; ATP-binding cassette; Act D; actinomycin D; ALL; acute lymphoblastic leukemia; COBRA; combined bisulfite restriction analysis; DNMT; DNA methyltransferase; DNR; daunorubicin; Dox; doxorubicin; FTC; fumitremorgin C; HDACi; histone deacetylase inhibito
Establishment of a luciferase assay-based screening system: Fumitremorgin C selectively inhibits cellular proliferation of immortalized astrocytes expressing an active form of AKT
Keywords: AKT; Fumitremorgin C; Glioblastoma; High-throughput screening