Keywords: فارماکوکور; Anticonvulsant; Pharmacophore; Benzothiazole; Pyridazinone; GABA AT;
مقالات ISI فارماکوکور (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: فارماکوکور; Alzheimer's disease; AChE inhibitors; Dual binding ligands; Fusing approach; Hybrid molecules; Linking strategy; MTDL; Pharmacophore;
Keywords: فارماکوکور; Aminobenzothiazole; Molecular docking; NCI; Pharmacophore; Pharmacokinetics; Pyrimidine; Tyrosine kinase;
Keywords: فارماکوکور; Prostate cancer; Cell proliferation; Phenoxyphenol; Pharmacophore;
Keywords: فارماکوکور; Biological activity; Drug design; Pharmacophore; Structural proteome; Virtual screening;
Molecular dynamics simulation of the human estrogen receptor alpha: contribution to the pharmacophore of the agonists
Keywords: فارماکوکور; Human estrogen receptor alpha; Agonist; Pharmacophore; Molecular dynamics simulation;
Keywords: فارماکوکور; Nicotinonitrile; Bronchodilation; QSAR; Pharmacophore;
Keywords: فارماکوکور; Pharmacophore; Molecular docking; Aldose reductase; Poly (ADP-ribose) polymerase; Protein kinase C beta;
Keywords: فارماکوکور; Angiogenesis; PDGFR-β; Pharmacophore; QSAR; Virtual screening; PANC-1;
Keywords: فارماکوکور; Brassinolide; Brassinosteroids; Rice lamina inclination; In silico screening; Pharmacophore
Keywords: فارماکوکور; Computer-Aided Drug Discovery and Design (CADDD); Target prediction; Pharmacophore; Hit identification; Lead optimization; Cancer; Descubrimiento y diseño de fármacos asistidos por ordenador; Predicción de blancos; Farmacóforo; Identificación de hits
Keywords: فارماکوکور; ATX/NPP2; autotaxin; DIPEA; N,N-diisopropylethylamine; DMF; N,N-dimethylformamide; DMSO; dimethylsulfoxide; GPCR; G-protein coupled receptor; GRI; Genomic Research Institute; HBTU; O-(benzotriazol-1-yl)-N,N,Nâ²,Nâ²-tetramethyluronium hexafluorophosphate
Keywords: فارماکوکور; Acetylcholinesterase inhibitors; Alzheimer's; Pharmacophore; Molecular docking; Drug design
Keywords: فارماکوکور; Virtual screening; Anti-cancer agents; Pharmacophore; Molecular docking
Keywords: فارماکوکور; Protein engineering; Boron neutron capture therapy; Pharmacophore; Lysozyme;
Keywords: فارماکوکور; Antimycobacterial; Formononetin; Pharmacophore; Structure; Activity;
Keywords: فارماکوکور; Drug design; 3D-QSAR; Histamine H3 receptor; Histamine N-methyltransferase; Pharmacophore; Virtual screening;
Keywords: فارماکوکور; Functionalized piperidines; Green synthesis; Acetylcholinesterase (AChE) inhibition; Pharmacophore; Docking; In silico;
Keywords: فارماکوکور; Pyrrolyl phenoxy derivatives; Anti-tubercular activity; Enoyl ACP reductase; Pharmacophore; Surflex-docking; JUSJMWZCOYHWQQ-UHFFFAOYSA-N; PUKMLOGPPZYPQR-UHFFFAOYSA-N; NJIUEVYKBDORSJ-UHFFFAOYSA-N; WCROUCSRHKCYIS-UHFFFAOYSA-N; HYPUHOHBNPMMGW-UHFFFAOYSA-N; H
Keywords: فارماکوکور; Pharmacophore; Dibenzo-epine; Multifunctional compound;
Keywords: فارماکوکور; Chk2; Drug design; Pharmacophore; Virtual screening;
Keywords: فارماکوکور; VKZMICHNLVMXRJ-UAPYVXQJSA-N; Histamine; Histamine H3 receptor; Pharmacophore; Half-life; Pharmacokinetics;
Keywords: فارماکوکور; Drug target prediction; Molecular docking; Pharmacophore; A probabilistic fusion method;
Keywords: فارماکوکور; Autotaxin; Binary QSAR; Docking; Hydrophobic tunnel; Pharmacophore;
Keywords: فارماکوکور; 3D; three-dimensional; AchR; acetylcholine receptor; ASA; water-accessible surface area; BP; blood pressure; CHGA; chromogranin A; CST; catestatin; DBP; diastolic blood pressure; DSI; Data Sciences International (St. Paul, MN); HR; heart rate; NMR; nuclea
Keywords: فارماکوکور; 4-anilinoquinoline-3-carboxamide; EGFR-TK inhibitors; Pharmacophore; Docking study; Binding energy; Anti-proliferative activity;
Synthesis of 3-aza[4.4.3]propellanes with high Ï1 receptor affinity
Keywords: فارماکوکور; 3-Aza[4.4.3]propellane; Conformational restriction; Schmidt rearrangement; Stereochemistry; X-ray crystal structure; Ï ligands; Ï1 affinity; Selectivity; Pharmacophore;
Network pharmacology-based analysis of Chinese herbal Naodesheng formula for application to Alzheimer's disease
Keywords: فارماکوکور; Alzheimer's disease; Network pharmacology; Docking; Pharmacophore; Machine learning;
Design, synthesis and biological evaluation of new substituted 5-benzylideno-2-adamantylthiazol[3,2-b][1,2,4]triazol-6(5H)ones. Pharmacophore models for antifungal activity
Keywords: فارماکوکور; Adamantlythiazoles; Anti-inflammatory; Antibacterial; Antifungal; Pharmacophore; SAR;
Discovery and biological activity of computer-assisted drug designed Akt pathway inhibitors
Keywords: فارماکوکور; Akt kinase; Pharmacophore; Anti-tumor; Solenopsin; Molecular modeling;
Discovery, optimization and biological evaluation for novel c-Met kinase inhibitors
Keywords: فارماکوکور; c-Met; Virtual screening; Pharmacophore; X-ray crystallography; Structural optimization;
New insight into the action of tryptanthrins against Plasmodium falciparum: Pharmacophore identification via a novel submolecular QSAR descriptor
Keywords: فارماکوکور; Tryptanthrin; Quantitative structure activity relationship; Density functional theory; Pharmacophore; Malaria; Anti-malarial; P. falciparum; Scanning tunneling microscopy; Tunneling barrier;
Discovery of new Gyrase β inhibitors via structure based modeling
Keywords: فارماکوکور; Antibacterial; Anticancer; DNA Gyrase Î; Pharmacophore; Structure based analysis;
Putative dual inhibitors of Janus kinase 1 and 3 (JAK1/3): Pharmacophore based hierarchical virtual screening
Keywords: فارماکوکور; Autoimmune disorder; Docking; Janus kinase 1; Janus kinase 3; Pharmacophore; Prime MM/GBSA;
In-silico screening of small molecule inhibitors against Lactate Dehydrogenase (LDH) of Cryptosporidium parvum
Keywords: فارماکوکور; Lactate dehydrogenase; CpLDH; Molecular docking; Pharmacophore; De novo drug design; Molecular dynamics simulation;
Design, 3D QSAR modeling and docking of TGF-β type I inhibitors to target cancer
Keywords: فارماکوکور; TGF-β superfamily; Serine/threonine-kinase receptors; Binding database; 3D-QSAR; TGF-β-type I; TGF-β inhibitors; Pharmacophore; SB431542; Galunisertib;
Molecular determinants of PPARγ partial agonism and related in silico/in vivo studies of natural saponins as potential type 2 diabetes modulators
Keywords: فارماکوکور; Type 2 diabetes; Saponins; PPARγ; Partial agonists; Pharmacophore; Docking; CAT; catalase; GSH; reduced glutathione; HB; hydrogen bond; MDA; malondialdehyde; NADPH; beta-nicotinamide adenine dinucleotide 2â²-phosphate; PDB; Protein Data Bank; PPARγ;
Role of p53 circuitry in tumorigenesis: A brief review
Keywords: فارماکوکور; p53; miRNA; Mdm2; Pirh2; COP1; Ubiquitin; Proteasome; Modulators; Pharmacophore;
Design, synthesis and identification of novel substituted 2-amino thiazole analogues as potential anti-inflammatory agents targeting 5-lipoxygenase
Keywords: فارماکوکور; Design; Inflammation; 5-Lipoxygenase; Pharmacophore/docking; Thiazoles; AA; Arachidonic acid; DMF; N,N-dimethylformamide; DMSO; Dimethyl sulphoxide; DPPH; 2,2 -diphenyl-1-picrylhydrazyl; EDTA; Ethylenediaminetetra acetic acid; 5-HPETE; 5(S) hydroperoxyeic
Research articleVirtual screening of B-Raf kinase inhibitors: A combination of pharmacophore modelling, molecular docking, 3D-QSAR model and binding free energy calculation studies
Keywords: فارماکوکور; B-Raf kinase inhibitors; Virtual screening; Pharmacophore; Molecular docking; 3D QSAR; Binding free energy calculation;
Identification and validation of small molecule modulators of the NusB-NusE interaction
Keywords: فارماکوکور; Protein-protein interaction; NusB-NusE; Antibiotic; Pharmacophore; In silico screening;
A structure-activity relationship study of ABCC2 inhibitors
Keywords: فارماکوکور; ABC; ATP binding cassette; ABCC2; ATP binding cassette protein subfamily C member 2; CDCF; 5(6)-Carboxy-2â²,7â²-dichlorofluorescein; SAR; Structure-activity relationship; Transporter; MRP2; Modulator; Vesicle assay; Pharmacophore;
Dihydropyrazole and dihydropyrrole structures based design of Kif15 inhibitors as novel therapeutic agents for cancer
Keywords: فارماکوکور; Motor protein; Pharmacophore; QSAR; Virtual screening; Docking;
Research ArticlePharmacophore based 3D-QSAR modeling, virtual screening and docking for identification of potential inhibitors of β-secretase
Keywords: فارماکوکور; BACE1; β-secretase; AD; Alzheimer's disease; Aβ; amyloid-β; BBB; blood brain barrier; PDB; protein data bank; rmsd; root mean square deviation; IC50; inhibitory concentration; β-secretase; Alzheimer's disease; Pharmacophore; Virtual screening; Doc
Exploration of interaction zones of β-tubulin colchicine binding domain of helminths and binding mechanism of anthelmintics
Keywords: فارماکوکور; GTP; Guanosine triphosphate; RMSD; Root mean square deviation; RCSB; Research Collaboratory for Structural Bioinformatics; HBA; Hydrogen bond acceptor; Anthelmintics; β-tubulin; Colchicine; Structure-based model; Pharmacophore; Docking; Nematode;
Combined pharmacophore-guided 3D-QSAR, molecular docking and molecular dynamics studies for evodiamine analogs as DNA topoisomerase I inhibitors
Keywords: فارماکوکور; DNA topoisomerase I; Evodiamine; 3D-QSAR; Pharmacophore; Molecular docking; Molecular dynamics;
Multicomplex-based pharmacophore modeling coupled with molecular dynamics simulations: An efficient strategy for the identification of novel inhibitors of PfDHODH
Keywords: فارماکوکور; Malaria; Dihydroorotate dehydrogenase; Pharmacophore; Docking; Drug-likeness; Molecular dynamics;
Design, synthesis, molecular modeling and anti-hyperglycemic evaluation of quinazolin-4(3H)-one derivatives as potential PPARγ and SUR agonists
Keywords: فارماکوکور; Quinazolin-4(3H)-one; PPARγ; Sulfonylurea; Docking; Pharmacophore; QSAR; Anti-hyperglycemic; VOWUQQBKMFKUCG-UHFFFAOYSA-N;
Combretastatin A-4 based thiophene derivatives as antitumor agent: Development of structure activity correlation model using 3D-QSAR, pharmacophore and docking studies
Keywords: فارماکوکور; 3D-QSAR; Pharmacophore; Thiophene; Combretastatin A-4;
Rational design, synthesis, and structure-activity relationships of 5-amino-1H-pyrazole-4-carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors
Keywords: فارماکوکور; Protein tyrosine phosphatase 1B; Pharmacophore; Permeability; Hydrophobic; Oxadiazole;