Keywords: ساختار مجاز; Indolin-2-one; Privileged structure; Cytotoxicity; Molecular mechanism;
مقالات ISI ساختار مجاز (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: ساختار مجاز; Estrogen receptor; Antagonist; Diphenylamine; Privileged structure;
Keywords: ساختار مجاز; Guanidines; A2A receptor; Privileged structure; Iminoimidazoline; Tic-H; tetrahydroisoquinoline-hydantoin; A2AR; adenosine A2A receptor;
Design and synthesis of 2,6-disubstituted-8-amino imidazo[1,2a]pyridines, a promising privileged structure
Keywords: ساختار مجاز; Privileged structure; Amino-imidazopyridine; A2A receptor; Palladium-catalyzed coupling reaction;
5-Hydroxypyrido[2,3-b]pyrazin-6(5H)-one derivatives as novel dual inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H and integrase
Keywords: ساختار مجاز; HAART; HIV-1 dual inhibitors; HIV-1 IN; RNase H; 5-hydroxypyrido[2,3-b]pyrazin-6(5H)-one derivatives; Privileged structure;
A novel solid-phase synthetic method for production of N-alkyl-4-alkylamino-1-aryl-1H-pyrazolo[3,4-d]pyrimidine-6-carboxamide library
Keywords: ساختار مجاز; Screening library; Privileged structure; Heterocycle; Pyrazolopyrimidine; Solid-phase organic synthesis;
An expeditious and atom-economic synthesis of lead-like, medicinally important 4,5-dihydropyrazolo[1,5-a]pyrazin-6-ones
Keywords: ساختار مجاز; Propargylamine; Sonogashira coupling; Ynone; Pyrazole; Intramolecular alkylation; Atom efficiency; Lead-likeness; Privileged structure;
A tandem copper (II)-promoted synthesis of 2-substituted pyrrolo[2,1-f][1,2,4] triazin-4(3H)-ones
Keywords: ساختار مجاز; Tandem annulation; Cupric chloride; 1-Amino-1H-pyrrole-2-amides; Privileged structure; Pyrrolo[2,1-f][1,2,4]triazin-4(3H)-ones;
Synthesis of novel 2H-spiro[1-benzofuran-3,4â²-piperidin]ol scaffolds
Keywords: ساختار مجاز; MDQBJWIJWPVYCJ-UHFFFAOYSA-N; XFVSCQRPRNFUPL-UHFFFAOYSA-N; WPFCOAVXWHNSHP-UHFFFAOYSA-N; Spiro[benzofuran-piperidine]; Scaffold; Privileged structure; Intramolecular Heck reaction; SNAr;
Design and synthesis of 2-aminothiazole based antimicrobials targeting MRSA
Keywords: ساختار مجاز; Privileged structure; 2-Aminothiazole; Antimicrobial; MIC; MRSA;
Structure-based design and biological profile of (E)-N-(4-Nitrobenzylidene)-2-naphthohydrazide, a novel small molecule inhibitor of IκB kinase-β
Keywords: ساختار مجاز; anti-Inflammatory; IKK-β inhibitor; Molecular docking; N-Acylhydrazone; Privileged structure; Structure-based designAA, arachidonic acid; ATP, adenosine-5′-triphosphate; CA, capsid protein; CB2, cannabinoid receptor type-2; DSSP, definition of secondary s
Spiroindane based amides as potent and selective MC4R agonists for the treatment of obesity
Keywords: ساختار مجاز; Spiroindane; Amide; Privileged structure; Melanocortin subtype-4 receptor; MC4R; Agonist; MK-0489; Obesity;
Discovery of benzhydrylpiperazine derivatives as CB1 receptor inverse agonists via privileged structure-based approach
Keywords: ساختار مجاز; Benzhydrylpiperazine; Privileged structure; Cannabinoid receptor 1(CB1); Anti-obesity
Discovery of highly potent and efficacious MC4R agonists with spiroindane N-Me-1,2,4-triazole privileged structures for the treatment of obesity
Keywords: ساختار مجاز; Spiroindane; Triazole; Privileged structure; Melanocortin subtype-4 receptor; MC4R; Agonist; Obesity
Design and synthesis of isoform-selective phospholipase D (PLD) inhibitors. Part II. Identification of the 1,3,8-triazaspiro[4,5]decan-4-one privileged structure that engenders PLD2 selectivity
Keywords: ساختار مجاز; PLD; Phospholipase; Cancer; Privileged structure
Facile conversion of Biginelli 3,4-dihydropyrimidin-2(1H)-thiones to 2-(2-hydroxy-2-arylvinyl) dihydropyrimidines via Eschenmoser coupling
Keywords: ساختار مجاز; Eschenmoser; Sulfide contraction; Eschenmoser coupling; Polymer supported; Triphenylphosphine; DHPM; Biginelli; Privileged structure; Drug research;
Synthesis and antiproliferative activity of 2,4-disubstituted 6-aryl-7H-pyrrolo[3,2-d]pyrimidin-7-one 5-oxides
Keywords: ساختار مجاز; Pyrrolo[3,2-d]pyrimidine; Privileged structure; Antitumor drugs; Cell cycle arrest;
Synthesis and structure–activity relationships of pyrazolodiazepine derivatives as human P2X7 receptor antagonists
Keywords: ساختار مجاز; IL-1β; Privileged structure; Pyrazolodiazepine; P2X7 Receptor
Melanocortin subtype 4 receptor agonists: Structure–activity relationships about the 4-alkyl piperidine core
Keywords: ساختار مجاز; Obesity; Erectile dysfunction; Privileged structure; G-protein-coupled receptor; Apetite; Metabolic disorder; Peptidomimetic
Privileged structure based ligands for melanocortin receptors—4,4-Disubstituted piperidine derivatives
Keywords: ساختار مجاز; Melanocortin; MC4; Privileged structure; G-protein coupled receptors; GPCR
Optimization of a privileged structure leading to potent and selective human melanocortin subtype-4 receptor ligands
Keywords: ساختار مجاز; Privileged structure; Melanocortin-4
Privileged structure-based quinazolinone natural product-templated libraries: Identification of novel tubulin polymerization inhibitors
Keywords: ساختار مجاز; Privileged structure; Quinazolinone; Natural product-templated library; Tubulin polymerization inhibitors
Design and synthesis of 3,4-methylenedioxy-6-nitrophenoxyacetylhydrazone derivatives obtained from natural safrole: New lead-agents with analgesic and antipyretic properties
Keywords: ساختار مجاز; N-Acylhydrazone; Safrole; Analgesic activity; Antipyretic activity; 1,3-Benzodioxole derivatives; Privileged structure
1-Aryltetralin privileged structure-based libraries: parallel synthesis of N-aryl and N-biaryl γ-lactam lignans
Keywords: ساختار مجاز; Biaryls; Lactam lignans; Privileged structure; Tandem reaction; InCl3; Ligandless Suzuki reaction; Parallel solution-phase synthesis;
Antiproliferative activity in HL60 cells by tetrasubstituted pyrroles: a structure–activity relationship study
Keywords: ساختار مجاز; Pyrroles; Privileged structure; Leukemia; Antitumor drugs
New 2-bromomethyl-8-substituted-benzo[c]chromen-6-ones. Synthesis and biological properties
Keywords: ساختار مجاز; Substituted-benzo[c]chromen-6-one; Coumarin-isocoumarin; Privileged structure;