Keywords: Peptoid; Peptidomimetic; Cyclic; Suzuki cross-coupling; Biaryl;
مقالات ISI (ترجمه نشده)
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Keywords: Drug design; Protein-protein interaction; Structure; Small molecule; Antibody; Peptide; Peptidomimetic; Design de médicaments; Interaction protéine-protéine; Structure; Petite molécule; Anticorps; Peptide; Peptidomimétiques;
Keywords: Anticancer; Antileukemic; Goralatide; Peptide; Peptidomimetic;
Keywords: Adenoviral protease inhibitor; Irreversible inhibitor; Peptidomimetic; X-ray co-crystal structure; Epidemic keratoconjunctivitis (EKC)
Keywords: Peptide; Heterocycles; Peptidomimetic; Proline; Coupling;
Keywords: Protein-protein interaction; Computational tools; Inhibitor design; Peptidomimetic; Protein structure;
Keywords: Glycopeptide; Isostere; Peptidomimetic; Deacetylation; Carbohydrate; Chemical biology
Keywords: Peptidomimetic; Macrocycle; Friedel-Crafts; Diversity; NMR solution structure;
Keywords: HER3; Nanobody; in silico; Docking; Peptidomimetic;
Utilization of the p-nitrobenzyloxycarbonyl (pNZ) amine protecting group and pentafluorophenyl (Pfp) esters for the solid phase synthesis of spiroligomers
Keywords: Spiroligomer; Bis-amino acid; Peptidomimetic; Solid phase synthesis; P-Nitrobenzyl carbamate; Pentafluorophenyl ester;
Solid-phase parallel synthesis of 1,3,4-oxadiazole based peptidomimetic library as a potential modulator of protein-protein interactions
Keywords: 1,3,4-Oxadiazole; Peptidomimetic; Solid-phase;
In vitro and in silico studies of naphthoquinones and peptidomimetics toward Plasmodium falciparum plasmepsin V
Keywords: Malaria; Naphthoquinone; Peptidomimetic; PEXEL; Plasmepsin V; DABCYL; 4-((4-(dimethylamino)phenyl)azo)benzoic acid; DMSO; dimethyl sulfoxide; EDANS; 5-((2-aminoethyl)amino)naphthalene-1-sulfonic acid; FRET; fluorescence resonance energy transfer; HIV-1; h
Antimicrobial activity profiles of Amphiphilic Xanthone derivatives are a function of their molecular Oligomerization
Keywords: Peptidomimetic; Membrane targeting; Oligomer; Antibiotic; Lipopolysaccharide;
αvβ3 and α5β1 integrin-specific ligands: From tumor angiogenesis inhibitors to vascularization promoters in regenerative medicine?
Keywords: Angiogenesis; Integrins; Biomaterials; Peptidomimetic; Regenerative medicine; Tissue engineering; Vascularization;
Enhanced antimalarial activity of plasmepsin V inhibitors by modification of the P2 position of PEXEL peptidomimetics
Keywords: Plasmepsin; Malaria; Protease; Peptidomimetic; PEXEL; Trafficking; Abu; aminobutyric acid; Cav; canavanine; CyHexGly; cyclohexylglycine; CyPenGly; cyclopentylglycine; EtNva; beta-ethyl-norvaline; GFP; green fluorescent protein; HBTU; O-(benzotriazol-1-yl)
Bortezomib inhibits mammalian carbonic anhydrases
Keywords: Carbonic anhydrase; Boronic acid; Peptidomimetic; Antitumor agent;
A structural investigation of FISLE-412, a peptidomimetic compound derived from saquinavir that targets lupus autoantibodies
Keywords: Systemic lupus erythematosus (SLE); Autoimmune; Autoantibodies; Peptidomimetic; Anti-DNA antibody; DWEYS; Saquinavir; Structure-Activity Relationship (SAR);
Low-cost and multi-gram scale synthesis of chiral Nβ-Boc protected α-Nα-hydrazino diesters
Keywords: Peptidomimetic; Pseudopeptide; α-Nα-hydrazino diester; SN2 reaction;
The prolyl oligopeptidase inhibitor IPR19 ameliorates cognitive deficits in mouse models of schizophrenia
Keywords: Schizophrenia; Prolyl oligopeptidase; Cognition; Peptidomimetic; Animal model;
Influence of chain length on the activity of tripeptidomimetic antagonists for CXC chemokine receptor 4 (CXCR4)
Keywords: CXCR4 antagonist; Peptidomimetic; Scaffold;
Design of a doxorubicin-peptidomimetic conjugate that targets HER2-positive cancer cells
Keywords: HER2; Lung cancer; Breast cancer; Doxorubicin; Peptidomimetic; Conjugate;
Facile synthesis and 18F-radiolabeling of α4β1-specific LLP2A-aryltrifluoroborate peptidomimetic conjugates
Keywords: Peptidomimetic; Radiotracer; Integrin receptor; F-18;
Spiro sugar-isoxazolidine scaffold as useful polyfunctional building block for peptidomimetics design
Keywords: exo-Glycal; Sugar scaffold; Peptidomimetic; Isoxazolidine; Nitrone cycloaddition;
Bridging computational modeling with amino acid replacements to investigate GHS-R1a-peptidomimetic recognition
Keywords: GPCR; Ghrelin receptor; Molecular modeling; Molecular dynamics simulation; G-7039; Peptidomimetic; UYRHBGCCDMFEFE-FUZODLBNSA-P; ACDXOVOYAHGXRI-LETRWZBTSA-P; JAWOEBYWOJFJIK-ATUXXYJQSA-P;
Synthesis, photophysical properties of triazolyl-donor/acceptor chromophores decorated unnatural amino acids: Incorporation of a pair into Leu-enkephalin peptide and application of triazolylperylene amino acid in sensing BSA
Keywords: Triazolyl donor-acceptor unnatural amino acids; Click reaction; Photophysical; BSA sensing; Leu-enkephalin analogue; Peptidomimetic; β-Turn;
Identification and activity of inhibitors of the essential nematode-specific metalloprotease DPY-31
Keywords: Nematode; Anthelmintic; Metalloprotease inhibitor; Docking; Peptidomimetic;
A new class of ghrelin O-acyltransferase inhibitors incorporating triazole-linked lipid mimetic groups
Keywords: Ghrelin; Ghrelin O-acyltransferase; 1,2,3-Triazole; Serine acylation; Peptidomimetic
Structure-based discovery of small molecule hepsin and HGFA protease inhibitors: Evaluation of potency and selectivity derived from distinct binding pockets
Keywords: Serine protease; Peptidomimetic; Benzamidine; Hepsin; Matriptase; HGFA; Small-molecule; Therapeutic; c-MET; RON; HGF; MSP; Receptor tyrosine kinase; Cancer; Cell-signaling; Growth factor; Structure-based drug design; Enzyme inhibitor;
Design and synthesis of potential dual NK1/NK3 receptor antagonists
Keywords: Schizophrenia; Neurokinin receptors; Peptidomimetic; NK1/NK3 receptor antagonists;
Synthesis, biological evaluation, hydration site thermodynamics, and chemical reactivity analysis of α-keto substituted peptidomimetics for the inhibition of Plasmodium falciparum
Keywords: Malaria; Peptidomimetic; Falcipain; Cruzain; Drug resistance
Peptidomimetics of Arg-Phe-NH2 as small molecule agonists of Mas-related gene C (MrgC) receptors
Keywords: Mas-related gene (Mrg) receptors; Agonist; Peptidomimetic; Arginine mimetic;
Molecular cloning and functional characterization of the diapause hormone receptor in the corn earworm Helicoverpa zea
Keywords: GPCR; Neuropeptide; Insect; Peptidomimetic;
α-Helix mimetics: Outwards and upwards
Keywords: Protein-protein interaction; Rational design; Peptidomimetic; Proteomimetic;
A small molecule peptidomimetic that binds to c-KIT1 G-quadruplex and exhibits antiproliferative properties in cancer cells
Keywords: Click chemistry; FID assay; FRET melting assay; G-quadruplex DNA; Necrosis; Peptidomimetic;
De novo design and synthesis of a μ-conotoxin KIIIA peptidomimetic
Keywords: Conotoxin; Peptidomimetic; Sodium channel blocker; KIIIA; Pain;
Structural studies of β-hairpin peptidomimetic antibiotics that target LptD in Pseudomonas sp.
Keywords: Antibacterial; Conformation; Peptide; Peptidomimetic; Pseudomonas aeruginosa; Lipopolysaccharide transport; β-Barrel membrane protein;
Peptide backbone replacement of hepatitis C virus NS3 serine protease C-terminal cleavage product analogs: Discovery of potent succinamide inhibitors
Keywords: Hepatitis C NS3 protease; Peptide backbone replacement; Succinamide; Peptidomimetic;
High in vitro antimicrobial activity of β-peptoid-peptide hybrid oligomers against planktonic and biofilm cultures of Staphylococcus epidermidis
Keywords: Peptidomimetic; Biofilm; Cytotoxicity; Staphylococcus;
Substrate-based peptidomimetic inhibitors of the Murray Valley encephalitis virus NS2B/NS3 serine protease: A P1-P4 SAR study
Keywords: Murray Valley encephalitis; Agmatine; Peptidomimetic; NS2B/NS3; Protease inhibitor;
Intracellular targets for a phosphotyrosine peptidomimetic include the mitotic kinesin, MCAK
Keywords: Signal transduction; SH2 domain; Drug delivery; Peptidomimetic; Kinesin; MCAK;
Evaluation of insect CAP2b analogs with either an (E)-alkene, trans- or a (Z)-alkene, cis-Pro isostere identifies the Pro orientation for antidiuretic activity in the stink bug
Keywords: Antidiuretic; Stink bug; Peptidomimetic; Neuropeptide; Cyclic
Design, synthesis and characterization of peptidomimetic conjugate of BODIPY targeting HER2 protein extracellular domain
Keywords: BODIPY; Breast cancer; EGFR; Protein–protein interactions; HER2; Peptidomimetic; Phosphorylation
Modulation of αvβ3- and α5β1-integrin-mediated adhesion by dehydro-β-amino acids containing peptidomimetics
Keywords: Dehydro-β-amino acids; Peptidomimetic; Cell adhesion; Signaling; Drug discovery
Cyclization of peptoids by formation of boronate esters
Keywords: Peptoid; Boronic acid; Peptidomimetic; Boronate ester; β-d-Galactose;
Studying protein-peptide interactions using benzophenone units: A case study of protein kinase B/Akt and its inhibitor PTR6154
Keywords: Peptidomimetic; Protein-protein interaction; Benzophenone; Protein kinase B (PKB/Akt); Solid phase peptide synthesis (SPPS);
Kappa agonist CovX-Bodies
Keywords: Kappa agonist; Bioconjugation; Peptidomimetic;
Long-acting peptidomimetics based DPP-IV inhibitors
Keywords: Peptidomimetic; DPP-IV inhibitors; Slow-binding; Selectivity; Antidiabetic; Long-acting
Proteasome inhibitors for cancer therapy
Keywords: BOP; (benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; DMSO; dimethyl sulfoxide; HMPA; hexamethyl phosphoramide; HOBt; 1-hydroxybenzotriazole; NMM; N-methylmorpholine; DMF; N,N-dimethyformamide; LDA; lithium diisopropylamide; THF;
Affinity of the alpha4–beta1 integrin-targeting peptide LLP2A to canine lymphoma
Keywords: Canine; Lymphoma; Peptidomimetic; Non-Hodgkin's; LLP2A
Synthesis of fluorinated N-aminoaziridines: access to new CF3-peptidomimetics
Keywords: N-Amino aziridine; Fluorine; Peptidomimetic; Iodobenzene diacetate; Amino acids;