Keywords: مهارکننده مکانیسم; Malt1; Malt1 inhibitors; Activity-based protein profiling; Mechanism-based inhibitor; Lymphoma;
مقالات ISI مهارکننده مکانیسم (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: مهارکننده مکانیسم; Covalent inhibitor; Targeted covalent inhibitor (TCI); Mechanism-based inhibitor; kinact/Ki; Warhead reactivity; Activity-based protein profiling (ABPP); Click chemistry;
Keywords: مهارکننده مکانیسم; Thrombin; Coumarins; Docking; Serine protease; Mechanism-based inhibitor
An improved synthesis of the potent and selective γ-glutamyl transpeptidase inhibitor GGsTop together with an inhibitory activity evaluation of its potential hydrolysis products
Keywords: مهارکننده مکانیسم; γ-Glutamyl transpeptidase; Mechanism-based inhibitor; GGsTop; Michael addition;
Phosphonate-based irreversible inhibitors of human γ-glutamyl transpeptidase (GGT). GGsTop is a non-toxic and highly selective inhibitor with critical electrostatic interaction with an active-site residue Lys562 for enhanced inhibitory activity
Keywords: مهارکننده مکانیسم; γ-Glutamyl transpeptidase; Phosphonate diesters; GGsTop; Mechanism-based inhibitor; Electrostatic interaction; Active-site residue Lys562; Selectivity; Cytotoxicity;
Aglycone-focused randomization of 2-difluoromethylphenyl-type sialoside suicide substrates for neuraminidases
Keywords: مهارکننده مکانیسم; Neuraminidase; Suicide substrate; Mechanism-based inhibitor; Focused library; Aglycone;
Reversible inactivation of bovine plasma amine oxidase by cysteamine and related analogs
Keywords: مهارکننده مکانیسم; Copper amine oxidase; Reversible inhibitor; Mechanism-based inhibitor; Cysteamine; Thiazolidine
To bind zinc or not to bind zinc: An examination of innovative approaches to improved metalloproteinase inhibition
Keywords: مهارکننده مکانیسم; Zinc-binding group; Mechanism-based inhibitor; MMP
Mechanism-based inhibitors of MenE, an acyl-CoA synthetase involved in bacterial menaquinone biosynthesis
Keywords: مهارکننده مکانیسم; Acyl-CoA synthetase; Mycobacterium tuberculosis; Staphylococcus aureus; Mechanism-based inhibitor; Antibiotic
Cyclobranol: A substrate for C25-methyl sterol side chains and potent mechanism-based inactivator of plant sterol methyltransferase
Keywords: مهارکننده مکانیسم; Sterol C24-methyltransferase; Mechanism-based inhibitor; Cyclobranol; Cycloartenol; Phytosterol; Sterol C-methylation
Inactivation of soybean sterol 24-C-methyltransferase by elongated sterol side chains at C26
Keywords: مهارکننده مکانیسم; Sterol methyltransferase; Mechanism-based inhibitor; Cycloartenol; Phytosterol; Sterol methylation
Inhibition of CYP2B4 by 2-ethynylnaphthalene: Evidence for the co-binding of substrate and inhibitor within the active site
Keywords: مهارکننده مکانیسم; Cytochrome P450; CYP2B4; Mechanism-based inhibitor; Reversible inhibition; Enzyme kinetics; Co-binding of substrate and inhibitor;
Highly potent 3-pyrroline mechanism-based inhibitors of bovine plasma amine oxidase and mass spectrometric confirmation of cofactor derivatization
Keywords: مهارکننده مکانیسم; Copper amine oxidase; Bovine plasma amine oxidase; Mechanism-based inhibitor; Enzyme inactivator; 3-Pyrroline;
γ-(Monophenyl)phosphono glutamate analogues as mechanism-based inhibitors of γ-glutamyl transpeptidase
Keywords: مهارکننده مکانیسم; γ-Glutamyl transpeptidase; γ-(Monophenyl)phosphono glutamate analogues; Mechanism-based inhibitor; Phosphonylation