Keywords: هیدروکسی اتیلین; Phthalimide; Hydroxyethylamine; Antimalarial; Drug resistance; Plasmepsins;
مقالات ISI هیدروکسی اتیلین (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: هیدروکسی اتیلین; QRJCFENHSFVGNL-MSOLQXFVSA-N; BYZAHKRALXCGNO-XAZDILKDSA-N; WSDASMLFNPNZOK-JFYQQWHZSA-N; Hydroxyethylamine; Molecular self-assembly; Falcipain-3; Antimalarial chemotheraphy; Hemoglobin hydrolysis;
G-score: A function to solve the puzzle of modeling the protonation states of β-secretase binding pocket
Keywords: هیدروکسی اتیلین; G-score; Population density; Molecular dynamics; GROMACS; BACE1; Reduced amide; Tertiary carbinamine; Hydroxyethylamine; Protonation state; Alzheimer; TMoLiC;
A PM7 dynamic residue-ligand interactions energy landscape of the BACE1 inhibitory pathway by hydroxyethylamine compounds. Part I: The flap closure process
Keywords: هیدروکسی اتیلین; BACE1; Hydroxyethylamine; Flap; PM7; MOPAC; Interaction energy; GROMACS; Molecular dynamics;
Evaluation of transition-state mimics in a superior BACE1 cleavage sequence as peptide-mimetic BACE1 inhibitors
Keywords: هیدروکسی اتیلین; BACE 1; Inhibitor; Transition state mimic; Hydroxyethylamine; Hydroxymethylcarbonyl;
Thermodynamic and kinetic characterization of hydroxyethylamine β-secretase-1 inhibitors
Keywords: هیدروکسی اتیلین; β-Secretase; Hydroxyethylamine; SPR; Kinetics; Thermodynamics; Residence time;
Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: Prime side chromane-containing inhibitors
Keywords: هیدروکسی اتیلین; Beta-secratase inhibitor; BACE-1; Alzheimer’s disease; Cat-D; Chromane; Hydroxyethylamine
BACE-1 hydroxyethylamine inhibitors using novel edge-to-face interaction with Arg-296
Keywords: هیدروکسی اتیلین; Alzheimer; BACE-1; Aspartic protease; Hydroxyethylamine; Edge-to-face;
Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: Structure–activity relationship of the aryl region
Keywords: هیدروکسی اتیلین; Alzheimer’s disease; Beta-secretase inhibitor; BACE-1; HEA; Hydroxyethylamine
Design and synthesis of 1,4-dihydropyridine derivatives as BACE-1 inhibitors
Keywords: هیدروکسی اتیلین; BACE-1 inhibitors; Hydroxyethylamine; 1,4-Dihydropyridine; Alzheimer's disease1,4-DHP, 1,4-Dihydropyridine; Aβ40, 40-Residue β-amyloid peptide; Aβ42, 42-Residue β-amyloid peptide; AD, Alzheimer's diseases; AP, Alkaline phosphatase; APP, β-Amyloid precurso
Synthesis, antimalarial evaluation and molecular modeling studies of hydroxyethylpiperazines, potential aspartyl protease inhibitors, Part 2
Keywords: هیدروکسی اتیلین; Protease inhibitor; Malaria; Hydroxyethylamine
Second generation of BACE-1 inhibitors part 3: Towards non hydroxyethylamine transition state mimetics
Keywords: هیدروکسی اتیلین; Alzheimer; BACE-1; Apartic protease; Hydroxyethylamine
Second generation of BACE-1 inhibitors part 2: Optimisation of the non-prime side substituent
Keywords: هیدروکسی اتیلین; Alzheimer; BACE-1; Hydroxyethylamine; Aspartic protease
Second generation of BACE-1 inhibitors. Part 1: The need for improved pharmacokinetics
Keywords: هیدروکسی اتیلین; Alzheimer; BACE-1; Aspartic protease; Hydroxyethylamine
Aspartic protease inhibitors via C1-homologation of peptidic aldehydes and studies on reduced amide isosteres
Keywords: هیدروکسی اتیلین; β-Secretase; Transition state isostere; Hydroxyethylamine; Reduced amide; Grignard reagent; Indole synthesis;
Potent and selective isophthalamide S2 hydroxyethylamine inhibitors of BACE1
Keywords: هیدروکسی اتیلین; BACE1; Isophthalamide; HEA; Alzheimer’s disease; Hydroxyethylamine; Inhibitor; S2 pocket; β-Secretase
Synthesis, biological evaluation, and modeling studies of inhibitors aimed at the malarial proteases plasmepsins I and II
Keywords: هیدروکسی اتیلین; Malaria; Plasmepsin; Hydroxyethylamine; Molecular modeling;