Keywords: کانال های یونی لیگاند; 5HT3R; 5-hydroxytryptamine receptor, subtype 3; ATP; Adenosine triphosphate; BK; big potassium channels; Cho; cholesterol; CTD; C-terminal domain; ECD; extracellular domain; ELIC; Erwinia chrysanthemi ligand-gated ion channel; GABAAR; gamma-aminobutyric a
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Keywords: کانال های یونی لیگاند; Ligand-gated ion channels; Glycine receptors α; 3 subunit; Allosteric modulation; Glucose as channel modulator; Pain pathways; Gain-of-function mutant α; 3(P185L);
Keywords: کانال های یونی لیگاند; Ligand-gated ion channels; Allostery; Crystallography; Neurotransmitters; Binding sites;
Keywords: کانال های یونی لیگاند; Acethylcholine receptor; Protein allostery; Ligand-gated ion channels; Gating mechanism; Agonism; Antagonism
Keywords: کانال های یونی لیگاند; Bioaffinity chromatography; G-protein coupled receptors; Ligand-gated ion channels; ATP-binding cassette transporters
GABAA receptor: Positive and negative allosteric modulators
Keywords: کانال های یونی لیگاند; γ-Aminobutyric acid type A receptors; Inhibitory neurotransmission; CNS depressant drug target; Anxiolytics/sedatives/general anesthetics; Ethanol; GABA; γ-aminobutyric acid; GABAAR; GABAA receptors; LGIC; ligand-gated ion channels; PLGIC; pentameric LG
The dual modulatory effects of efavirenz on GABAA receptors are mediated via two distinct sites
Keywords: کانال های یونی لیگاند; Recombinant GABAA receptors; Adverse CNS side effects; Picrotoxin; AIDS; Antiretroviral; BDZ; benzodiazepine; CNS; central nervous system; DMSO; dimethyl sulfoxide; DZ; diazepam; EFAV; efavirenz; FLU; flumazenil; LGICs; ligand-gated ion channels; HEK293;
Progress in the discovery of small molecule modulators of the Cys-loop superfamily receptors
Keywords: کانال های یونی لیگاند; Cys-loop receptors; Ligand-gated ion channels; Nicotinic acetylcholine receptors; Serotonin type 3 receptors; γ-Aminobutyric acid receptor; Glycine receptors;
PharmacologyIon channels, receptors, agonists and antagonists
Keywords: کانال های یونی لیگاند; G-protein-coupled receptors; inverse agonists; ligand-gated ion channels; voltage-gated ion channels;
Imidacloprid and thiacloprid neonicotinoids bind more favourably to cockroach than to honeybee α6 nicotinic acetylcholine receptor: Insights from computational studies
Keywords: کانال های یونی لیگاند; nAChR; nicotinic acetylcholine receptor; Ac-AChBP; Aplysia californica-acetylcholine binding protein; LGICs; ligand-gated ion channels; GABA; gamma-aminobutyric acid; 5-HT3; 5-hydroxytryptamine receptor subtype 3; CHARMM; Chemistry at Harvard Molecular Me
Effects of monoterpenes on ion channels of excitable cells
Keywords: کانال های یونی لیگاند; Terpenes; Monoterpenes; Voltage-gated ion channels; Ligand-gated ion channels; TRP channels; ACh; Acetylcholine; CAP; Compound action potential; CNS; Central nervous system; DRG; Dorsal root ganglion; GABA; Gamma-aminobutyric acid; GPCR; G-protein coupled
Design and validation of a homogeneous time-resolved fluorescence cell-based assay targeting the ligand-gated ion channel 5-HT3A
Keywords: کانال های یونی لیگاند; Ligand-gated ion channels; 5-HT3A-R; Tag-lite; HTRF; Fluorescent probes;
Constrained geometric simulation of the nicotinic acetylcholine receptor
Keywords: کانال های یونی لیگاند; Nicotinic acetylcholine receptor; froda; first; Membrane protein; Cys-loop receptors; Ligand-gated ion channels
Ion channels, receptors, agonists and antagonists
Keywords: کانال های یونی لیگاند; G-protein-coupled receptors; inverse agonists; ligand-gated ion channels; voltage-gated ion channels
Moving through the gate in ATP-activated P2X receptors
Keywords: کانال های یونی لیگاند; purinergic receptor; structure; ligand-gated ion channels; gating; neurotransmitter
Synthesis of novel cognition enhancers with pyrazolo[5,1-c][1,2,4]benzotriazine core acting at γ-aminobutyric acid type A (GABAA) receptor
Keywords: کانال های یونی لیگاند; α7nACh-R; α7nicotinic acetylcoline receptor; AD; Alzheimer's disease; BMS; borane methylsulfide; Bz site/GABAA-R; benzodiazepine site on GABAA receptor; CMC; carboxymethylcellulose; CNS; central nervous system; DAZ; diazepam, 7-chloro-1-methyl-5-pheny
Moxidectin and the avermectins: Consanguinity but not identity
Keywords: کانال های یونی لیگاند; Avermectin; Ivermectin; Moxidectin; Nematode; Toxicity; ATP binding cassette transporter; Ligand-gated ion channels
The Haemonchus contortus UNC-49B subunit possesses the residues required for GABA sensitivity in homomeric and heteromeric channels
Keywords: کانال های یونی لیگاند; 5-HT3; serotonin (5-hydroxytryptamine)-gated ion channel receptor; AChBP; acetylcholine binding protein; cRNA; copy RNA; LGIC; ligand-gated ion channels; MS-222; 3-aminobenzoic acid ethyl ester, methanesulphonate salt; nAChR; nicotinic acetylcholine recep
Allostery in pharmacology: Thermodynamics, evolution and design
Keywords: کانال های یونی لیگاند; Receptor activation; Ligand-gated ion channels; Homo/hetero/tropic cooperativity; Thermodynamic discrimination of efficacy; Conformational fluctuations; Statistical–energetic couplingGABAA, A-type γ-aminobutyric acid; KNF, Koshland, Némethy and Filmer; MW
Cysteine accessibility analysis of the human alpha7 nicotinic acetylcholine receptor ligand-binding domain identifies L119 as a gatekeeper
Keywords: کانال های یونی لیگاند; Ligand-gated ion channels; Molecular modeling; Electrophysiology; Voltage clamp; Site-directed mutations; Signal transduction
Ion channels, receptors, agonists and antagonists
Keywords: کانال های یونی لیگاند; G-protein-coupled receptors; inverse agonists; ligand-gated ion channels; voltage-gated ion channels
Cave Canalem: How endogenous ion channels may interfere with heterologous expression in Xenopus oocytes
Keywords: کانال های یونی لیگاند; Endogenous ion channels; Voltage-gated ion channels; Ligand-gated ion channels; Heterologous expression; Xenopus oocytes;
A nomenclature for ligand-gated ion channels
Keywords: کانال های یونی لیگاند; Ligand-gated ion channels; Nomenclature;
Effect of homologous serotonin receptor loop substitutions on the heterologous expression in Pichia of a chimeric acetylcholine-binding protein with α-bungarotoxin-binding activity
Keywords: کانال های یونی لیگاند; α-Bungarotoxin; AChBP; Acetylcholine-binding protein; Serotonin receptor; Cys-loop; Ligand-gated ion channels
Design and expression of human α7 nicotinic acetylcholine receptor extracellular domain mutants with enhanced solubility and ligand-binding properties
Keywords: کانال های یونی لیگاند; α-bgtx; α-bungarotoxin; α7-dm-ECD; double mutant of the α7-ECD; α7-wt-ECD; wild-type of the α7-ECD; ACh; acetylcholine; AChBP; acetylcholine-binding protein; BSA; bovine serum albumin; CCh; carbamylcholine; CD; circular dichroism; DLS; dynamic light
Slow intracellular accumulation of GABAA receptor δ subunit is modulated by brain-derived neurotrophic factor
Keywords: کانال های یونی لیگاند; ligand-gated ion channels; internalization; hippocampus; PLCγ; PKC; biotinylation assay; ANOVA; analysis of variance; AP2; adapter protein 2; BDNF; brain-derived neurotrophic factor; GABARs; GABAA receptors; PBS; phosphate buffered saline; PDBu; phorbol
Ion channels, receptors, agonists and antagonists
Keywords: کانال های یونی لیگاند; G-protein-coupled receptors; inverse agonists; ligand-gated ion channels; voltage-gated ion channels
Cyclophane and acyclic cyclophane: Novel channel blockers of N-methyl-d-aspartate receptor
Keywords: کانال های یونی لیگاند; Cyclophane; Acyclic cyclophane; Ligand-gated ion channels; N-Methyl-d-aspartate receptor; Voltage-clamp recording; Xenopus oocytes; Open-channel blockers
Aequorin luminescence-based assay for 5-hydroxytryptamine (serotonin) type 3 receptor characterization
Keywords: کانال های یونی لیگاند; 5-HT3 receptor; Aequorin luminescence; HEK293 cells; Ca2+ influx; Ligand-gated ion channels
Molecular modelling of the GABAA ion channel protein
Keywords: کانال های یونی لیگاند; γ-Aminobutyric acid (GABA); γ-Aminobutyric acid type-A receptor (GABAA); Ligand-gated ion channels; Molecular modelling; Transmembrane domain; General anaesthetic
Functional and structural characterization of a protein based on analysis of its hydrogen bonding network by hydrogen bonding plot
Keywords: کانال های یونی لیگاند; Hydrogen bond; Protein structure; Cytochrome P450; Tertiary hydrogen bond; Hydrogen bonding network; Information flow; Ligand-gated ion channels
Chain length dependence of the interactions of bisquaternary ligands with the Torpedo nicotinic acetylcholine receptor
Keywords: کانال های یونی لیگاند; Torpedo nicotinic acetylcholine receptor; Bisquaternary agonists; Suberyldicholine; Xenopus oocyte expression; Ligand-gated ion channels
Functional expression of P2X7 receptors in non-neuronal cells of rat dorsal root ganglia
Keywords: کانال های یونی لیگاند; Excitable membrane and synaptic transmission; Ligand-gated ion channels; BzATP; 2â²,3â²-O-(4-benzoylbenzoyl)-ATP; PPADS; pyridoxal-phosphate-6-azophenyl-,2â²,4â²-disulphonic acid; TNP-ATP; trinitrophenyl-adenosine triphosphate; P2X7; A-317491; Pain; D
Cloning and expression of ligand-gated ion-channel receptor L2 in central nervous system
Keywords: کانال های یونی لیگاند; Ligand-gated ion channels; In silico cloning; L2 receptor; Hippocampal neurons; GFP; HEK293 cells; Immunolocalization;
Allosteric modulation of ligand-gated ion channels
Keywords: کانال های یونی لیگاند; Ligand-gated ion channels; Allosteric modulation; P2X receptors; Glutamate receptors; Nicotinic acetylcholine receptors; nAChRs; Divalent cations;
Chronic intermittent ethanol exposure enhances NMDA-receptor-mediated synaptic responses and NMDA receptor expression in hippocampal CA1 region
Keywords: کانال های یونی لیگاند; Excitable membranes and synaptic transmission; Ligand-gated ion channels; Alcohol; Glutamate; Rat; Slice; Field potential; Electrophysiology; Immunoblot;
Properties of presynaptic P2X7-like receptors at the neuromuscular junction
Keywords: کانال های یونی لیگاند; Excitable membranes and synaptic transmission; Ligand-gated ion channels; Vesicle release; Adenosine triphosphate; Terminals; Purinergic;
Fast neurotransmission in the rat medial preoptic nucleus
Keywords: کانال های یونی لیگاند; Excitable membranes and synaptic transmission; Ligand-gated ion channels; Medial preoptic nucleus; Synaptic transmission; Glutamate; GABA; 5-HT;
Cloning and characterization of the chick NMDA receptor subunit-1 gene
Keywords: کانال های یونی لیگاند; Excitable membranes and synaptic transmission; Ligand-gated ion channels; Avian; Gene regulation; Glutamate receptors;