Keywords: پذیرنده مایکل; Nitroalkene; Nitrooleate; Apoptosis; Cancer; ROS; Michael acceptor;
مقالات ISI پذیرنده مایکل (ترجمه نشده)
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Keywords: پذیرنده مایکل; Catalytic asymmetric reaction; Chiral ligand; 14-Addition; Michael acceptor; Non-linear effect;
Keywords: پذیرنده مایکل; Coumarin-pyrazolone hybrid; Fluorescence turn-on probe; Biothiols detection; Michael acceptor; ICT inhibition; DFT calculations;
Keywords: پذیرنده مایکل; PDA; pyridoxylamine; NBT; nitrobenzenethiol; ACD; allergic contact dermatitis; LLNA; local lymph node assay; SBF; Schiff Base Formers; MA; Michael acceptor; SN1/SN2; Nucleophilic Substitution (1 or 2); SNAr; Nucleophilic Substitution (aromatic); AA; acyla
Keywords: پذیرنده مایکل; Fluorescent probe; Michael acceptor; Malonyl urea (thiourea); Cyanide detection; Bioimaging;
Design and synthesis of pregnenolone/2-cyanoacryloyl conjugates with dual NF-κB inhibitory and anti-proliferative activities
Keywords: پذیرنده مایکل; Pregnenolone; NF-κB; 2-Cyanoacryloyl; Michael acceptor; Anti-proliferative activity;
Design, synthesis and biological evaluation of 3-substituted-2-oxindole hybrid derivatives as novel anticancer agents
Keywords: پذیرنده مایکل; 2-Oxindole derivatives; α-bromoacryloyl; Michael acceptor; In vitro antiproliferative activity; GSH depletion;
A novel quinazoline-based analog induces G2/M cell cycle arrest and apoptosis in human A549 lung cancer cells via a ROS-dependent mechanism
Keywords: پذیرنده مایکل; Reactive oxygen species; Cell cycle; G2/M arrest; Michael acceptor; Quinazoline;
Design, synthesis, and evaluation of curcumin derivatives as Nrf2 activators and cytoprotectors against oxidative death
Keywords: پذیرنده مایکل; Nrf2; Curcumin; Cytoprotective activity; Michael acceptor; Catechol;
Design, synthesis, and biological evaluation of anti-EV71 agents
Keywords: پذیرنده مایکل; Enterovirus 71; 3C protease inhibitor; Michael acceptor
Michael acceptor in gambogic acid—Its role and application for potent antitumor agents
Keywords: پذیرنده مایکل; Gambogic acid; Michael acceptor; Intramolecular hydrogen bond
N-Heterocyclic carbene catalyzed tail-to-tail oligomerization of N,N-dimethylacrylamide (DMAA) and the search for the Stetter reaction of DMAA with benzaldehyde
Keywords: پذیرنده مایکل; N-Heterocyclic carbene; Michael acceptor; Umpolung; Tail-to-tail oligomerization; Organocatalysis;
Design and synthesis of new non nucleoside inhibitors of DNMT3A
Keywords: پذیرنده مایکل; DNA methylation; DNMT3A; Reactive inhibitor; Michael acceptor;
Investigation of fatty acid conjugates of 3,5-bisarylmethylene-4-piperidone derivatives as antitumor agents and human topoisomerase-IIα inhibitors
Keywords: پذیرنده مایکل; Curcumin analogs; Fatty acid amides; 3,5-Bisarylmethylene-4-piperidones; Michael acceptor; Anti-oxidant; Cytostatic activity; Topoisomerase IIα inhibitors; QSAR
Protolichesterinic acid derivatives: α-Methylene-γ-lactones as potent dual activators of PPARγ and Nrf2 transcriptional factors
Keywords: پذیرنده مایکل; Protolichesterinic acid; α-Methylene-γ-lactones; Michael acceptor; Nrf2; PPARγ;
All trans 1-(3-arylacryloyl)-3,5-bis(pyridin-4-ylmethylene)piperidin-4-ones as curcumin-inspired antineoplastics
Keywords: پذیرنده مایکل; Curcumin; Michael acceptor; Anti-oxidant; Cytostatic activity; Topoisomerase II inhibitors; QSAR;
Stereoselective synthesis of side chain-functionalized tetrahydropyrans from 5-hexenols
Keywords: پذیرنده مایکل; Addition; Aerobic oxidation; Alkenol; Alkene; Bromocyclization; Catalysis; Dioxygen; Cobalt(II) complexes; Michael acceptor; Radical; Stereoselective synthesis; Tetrahydropyran;
Design, synthesis and biological evaluation of FLT3 covalent inhibitors with a resorcylic acid core
Keywords: پذیرنده مایکل; FLT3; Covalent inhibitor; Michael acceptor; Maleimide; Acrylamide; Resorcylic acid lactones;
Design, synthesis and biological evaluation of arylcinnamide hybrid derivatives as novel anticancer agents
Keywords: پذیرنده مایکل; Apoptosis; Phenylcinnamides; Michael acceptor; In vitro antiproliferative activity; GSH depletion; Oxidative stress;
Coumarin–indanedione conjugate as a doubly activated Michael addition type probe for the colorimetric and ratiometric fluorescent detection of cyanide
Keywords: پذیرنده مایکل; Michael acceptor; Coumarin; Indanedione; Ratiometric; Colorimetric; Cyanide
3-Amidocoumarins as chemodosimeters to trap cyanide through both Michael and intramolecular cyclization reaction
Keywords: پذیرنده مایکل; Michael acceptor; Cyclization reaction; Cyanide anion; Amidocoumarins
Chalcone derivatives as fluorescence turn-on chemosensors for cyanide anions
Keywords: پذیرنده مایکل; Chalcone derivative; Cyanide anion; Chemosensor; Turn-on fluorescence; Michael acceptor; Crystal structure
Synthesis of highly N-substituted indole library via conjugate additions of indoline and their synthetic tool potentials
Keywords: پذیرنده مایکل; Indoline; Conjugate addition; Michael acceptor; Substitution; Catalyst;
Aspartic vinyl sulfones: Inhibitors of a caspase-3-dependent pathway
Keywords: پذیرنده مایکل; Vinyl sulfone; Caspase-3 inhibitor; Michael acceptor; Irreversible inhibitor; Yeast cell-based assay;
α,β-Unsaturated monoterpene acid glucose esters: Structural diversity, bioactivities and functional roles
Keywords: پذیرنده مایکل; Carboxylic acid; Cuniloside; Eucalyptus; Glucosyl ester; Menthiafolic acid; Michael acceptor; Monoterpene glycoside; Monoterpenoid ester; Oleuropeic acid; Plant defence;
Synthesis and evaluation of vinyl sulfones as caspase-3 inhibitors. A structure–activity study
Keywords: پذیرنده مایکل; Vinyl sulfone; Caspase-3 inhibitor; Michael acceptor; Irreversible inhibitor
Synthesis and antitumor evaluation of methyl spongoate analogs
Keywords: پذیرنده مایکل; Synthesis; Methyl spongoate analogs; Cytotoxicity; Michael acceptor;
Dual irreversible kinase inhibitors: Quinazoline-based inhibitors incorporating two independent reactive centers with each targeting different cysteine residues in the kinase domains of EGFR and VEGFR-2
Keywords: پذیرنده مایکل; Dual; Irreversible; Kinase; Inhibitors; Quinazoline-based; Independent reactive centers; Cysteine residues; EGFR; VEGFR-2; KDR; Quinone; Michael acceptor; Epidermal; Growth; Factor; Receptor; Vascular; Endothelial
Regioselective construction of polysubstituted benzene ring from Baylis-Hillman adduct via [4+2] annulation strategy
Keywords: پذیرنده مایکل; Polysubstituted benzenes; Baylis-Hillman adducts; Michael acceptor;
Regioselective synthesis of pentasubstituted benzene derivatives: TBAF as an effective catalyst for the sequential Michael addition-intramolecular aldolization
Keywords: پذیرنده مایکل; Polysubstituted benzenes; Baylis-Hillman adducts; TBAF; Michael acceptor;
Regioselective synthesis of polysubstituted benzenes from Baylis-Hillman adducts via [4+2] annulation protocol
Keywords: پذیرنده مایکل; Polysubstituted benzenes; Baylis-Hillman adducts; Michael acceptor; Schweizer reagent;