Keywords: حمل و نقل پپتیده; absorption; computational ADME; efflux pumps; in vitro models; organic cation transporters; P-glycoprotein; peptide transporters; pulmonary delivery/absorption; ABC transporters; organic anion-transporting polypeptide transporters; BAL; bronchoalveolar l
مقالات ISI حمل و نقل پپتیده (ترجمه نشده)
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Keywords: حمل و نقل پپتیده; Prodrugs; Prednisolone; Peptide transporters; Efflux; Homogenate;
Keywords: حمل و نقل پپتیده; pharamcokinetics; drug interaction; intestinal absorption; peptide transporters; renal excretion; organic anion transporters; DDIs, drug-drug interactions; PEPT, H+/peptide transporter; OAT, organic anion transporter; OCT, organic cation transporter; ACEI
Keywords: حمل و نقل پپتیده; Nasal epithelium; Peptide transporters; Organic cation transporters; OCT1-3; OCTN1; OCTN2; PEPT1; PEPT2;
Carrier-Mediated Prodrug Uptake to Improve the Oral Bioavailability of Polar Drugs: An Application to an Oseltamivir Analogue
Keywords: حمل و نقل پپتیده; active transport; absorption potential; Caco-2 cells; cell culture; membrane transport and transporters; permeability; peptide transporters; prodrugs;
Synthesis and evaluation of 18F labeled FET prodrugs for tumor imaging
Keywords: حمل و نقل پپتیده; ASC; alanine-serine-cysteine preferring amino acid transporter system; ASCT2; system ASC transporter subtype 2; BCH; 2-amino-bicylo[2.2.1]heptane-2-carboxylic acid; FACBC; 3-[18F]fluoro-cyclobutyl-1-carboxylic acid; FC; flash chromatography; FDG; 2-[18F]f
Influence of overexpression of efflux proteins on the function and gene expression of endogenous peptide transporters in MDR-transfected MDCKII cell lines
Keywords: حمل و نقل پپتیده; Peptide transporters; MDCK cells; Efflux pumps; MDR transfection;
Proton-coupled oligopeptide transporter family SLC15: Physiological, pharmacological and pathological implications
Keywords: حمل و نقل پپتیده; Mimetic; Peptide; Peptide transporters; SLC15;
Transport of the Synthetic Opioid Peptide DADLE ([d-Ala2,d-Leu5]-Enkephalin) in Neuronal Cells
Keywords: حمل و نقل پپتیده; peptide transporters; active transport; drug transport; opioid peptides; cell-penetrating peptides; neuronal cells; retinal ganglion cell; peptide delivery;
The Effects of Media on Pharmaceutically Relevant Transporters in the Human HT-29 Adenocarcinoma Cell Line: Does Culture Media Need to be Controlled?
Keywords: حمل و نقل پپتیده; Caco-2 cells; peptide drug delivery; drug transport; in vitro models; transporters; peptide transporters; polymerase chain reaction; solute transporters; ABC transporters; permeability;
Stereoselective Evasion of P-glycoprotein, Cytochrome P450 3A, and Hydrolases by Peptide Prodrug Modification of Saquinavir
Keywords: حمل و نقل پپتیده; prodrugs; structure–activity relationship (SAR); P-glycoprotein; peptide transporters; metabolism; CYP enzymes; stability
Peptide Transporter 1 Is Responsible for Intestinal Uptake of the Dipeptide Glycylsarcosine: Studies in Everted Jejunal Rings from Wild-type and Pept1 Null Mice
Keywords: حمل و نقل پپتیده; in vitro models; intestinal absorption; membrane transport/transporters; peptide transporters; pharmacokinetics; transgenics;
Effect of Milk on the Pharmacokinetics of Oseltamivir in Healthy Volunteers
Keywords: حمل و نقل پپتیده; intestinal absorption; bioavailability; food interactions; peptide transporters; pharmacokinetics
Evaluation of Transport Mechanism of Prodrugs and Parent Drugs Formed by Intracellular Metabolism in Caco-2 Cells with Modified Carboxylesterase Activity: Temocapril as a Model Case
Keywords: حمل و نقل پپتیده; Caco-2 cells; prodrugs; metabolism; intestinal absorption; membrane transport; inhibition; transporters; peptide transporters; multidrug resistance-associated proteins; P-glycoprotein
Pdz Adaptors: Their Regulation of Epithelial Transporters and Involvement in Human Diseases
Keywords: حمل و نقل پپتیده; ABC transporters; cell biology; drug transport; membrane transporter; MRP; organic cation transporters (OCTs); peptide transporters; solute transporters
The Intestinal Absorption of a Prodrug of the mGlu2/3 Receptor Agonist LY354740 is Mediated by PEPT1: In Situ Rat Intestinal Perfusion Studies
Keywords: حمل و نقل پپتیده; peptide transporters; PEPT1; prodrugs; intestinal absorption; in situ intestinal perfusion; LY544344; LY354740; membrane transport/transporters; active transport; GlyâSar;
Drug transporters in the lung-do they play a role in the biopharmaceutics of inhaled drugs?
Keywords: حمل و نقل پپتیده; drug inhalation; pulmonary delivery; multidrug resistance transporters; peptide transporters; organic cation transporters; organic anion transporters; Calu-3 cells; isolated perfused lungs; cell culture; permeability;
Prodrugs of nucleoside analogues for improved oral absorption and tissue targeting
Keywords: حمل و نقل پپتیده; prodrugs; absorption; transport; peptide transporters; nucleoside transporters; permeability; drug targeting;
Transport of levovirin prodrugs in the human intestinal Caco-2 cell line
Keywords: حمل و نقل پپتیده; levovirin; prodrugs; hepatitis C; Caco-2 cells; transport; permeability; peptide transporters;