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Structure-activity relationship studies on 1-(2-oxopropyl)indole-5-carboxylic acids acting as inhibitors of cytosolic phospholipase A2α: Effect of substituents at the indole 3-position on activity, solubility, and metabolic stability
Keywords: کاهش کتون; Cytosolic phospholipase A2α; Inhibitors; Indole derivatives; Metabolic stability; Ketone reduction; Glucuronidation; Aqueous solubility;