دانلود مقالات ISI درباره H3R + ترجمه فارسی

Functional histamine H3 and adenosine A2A receptor heteromers in recombinant cells and rat striatum

Keywords: A2AR; Adenosine A2A receptor; cAMP; Cyclic adenosine monophosphate; D1R; Dopamine D1 receptor; D2R; Dopamine D2 receptor; dMSNs; Direct pathway striatal medium-sized spiny neurons; GABA; γ-Aminobutyric acid; GPCRs; G-protein coupled receptors; H2R; Hista

دانلود رایگان متن کامل مقاله ISI 47 صفحه سال انتشار : 2018 سفارش ترجمه

The naturally occurring mutation Y197C does not affect the expression or signaling of the human histamine H3 receptor

Keywords: GPCR; G protein-coupled receptor; H3R; histamine H3 receptor; hH3R; human histamine H3 receptor; RAMH; (R)-α-methylhistamine; TM; transmembrane domain; Histamine; H3 receptor; Mutation; Y197C mutation; Signaling; CHO-K1 cells;

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2017 سفارش ترجمه

The dual-acting AChE inhibitor and H3 receptor antagonist UW-MD-72 reverses amnesia induced by scopolamine or dizocilpine in passive avoidance paradigm in rats

Keywords: AChE; acetylcholine esterase; BChE; butyrylcholinesterase; AChEI; acetylcholine esterase inhibitor; H3R; histamine H3 receptor; H1R; histamine H1 receptor; H2R; histamine H2 receptor; AD; Alzheimer's disease; SCO; scopolamine; NMDA; N-methyl-d-aspartate;

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2016 سفارش ترجمه

Histamine H3 receptor activation inhibits dopamine synthesis but not release or uptake in rat nucleus accumbens

Keywords: Histamine; Dopamine; H3 receptor; Nucleus accumbens; Dopamine synthesis; Dopamine release; D2R; dopamine D2 receptor; DOPA; l-dihydroxyphenylalanine; GABA; γ-aminobutyric acid; H3R; histamine H3 receptor; MSNs; medium spiny neurons; RAMH; (R)(-)-α-methy

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2016 سفارش ترجمه

Donepezil, an acetylcholine esterase inhibitor, and ABT-239, a histamine H3 receptor antagonist/inverse agonist, require the integrity of brain histamine system to exert biochemical and procognitive effects in the mouse

Keywords: HDC-KO mice; a-fluoromethylhistidine; Object recognition test; Memory; Acetylcholine; GSK-3β; a-FMHis; alpha-fluromethylhistidine; H3R; histamine H3 receptor; HDC; histidine decarboxylase; ORT; object recognition test; T1; training session; T2; test sess

دانلود رایگان متن کامل مقاله ISI 36 صفحه سال انتشار : 2016 سفارش ترجمه

Epidermal growth factor receptor inhibitor cancer drug gefitinib modulates cell growth and differentiation of acute myeloid leukemia cells via histamine receptors

Keywords: 4-MH; 4-methylhistamine; AML; acute myelogenous leukemia; CML; chronic myelogenous leukemia; cAMP; cyclic adenosine monophosphate; CRE; cAMP response element; EGFR; epidermal growth factor receptor; ER; estrogen receptor alpha; FSK; Forskolin; GPCR; G-pro

دانلود رایگان متن کامل مقاله ISI 40 صفحه سال انتشار : 2016 سفارش ترجمه

Histamine H3 receptor activation stimulates calcium mobilization in a subpopulation of rat striatal neurons in primary culture, but not in synaptosomes

Keywords: Histamine; H3 receptor; Striatum; Calcium mobilization; Primary culture; Synaptosomes; ACPD; (±)-trans 1-Amino-1,3-dicarboxycyclopentane; [Ca2+]i; intracellular concentration of Ca2+; CNS; Central Nervous System; D1R; dopamine D1 receptor; D2R; dopamine

دانلود رایگان متن کامل مقاله ISI 47 صفحه سال انتشار : 2016 سفارش ترجمه

The novel non-imidazole histamine H3 receptor antagonist DL77 reduces voluntary alcohol intake and ethanol-induced conditioned place preference in mice

Keywords: BEC; blood ethanol concentration; CPP; conditioned-place preference; EtOH; ethanol; H3R; histamine H3 receptor; PYR; pyrilamine; RAMH; R-(alpha)-methyl-histamine; Conditioned place preference; Ethanol; Histamine H3 receptor; Pyrilamine; R-(alpha)-methyl-h

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2015 سفارش ترجمه

Betahistine co-treatment ameliorates dyslipidemia induced by chronic olanzapine treatment in rats through modulation of hepatic AMPKα-SREBP-1 and PPARα-dependent pathways

Keywords: ACC1; acetyl-CoA carboxylase 1; AMPKα; AMP-activated protein kinaseα; CPT1A; carnitine palmitoyltransferase 1A; FASN; fatty acid synthetase; H1R; histamine H1 receptors; H3R; histamine H3 receptors; HDL-C; high density lipoprotein cholesterol; HMGCoA; 3

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2015 سفارش ترجمه

Homologous desensitization of human histamine H3 receptors expressed in CHO-K1 cells

Keywords: Histamine; H3 receptor; Desensitization; GRK; CHO-K1 cells; Neuromodulation; H3R; histamine H3 receptor; GPCR; G protein-coupled receptor; GRK; GPCR kinase; RAMH; R-α-methylhistamine;

دانلود رایگان متن کامل مقاله ISI 11 صفحه سال انتشار : 2014 سفارش ترجمه

Efficacy of the histamine 3 receptor (H3R) antagonist pitolisant (formerly known as tiprolisant; BF2.649) in epilepsy: Dose-dependent effects in the human photosensitivity model

Keywords: Histamine 3 antagonist; H3R; Pitolisant; Tiprolisant; BF2.649; Nonimidazole; Epilepsy; Proof of concept; Photosensitivity model; PPR;

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2013 سفارش ترجمه

Selective brain region activation by histamine H3 receptor antagonist/inverse agonist ABT-239 enhances acetylcholine and histamine release and increases c-Fos expression

Keywords: Acetylcholine; c-Fos; Histamine; Histamine H3 receptor; Microdialysis; H3R; histamine H3 receptor; ACh; acetylcholine; ADHD; attention-deficit hyperactivity disorder; i.p.; intraperitoneally; PBS; phosphate-buffer saline; TMN; tuberomamillary nucleus; NBM

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2013 سفارش ترجمه

Ligand based design of novel histamine H4 receptor antagonists; fragment optimization and analysis of binding kinetics

Keywords: Histamine; H4R antagonist; GPCR; Binding kinetics; Fragment optimization; GPCRs; G protein-coupled receptors; H1R; histamine H1 receptor; H2R; histamine H2 receptor; H3R; histamine H3 receptor; H4R; histamine H4 receptor; SAR; structure-activity relatio

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2012 سفارش ترجمه

Novel and highly potent histamine H3 receptor ligands. Part 1: withdrawing of hERG activity

Keywords: Histamine; H3R; HERG; QSAR;

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2011 سفارش ترجمه

The hydrophobic amino acids in putative helix 8 in carboxy-terminus of histamine H3 receptor are involved in receptor-G-protein coupling

Keywords: GPCR; G-protein coupled receptor; H3R; histamine H3 receptor; HEK; human embryonic kidney; CLIC4; chloride intracellular channel 4; DMEM; Dulbecco's modified Eagle's medium; PBS; phosphate buffered saline; PAGE; polyacrylamide gel electrophoresis; RAMH; R

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2011 سفارش ترجمه

Searching for the Multi-Target-Directed Ligands against Alzheimer's disease: Discovery of quinoxaline-based hybrid compounds with AChE, H3R and BACE 1 inhibitory activities

Keywords: Alzheimer's disease; BACE 1; AChE; H3R; Multi-Target-Directed Ligands;

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2011 سفارش ترجمه

Cellular and Molecular NeuroscienceResearch PaperPre-synaptic histamine H3 receptors modulate glutamatergic transmission in rat globus pallidus

Keywords: histamine; H3 receptor; globus pallidus; basal ganglia; glutamate release; GABA; γ-aminobutyric acid; GP; globus pallidus; H3R; histamine H3 receptor; [3H]-NMHA; N-α-[methyl-3H]histamine;

دانلود رایگان متن کامل مقاله ISI 12 صفحه سال انتشار : 2011 سفارش ترجمه

Discovery of substituted benzyl tetrazoles as histamine H3 receptor antagonists

Keywords: Histamine; H3R; Antagonists; CNS; GPCR; Drug discovery

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2010 سفارش ترجمه