Keywords: دامنه اتصال لیگاند; NRs; nuclear recepors; LBD; ligand-binding domain; DBD; DNA-binding domain; CRM-1; chromosome region maintenance 1; CRT; calreticulin; NES; nuclear export sequence; BC; breast cancer; PC; prostate cancer; LMB; leptomycin B; Nuclear receptors; Nuclear expo
مقالات ISI دامنه اتصال لیگاند (ترجمه نشده)
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Keywords: دامنه اتصال لیگاند; ARSIs; androgen receptor signaling inhibitors; AA; abiraterone acetate; AR; androgen receptor; BPH; benign prostatic hyperplasia; CNV; copy number variation; CRPC; castration resistant prostate cancer; CTC; circulating tumor cells; ctDNA; cell-free circul
Keywords: دامنه اتصال لیگاند; HCV; hepatitis C virus; VDR; vitamin D receptor; IFN-α; interferon-α; ISG; interferon-stimulated gene; LBD; ligand-binding domain; CoA; coactivator; CoR; corepressor; IGF-2; insulin-like growth factor 2; IL-32; interleukin-32; CCL20; C-C motif chemokine
Keywords: دامنه اتصال لیگاند; TFR; transcription factor of the TetR family; EMSA; electrophoretic mobility shift assay; LBD; ligand-binding domain; DBD; DNA-binding domain; Whole cell biosensor; Actinobacteria; Secondary metabolite; Antibiotic; Polyketide; TetR repressor protein;
Keywords: دامنه اتصال لیگاند; AF-1; activation function-1; AF-2; activation function-2; AP-1; activator protein 1; dppp; 1,3-bis(diphenylphosphino)propane; DEX; dexamethasone; DIEA; N,N-diisopropylethylamine; FKBP5; FK506-binding protein 5; GR; glucocorticoid receptor; GRE; glucocorti
Keywords: دامنه اتصال لیگاند; Kainate receptors; N-terminal domain; Ligand-binding domain; Crystal structures; Ligands; Mutations; AMPA; α-amino-3-hydroxy-5-methyl-4-isoxazolepropionate; iGluRs; ionotropic glutamate receptors; LBDs; ligand-binding domains; NMDA; N-methyl-d-aspartate;
Keywords: دامنه اتصال لیگاند; BC; Breast cancer; CRM-1; Chromosome region maintenance 1; DBD; DNA-binding domain; E2; 17-beta-estradiol; EGF; Epidermal growth factor; ERα; Estrogen receptor alpha; Ful; Fulvestrant; GFP-ER; ER tagged with green fluorescent protein; HSP70; Heat shock p
Keywords: دامنه اتصال لیگاند; 11KT; 11-ketotestosterone; 17bhsd; 17β-hydroxysteroid dehydrogenase; 17P; 17α-hydroxyprogesterone; 17,20bP; 17,20β-dihydroxy-4-pregnen-3-one; 20b-HSD; 20β-hydroxysteroid dehydrogenase; 20βS; 17,20β,21-trihydroxy-4-pregnen-3-one; actRIIB; activin rec
Keywords: دامنه اتصال لیگاند; PR; progesterone receptor; SHR; steroid hormone receptor; CoR; co-regulatory protein; LBD; ligand-binding domain; DBD; DNA-binding domain; NTD; amino-terminal domain; ID; intrinsically disordered; AF; activation function; HDX; hydrogen-deuterium exchang
Keywords: دامنه اتصال لیگاند; Ciona intestinalis; Botryllus schlosseri; Pregnane X receptor; Saccharomyces cerevisiae; Marine biotoxins; Bioassay; AD; activation domain; AF-2; transcription activation function domain; BsVDR/PXRα; Botryllus schlosseri VDR/PXR orthologue α; BPA; bisph
Keywords: دامنه اتصال لیگاند; AA; abiraterone acetate; ADT; androgen deprivation therapy; AR; androgen receptor; AR-V; AR splice variant; CRPC; castration-resistant prostate cancer; CTC; circulating tumor cell; CYP; cytochrome P450; FDA; Food and Drug Administration; LBD; ligand-bindi
Keywords: دامنه اتصال لیگاند; AR; androgen receptor; CAR; constitutive androstane receptor; DBD; DNA-binding domain; EDC; endocrine disrupting chemical; ER; estrogen receptor; FXR; farnesoid X receptor; GR; glucocorticoid receptor; HRE; hormone responsive elements; LBD; ligand-binding
Keywords: دامنه اتصال لیگاند; Ac; Aplysia californica; CH-IMI; nitromethylene analogue of imidacloprid; IMI; imidacloprid; LBD; ligand-binding domain; Ls; Lymnaea stagnalis; nAChR; nicotinic acetylcholine receptor; NIA; propargyl propyl phenylphosphonate (Niagara 16388); QSAR; quantit
Keywords: دامنه اتصال لیگاند; Macrophage; dendritic cell; lipid; nuclear receptor; retinoid X receptor; retinoic acid receptor; peroxisome proliferator-associated receptor; liver X receptor; vitamin D receptor; rheumatoid arthritis; inflammatory bowel disease; systemic lupus erythemat
Identification of novel quinazolinedione derivatives as RORγt inverse agonist
Keywords: دامنه اتصال لیگاند; AUC; area under the plasma concentration-time curve; BA; bioavailability; EAE; experimental autoimmune encephalomyelitis; LBD; ligand-binding domain; RORγt; retinoic acid receptor-related orphan receptor-gamma t; SAR; structure-activity relationship; T
Intrinsically disordered N-terminal domain of the Helicoverpa armigera Ultraspiracle stabilizes the dimeric form via a scorpion-like structure
Keywords: دامنه اتصال لیگاند; NRs; nuclear receptors; NTD; N-terminal domain; DBD; DNA-binding domain; LBD; ligand-binding domain; EcR; ecdysone receptor; Usp; Ultraspiracle; IDR; intrinsically disordered region; HaUsp; Usp from Helicoverpa armigera; HaUsp_ÎNTD; Usp from Helicoverpa
Molecular cloning of androgen receptor and gene expression of sex steroid hormone receptors in the brain of newborn Chinese alligator (Alligator sinensis)
Keywords: دامنه اتصال لیگاند; AR; androgen receptor; ARα and ARβ; androgen receptor alpha and androgen receptor beta; ESR1; estrogen receptor 1; ESR2; estrogen receptor 2; PR; progesterone receptor; TSD; temperature-dependent sex determination; SFA; State Forest Administration; ARCC
Natural products as modulators of the nuclear receptors and metabolic sensors LXR, FXR and RXR
Keywords: دامنه اتصال لیگاند; Natural products; Nuclear receptors; Liver X receptor; Farnesoid X receptor; Retinoid X receptor; Metabolic syndrome; Precision medicine; 6-ECDCA; 6α-ethyl-chenodeoxycholic acid (obeticholic acid); AA; arachidonic acid; ABC; ATP-binding cassette transpor
SRC2-3 binds to vitamin D receptor with high sensitivity and strong affinity
Keywords: دامنه اتصال لیگاند; VDR; vitamin D receptor; LBD; ligand-binding domain; DRIP; vitamin D receptor interacting protein; SRC; steroid receptor coactivator; SPR; surface plasmon resonance; AF2; activation-function 2; Vitamin D; Nuclear receptor; Coactivator; SRC2-3; Surface pla
Disruption of a putative intersubunit electrostatic bond enhances agonist efficacy at the human α1 glycine receptor
Keywords: دامنه اتصال لیگاند; β-ABA; β-aminobutyric acid; β-AIBA; β-aminoisobutyric acid; GlyR; glycine receptor; LBD; ligand-binding domain; MBS; Modified Barth's Saline; Popen; probability of channel being open; SEM; standard error of the mean; Ï; dwell-time; TM; transmembran
Structural basis for differential activities of enantiomeric PPARγ agonists: Binding of S35 to the alternate site
Keywords: دامنه اتصال لیگاند; PPAR; peroxisome proliferator-activated receptor; LBD; ligand-binding domain; LBP; ligand-binding pocket; TZD; thiazolidinedione; Cdk5; cyclin-dependent kinase 5; SRC-1; steroid receptor coactivator-1; r.m.s.; root-mean-square; Crystal structure; Alternat
GRIN2B gain of function mutations are sensitive to radiprodil, a negative allosteric modulator of GluN2B-containing NMDA receptors
Keywords: دامنه اتصال لیگاند; GRIN2B; Mutation; Encephalopathy; Electrophysiology; Radiprodil; NMDA inhibitors; ANOVA; analysis of variance; ATD; amino-terminal domain; DMSO; dimethyl sulfoxide; LBD; ligand-binding domain; NAM; negative allosteric modulator; NMDA; N-methyl-d-aspartate
A novel NMDA receptor positive allosteric modulator that acts via the transmembrane domain
Keywords: دامنه اتصال لیگاند; NMDA receptor; Positive allosteric modulator; Transmembrane domain; ATD; amino terminal domain; iGluR; ionotropic glutamate receptor; LBD; ligand-binding domain; NAM; negative allosteric modulator; PAM; positive allosteric modulator; TMD; transmembrane do
Mechanism and properties of positive allosteric modulation of N-methyl-d-aspartate receptors by 6-alkyl 2-naphthoic acid derivatives
Keywords: دامنه اتصال لیگاند; l-glutamate; N-methyl-d-aspartate; Potentiator; Positive allosteric modulator; Deactivation; Ligand-binding domain;
Characterization of rodent constitutively active estrogen receptor α variants and their constitutive transactivation mechanisms
Keywords: دامنه اتصال لیگاند; AF-1; activation function-1; AF-2; activation function-2; AR; androgen receptor; CTERP; C-terminally-truncated estrogen receptor α product; E2; 17β-estradiol; ERα; estrogen receptor α; ERα66; 66-kDa estrogen receptor α; ERαÎ5; Îexon 5 estrogen re
RNAi suppression of nuclear receptor genes results in increased susceptibility to sulfoxaflor in brown planthopper, Nilaparvata lugens
Keywords: دامنه اتصال لیگاند; AHR; aryl hydrocarbon receptor; BLAST; basic local alignment search tool; CAR; constitutive androstane receptor; CYP; cytochrome P450; DBD; DNA-binding domain; ERR; estrogen-related receptor; EST; expressed sequence tag; GR; glucocorticoid receptor; HNF4;
Molecular cloning of ESR2 and gene expression analysis of ESR1 and ESR2 in the pituitary gland of the Chinese alligator (Alligator sinensis) during female reproductive cycle
Keywords: دامنه اتصال لیگاند; ESRs; estrogen receptors; ERα/ESR1; estrogen receptor alpha; ERβ/ ESR2; ESTROGEN receptor beta; cDNA; DNA complementary to RNA; mRNA; Messenger RNA; PCR; polymerase chain reaction; RT; reverse transcription; qPCR; quantitative real-time PCR; 3D; three d
Identification of novel inverse agonists of estrogen-related receptors ERRγ and ERRβ
Keywords: دامنه اتصال لیگاند; ERRs; estrogen-related receptors; ER; estrogen receptor; NRs; nuclear receptors; LBD; ligand-binding domain; SAR; structureactivity relationship; MCAD; medium-chain acyl coenzyme A dehydrogenase; IC50; half maximal inhibitory concentration; Estrogen-relat
Radioligand binding assay for accurate determination of nuclear retinoid X receptors: A case of triorganotin endocrine disrupting ligands
Keywords: دامنه اتصال لیگاند; ATRA; all-trans retinoic acid; Bmax; maximal binding capacity (pmol/mg); DNA; deoxyribonucleic acid; DR; direct repeat; DTT; 1,4-dithiothreitol; FXR; farnesoid X receptor; Ka; affinity (l/mol); LBD; ligand-binding domain; LXR; liver X receptor; PMSF; phen
The antiproliferative and proapoptotic effects of cladosporols A and B are related to their different binding mode as PPARγ ligands
Keywords: دامنه اتصال لیگاند; CAD; caspase-activated deoxyribonuclease; CRC; colorectal cancer; HR-ESI-MS; high resolution electrospray ionization mass; LBD; ligand-binding domain; MDA; malondialdehyde; NCoEx; nuclear corepressor exchange factor; PPARs; peroxisome proliferator-activat
Cell-based and in silico evidence against quercetin and structurally-related flavonols as activators of vitamin D receptor
Keywords: دامنه اتصال لیگاند; CAS; chemical abstracts service; CYP24A1; cytochrome P450 24A1; DMSO; dimethyl sulfoxide; hRXRα; human retinoid X receptor alpha; hSRC-1; human steroid receptor coactivator-1; hVDR; human vitamin D receptor; mVDR; mouse vitamin D receptor; LBD; ligand-bi
ATF3 inhibits PPARγ-stimulated transactivation in adipocyte cells
Keywords: دامنه اتصال لیگاند; aP2; adipocyte fatty acid binding protein; ATF3; activation transcription factor 3; ATF/CRE; ATF/CREB responsive element; ChIP; chromatin immunoprecipitation; ER; endoplasmic reticulum; LBD; ligand-binding domain; PPARγ; peroxisome proliferator activated
The unfulfilled gene and nervous system development in Drosophila
Keywords: دامنه اتصال لیگاند; Burs; bursicon; CCAP; crustacean cardioactive peptide; DBD; DNA-binding domain; EH; eclosion hormone; fax-1; fasciculation of axons defective-1; GFP; green fluorescent protein; KC; Kenyon cells; LBD; ligand-binding domain; MARCM; mosaic analysis with a re
Fine tuning of agonistic/antagonistic activity for vitamin D receptor by 22-alkyl chain length of ligands: 22S-Hexyl compound unexpectedly restored agonistic activity
Keywords: دامنه اتصال لیگاند; VDR; vitamin D receptor; LBD; ligand-binding domain; 1α,25-(OH)2D3; 1α,25-dihydroxyvitamin D3; SERM; selective estrogen receptor modulator; ERα; estrogen receptor α; PPARγ; peroxisome proliferator-activated receptor γ; Vitamin D; Nuclear receptor; X
Synthesis, biological evaluation and molecular modeling studies of the PPARβ/δ antagonist CC618
Keywords: دامنه اتصال لیگاند; PPARβ/δ; Antagonist; Covalent; Cys249; LC-MS/MS; PPAR; peroxisome proliferator-activated receptor; LC-MS; liquid chromatography - mass spectrometry; LBD; ligand-binding domain; LBP; ligand-binding pocket; ABC; ammonium bicarbonate;
A step ahead of PPARγ full agonists to PPARγ partial agonists: Therapeutic perspectives in the management of diabetic insulin resistance
Keywords: دامنه اتصال لیگاند; DIO mouse; diet-induced obesity mouse; LBD; ligand-binding domain; PPAR; peroxisome proliferator-activated receptor; RXR; retinoid X receptor; SGK-1; serum/glucocorticoid-regulated kinase-1; T2DM; type 2 diabetes mellitus; ZDF rat; Zucker Diabetic Fatty r
Tunicate pregnane X receptor (PXR) orthologs: Transcript characterization and natural variation
Keywords: دامنه اتصال لیگاند; AF-1; transcription activation function 1; AR; androgen receptor; BsVDR/PXRα; Botryllus schlosseri VDR/PXR ortholog α; BSA; bovine serum albumin; bp; base pair; CAR; constitutive androstane receptor; CiVDR/PXRα; Ciona intestinalis VDR/PXR ortholog α;
L312, a novel PPARγ ligand with potent anti-diabetic activity by selective regulation
Keywords: دامنه اتصال لیگاند; BAT; Brown adipose tissue; CBP; cAMP responsive element binding protein (CREBP) binding protein; CDK5; Cyclin-dependent kinase 5; EC50; half-maximal effective concentration; FFA; Free fatty acids; HOMA-IR; HOMA of insulin resistance; ITT; Insulin toleranc
Environmental contaminants activate human and polar bear (Ursus maritimus) pregnane X receptors (PXR, NR1I2) differently
Keywords: دامنه اتصال لیگاند; CMV; cytomegalovirus; DBD; DNA-binding domain; GAL4; yeast regulatory protein GAL4; hPXR; human PXR; LBD; ligand-binding domain; NR1I2; nuclear receptor subfamily 1 group I member 2, a. k. a pregnane X receptor; pbPXR; polar bear PXR; PXR; pregnane X rece
N-terminal targeting of androgen receptor variant enhances response of castration resistant prostate cancer to taxane chemotherapy
Keywords: دامنه اتصال لیگاند; Prostate cancer; Androgen signaling; Taxanes; Therapeutic resistance; Epithelial-mesenchymal transition; ADT; androgen deprivation therapy; AR; androgen receptor; AR-V; androgen receptor splice variant; CRPC; castration-resistant prostate cancer; DHT; dih
Utility of an appropriate reporter assay: Heliotrine interferes with GAL4/upstream activation sequence-driven reporter gene systems
Keywords: دامنه اتصال لیگاند; Firefly luciferase inhibition; Nuclear receptor; Transactivation assay; LBD; ligand-binding domain; DBD; DNA-binding domain; UAS; upstream activating sequence; PXR; pregnane X receptor; mRNA; messenger RNA;
A ligand-entry surface of the nuclear receptor superfamily consists of the helix H3 of the ligand-binding domain
Keywords: دامنه اتصال لیگاند; hAR; human androgen receptor; hCAR; human constitutive androstane receptor; hCOUP-TFI; human chicken ovalbumin upstream promoter-transcription factor-I; hCOUP-TFII; human chicken ovalbumin upstream promoter-transcription factor-II; ssDAF-12; Strongyloides
A novel dualistic profile of an allosteric AMPA receptor modulator identified through studies on recombinant receptors, mouse hippocampal synapses and crystal structures
Keywords: دامنه اتصال لیگاند; ACSF; artificial cerebrospinal fluid; AMPA; 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid; BDNF; brain-derived neurotrophic factor; CA1; cornu ammonis area 1; CTZ; cyclothiazide; DEPC; diethylpyrocarbonate; DMSO; dimethyl sulfoxide; fEPSP; fie
Droplet digital polymerase chain reaction assay for screening of ESR1 mutations in 325 breast cancer specimens
Keywords: دامنه اتصال لیگاند; LBD; ligand-binding domain; ERα; estrogen receptor α; NGS; next generation sequencing; ER+; ER-positive; AIs; aromatase inhibitors; MBC; metastatic breast cancer; ddPCR; droplet digital polymerase chain reaction; FFPE; formalin-fixed paraffin embedded;
Stereoselective synthesis, biological evaluation, and modeling of novel bile acid-derived G-protein coupled Bile acid receptor 1 (GP-BAR1, TGR5) agonists
Keywords: دامنه اتصال لیگاند; GPCR; G protein-coupled receptor; BAs; bile acids; CDCA; chenodeoxycholic acid; CA; cholic acid; LCA; lithocholic acid; UDCA; ursodeoxycholic acid; FXR; farnesoid X receptor; NRs; nuclear receptors; LBD; ligand-binding domain; cAMP; cyclic adenosine monop
The dipeptide H-Trp-Glu-OH (WE) shows agonistic activity to peroxisome proliferator-activated protein-α and reduces hepatic lipid accumulation in lipid-loaded H4IIE cells
Keywords: دامنه اتصال لیگاند; WE; H-Trp-Glu-OH; PPARs; peroxisome proliferator-activated proteins; LBD; ligand-binding domain; SPR; surface plasmon resonance; TR-FRET; time-resolved fluorescence resonance energy transfer; FATP4; fatty-acid transport protein 4; ACS; acyl-CoA synthetase
Molecular cloning and mRNA tissue expression of thyroid hormone receptors in yellow catfish Pelteobagrus fulvidraco and Javelin goby Synechogobius hasta
Keywords: دامنه اتصال لیگاند; DBD; DNA-binding domain; LBD; ligand-binding domain; MS-222; 3-aminobenzoic acid ethyl ester methanesulfonate; Q-PCR; real-time quantitative PCR; RACE; rapid amplification of cDNA ends; TH; thyroid hormones; TR; thyroid hormone receptors; Pelteobagrus ful
Research ArticleCharacterization of a novel PXR isoform with potential dominant-negative properties
Keywords: دامنه اتصال لیگاند; PXR; Pregnane X Receptor; TSS; transcription start site; DBD; DNA-binding domain; LBD; ligand-binding domain; CGI; CpG island; MSP PCR; Methylation-specific PCR; EMAS; Electrophoretic mobility shift assay; Hepatocyte; Nuclear receptor; Epigenetic regulati
Identification of a novel partial agonist of liver X receptor α (LXRα) via screening
Keywords: دامنه اتصال لیگاند; ABC; ATP-binding cassette; ApoE; apolipoprotein E; DRIP205; vitamin D receptor-interacting protein 205; FAS; fatty acid synthase; GAPDH; glyceraldehyde-phosphate dehydrogenase; HDL; high-density lipoprotein; LBD; ligand-binding domain; LXR; liver X recept
NR4A nuclear receptors are orphans but not lonesome
Keywords: دامنه اتصال لیگاند; 6-MP; 6-mercaptopurine; 9-cis-RA; 9-cis-retinoic acid; AMP; adenosine monophosphate; AMPK; AMP-activated protein kinase; Cam-kinase; calcium/calmodulin-dependent protein kinase; CREB; cAMP response element binding protein; DBD; DNA-binding domain; DSB; DN