Keywords: Anticancer activity; Cytotoxicity; Fluorescent cyanine; Pentamethinium salt; Recognition; Sulfated polysaccharides; A549; cells of lung adenocarcinoma; AIDS; acquired immune deficiency syndrome; BJ; human fibroblasts (non-malignant cell line); BrdU; 5-bro
مقالات ISI (ترجمه نشده)
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Keywords: Carbazoles; Guanidinocarbazoles; Guanidines; KB; HL60; MCF7; HCT116; PC3; MRC5;
Chitosan oligosaccharides with degree of polymerization 2-6 induces apoptosis in human colon carcinoma HCT116 cells
Keywords: Chitosan oligosaccharides; Degree of polymerization; Colon cancer; HCT116; Apoptosis;
Design and synthesis of novel imidazo[4,5-b]pyridine based compounds as potent anticancer agents with CDK9 inhibitory activity
Keywords: Imidazo[4,5-b]pyridines; Anticancer; CDK9; HCT116; MCF-7;
Biological applications of Ru(II) polypyridyl complexes
Keywords: FDA; United States Food and Drug Administration; PDT; photodynamic therapy; PS; photosensitizer; ROS; reactive oxygen species; PACT; photodynamic antimicrobial chemotherapy; NKP-1339; sodium salt of indazolium trans-[tetrachlorobis(1H-indazole)ruthenate(I
The involvement of ROS generation on Epoxiconazole-induced toxicity in HCT116 cells
Keywords: EPX; Epoxiconazole; ROS; Reactive oxygen species; ÎΨm; mitochondrial transmembrane potential; EBI; Ergosterol Binding inhibitor; Epoxiconazole; Oxidative stress; HCT116; DNA fragmentation;
Chemical characterization and cytotoxic, genotoxic, and mutagenic properties of Baccharis trinervis (Lam, Persoon) from Colombia and Brazil
Keywords: CHO; Chinese Hamster Ovary; AE; Aqueous extracts; B; Brazil; C; Colombia; EAF; Ethyl Acetate Fraction; BF; Butanol Extract; ARF; Aqueous Residue Fraction; HPLC; High Performance Liquid Chromatography; HRMS; High Resolution Mass Spectrometry; MTT; 3-(4.5-d
Comprehensive review on flavonoids biological activities of Erythrina plant species
Keywords: 5-LOX; 5-lipoxygenase; AMPK; adenosine monophosphate-activated protein kinase; Bax; Bcl-2-associated X protein; BC; lymphoma cell line; Bcl-2; B-cell CLL/lymphoma 2; Caco2; human epithelial colorectal adenocarcinoma cells; CCRF-CEM; T lymphoblastoid cell
Trans-C versus Cis-C thermally induced isomerisation of a terpyridine adduct of cytotoxic cycloruthenated compound
Keywords: Cyclometalated compounds; Antisymbiotic effect; Isomerisation; Substitution of ligands; Cytotoxicity; HCT116;
Pharmacological inhibition of MAGL attenuates experimental colon carcinogenesis
Keywords: 2-AG; 2-arachidonoyl glycerol; ACF; aberrant crypt foci; AEA; anandamide; AOM; azoxymethane; BSA; bovine serum albumin; HCT116; colon adenocarcinoma cell line; CRC; colorectal cancer; DMSO; dimethyl sulphoxide; DMEM; Dulbecco's modified Eagle's medium
Synthesis, characterization, crystal structure and in vitro anticancer potentials of mono and bimetallic palladium(II)-N-heterocyclic carbene complexes
Keywords: Anticancer activity; HCT116; MTT assay; Palladium-NHC complex; X-ray diffraction;
DFT analysis and bioactivity of 2-((E)-(4-methoxybenzylimino)methyl)phenol and its Ni(II) and Pd(II) complexes
Keywords: Schiff base; Ni(II); Pd(II); HCT116; Escherichia coli; DFT;
Preliminary investigation of catalytic, antioxidant, anticancer and bactericidal activity of green synthesized silver and gold nanoparticles using Actinidia deliciosa
Keywords: Green synthesis; Antioxidant; Anticancer; HCT116; TEM;
P53 tumor suppressor is required for efficient execution of the death program following treatment with a cytotoxic limonoid obtained from Melia azedarach
Keywords: Meliartenin; 12-Hydroxyamoorastatin; Cytotoxicity; Apoptosis; Cell cycle arrest; HCT116; p53; ALL; acute lymphoblastic leukemia; BrdU; 5-bromo-2'-deoxyuridine; CML; chronic myeloid leukemia; DMSO; dimethyl sulfoxide; DOX; doxorubicin; FBS; fetal bovine
A cytotoxic C-glycosylated derivative of apigenin from the leaves of Ocimum basilicum var. thyrsiflorum
Keywords: Ocimum basilicum; HCT116; Cytotoxic; Antioxidant; C-glycosylation; Apigenin derivative;
Short communicationTLR3 signaling is downregulated by a MAVS isoform in epithelial cells
Keywords: TLR3; MAVS; Isoform; Interferon beta; Regulation; Epithelial cells; miniMAVS; HCT116;
Computer-aided design, synthesis, and biological evaluation of new indole-2-carboxamide derivatives as PI3Kα/EGFR inhibitors
Keywords: PI3Kα; EGFR; HCT116; MDA231; Docking;
Molecular modeling based approach, synthesis, and cytotoxic activity of novel benzoin derivatives targeting phosphoinostide 3-kinase (PI3Kα)
Keywords: PI3Kα; Cancer; Docking; HCT116; Benzoin;
In-vitro assessment of cytotoxicity of halloysite nanotubes against HepG2, HCT116 and human peripheral blood lymphocytes
Keywords: Halloysite nanotubes; HepG2; HCT116; Peripheral blood lymphocytes; In-vitro cytotoxicity; Pharmaceutical excipients; Size distribution;
CYP2S1 depletion enhances colorectal cell proliferation is associated with PGE2-mediated activation of β-catenin signaling
Keywords: CYP2S1; HCT116; PGE2; β-catenin; ShRNA; Colorectal cancer cell;
κ-Carrageenan from marine red algae, Kappaphycus alvarezii – A functional food to prevent colon carcinogenesis
Keywords: Low-molecular weight carrageenan; Dietary fibre; Functional food; Apoptosis; HCT116; ROS
Synthesis and evaluation of an imidazole derivative–fluorescein conjugate
Keywords: MDM2; p53; Fluorescence imaging; FAM; Nutlin-2; Glycine; PET; SJSA-1; HCT116
Paclitaxel-incorporated nanoparticles of hydrophobized polysaccharide and their antitumor activity
Keywords: Nanoparticles; Paclitaxel; Pullulan; Polysaccharide; HCT116
Synthesis and in vitro antiproliferative activity of new 11-aminoalkylamino-substituted chromeno[2,3-b]indoles
Keywords: Chromeno[2,3-b]indole; Aminoalkylamino-substituted indole derivatives; Antiproliferative activity; MV4-11; HCT116
Synthesis and antitumor activity of novel 6-aryl and 6-alkylpyrazolo[3,4-d]pyrimidin-4-one derivatives
Keywords: Pyrazolo[3,4-d]pyrimidin-4-one; Antitumor activity; HCT116
An investigation of the occurrence and properties of the mitochondrial intermediate-conductance Ca2+-activated K+ channel mtKCa3.1
Keywords: BKCa; big conductance Ca2+-activated K+-channel (KCa1.1); Clotrimazole; 1-[(2-chlorophenyl)-diphenyl-methyl]imidazole; CsA; Cyclosporin A; DC-EBIO; 5,6-dichloro-1-ethyl-1,3-dihydro-2H-benzimidazol-2-one; DMEM; Dulbecco's modified Eagle medium; ER; endopla
Modulation of transplanaramine platinum complex reactivity by systematic modification of carrier and leaving groups
Keywords: Trans platinum; HCT116; Interstrand cross-links; Platinum accumulation;
HCT116 cells deficient in p21Waf1 are hypersensitive to tyrosine kinase inhibitors and adriamycin through a mechanism unrelated to p21 and dependent on p53
Keywords: Chx; cycloheximide; PARP; poy(ADP-ribose)polymerase; PI; propidium iodide; p53; Adriamycin; Imatinib; Gefitinib; Apoptosis; HCT116; Myc;
PCDH24-induced contact inhibition involves downregulation of β-catenin signaling
Keywords: PCDH24; Contact inhibition; β-catenin; HCT116; Actin; VimentinqRT-PCR, quantitative real-time-PCR; LMB, leptomycin B; 2-DE/MS, two-dimensional gel electrophoresis/mass spectrometry; PLAUR, plasminogen activator urokinase receptor
The isolation, structure determination and cytotoxicity of the new fungal metabolite, trichodermamide C
Keywords: Trichodermamide C; X-ray structure; Cytotoxicity; High content screening; A549; HCT116
Flavonoid, Silibinin, Inhibits Proliferation and Promotes Cell-Cycle Arrest of Human Colon Cancer
Keywords: silibinin; milk thistle; colon cancer; Fet; Geo; HCT116