Keywords: FAP, fibroblast activation protein; POP, prolyl oligopeptidase; TME, tumor microenvironment; DPPIV, dipeptidyl peptidase IV; ECM, extracellular matrix; IHC, immunohistochemistry; CAFs, cancer-associated fibroblasts; MMPs, matrix metalloproteinases
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A 914-bp promoter is sufficient to reproduce the endogenous prolyl oligopeptidase gene localization in the mouse placenta if not subject to position effect
Keywords: ANOVA, analysis of variance; E, embryonic day; EGFP, enhanced green fluorescent protein; LCR, locus control region; PCR, polymerase chain reaction; POP, prolyl oligopeptidase; qPCR, quantitative polymerase chain reaction; qRT-PCR, quantitative reverse tra
Characterization of a novel acylaminoacyl peptidase with hexameric structure and endopeptidase activity
Keywords: AAP, acylaminoacyl peptidase; PhAAP⁎, Pyrococcus horikoshii OT3 AAP (gene PH0863); PhAAP, Pyrococcus horikoshii OT3 AAP (gene PH0594); ApAAP, Aeropyrum pernix K1 AAP; POP, prolyl oligopeptidase; Ac, acetyl; Abz, 2-aminobenzoyl; Nap, 2-naphthylamide; Nan,
Glu88 in the non-catalytic domain of acylpeptide hydrolase plays dual roles: Charge neutralization for enzymatic activity and formation of salt bridge for thermodynamic stability
Keywords: APH, acylpeptide hydrolase; POP, prolyl oligopeptidase; apAPH, acylpeptide hydrolase from Aeropyrum pernix K1; IPTG, isopropyl-thiogalactopyranoside; Ac-Leu-pNA, Ac-Leu-p-nitroanilide; pNPC8, p-nitrophenyl caprylate; GdmCl, guanidine hydrochoride; DSC, di
The conserved N-terminal helix of acylpeptide hydrolase from archaeon Aeropyrum pernix K1 is important for its hyperthermophilic activity
Keywords: APH, acylpeptide hydrolase; POP, prolyl oligopeptidase; OB, oligopeptidase B; apAPH, APH protein from Aeropyrum pernix K1; E. coli, Escherichia coli; pNA, p-nitroanilide; pNPC8, p-nitrophenyl caprylate; WT, wild type protein; DSC, differential scanning ca
Baicalin, a prodrug able to reach the CNS, is a prolyl oligopeptidase inhibitor
Keywords: POP, prolyl oligopeptidase; SZ, schizophrenia; BD, bipolar affective disorder; IP3, inositol-1,4,5-P3; TCM, traditional Chinese medicine; STD, saturation transfer difference; DPPIV, dipeptidyl peptidase IV; CNS, central nervous system; FP-Rh, Fluorophospo
Novel Inhibitor for Prolyl Tripeptidyl Aminopeptidase from Porphyromonas gingivalis and Details of Substrate-recognition Mechanism
Keywords: PTP, prolyl tripeptidyl aminopeptidase; POP, prolyl oligopeptidase; DPIV, dipeptidyl aminopeptidase IV; PTP39, PTP truncated the 38 N-terminal residues; −βNA, -β-naphtykamide; -TBODA, 2-ter-butyl-[1, 3, 4]-oxadiazole; PAP, prolyl aminopeptidase; TMP, (2,
Fluorescence resonance energy transfer (FRET) peptides and cycloretro-inverso peptides derived from bradykinin as substrates and inhibitors of prolyl oligopeptidase
Keywords: POP, prolyl oligopeptidase; ACN, acetonitrile; DTT, dithiothreitol; Abz, ortho-aminobenzoic acid; EDDnp, N-(2,4-dinitrophenyl)ethylenediamine; tBu, tert-butyl; Fmoc, fluoren-9-ylmethoxycarbonyl; Pmc, 2,2,5,7,8-pentamethylchroman-6-sulfonyl; EDDP, N-[ethyl
Properties of the prolyl oligopeptidase homologue from Pyrococcus furiosus
Keywords: POP, prolyl oligopeptidase; Pfu, Pyrococcus furiosus; PCR, polymerase chain reaction; EDTA, ethylenediaminetetraacetatic acid; SDS–PAGE, sodium dodecyl sulfate polyacrylamide gel electrophoresis; Z, benzyloxycarbonyl; Nap, 2-naphthylamine; Nan, 4-nitroani
Peptide substrate profiling defines fibroblast activation protein as an endopeptidase of strict Gly2-Pro1-cleaving specificity
Keywords: FAP, fibroblast activation protein; DPP-4, dipeptidyl peptidase-4; POP, prolyl oligopeptidase; α2AP, α2-antiplasmin; cmk, chloromethyl ketone; AFC, 7-amino-4-trifluoromethyl coumarin; Ac, acetyl; EDANS, 5-[(2-Aminoethyl)amino]naphthalene-1-sulfonic acid;
Rigidity and Flexibility of Dipeptidyl Peptidase IV: Crystal Structures of and Docking Experiments with DPIV
Keywords: dipeptidyl peptidase (DPIV); serine proteinase; crystal structure; diabetes mellitus; flexibilityDPIV, dipeptidyl peptidase; POP, prolyl oligopeptidase; GLP, glucagon-like peptide; rmsd, root-mean-square deviation; tBu-GPI, tert-butyl-Gly-l-Pro-l-Ile; bor