Keywords: پیریمتیامین; Minipig; Embryo-fetal development study; Mid-term fetal examinations; Pyrimethamine; Skeleton double staining;
مقالات ISI پیریمتیامین (ترجمه نشده)
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Keywords: پیریمتیامین; Intrinsic dissolution rate; Polymorph; Pyrimethamine; Solid dispersion; Thermogelling; Supramolecular synthon;
Keywords: پیریمتیامین; Drug resistence; Plasmodium falciparum; Mathematical model; Malaria; Optimal control; Pyrimethamine;
Keywords: پیریمتیامین; Extremely randomized trees; Decision trees; Structure-activity relationship; Molecular modeling; Antimalarials; Dihydrofolate reductase; Trimethoprim; Pyrimethamine; Cycloguanil; Hydrophobic feature;
Synergic in vitro combinations of artemisinin, pyrimethamine and methylene blue against Neospora caninum
Keywords: پیریمتیامین; Neospora caninum; Artemisinin; Methylene blue; Pyrimethamine;
Nicotinamide inhibits the growth of P. falciparum and enhances the antimalarial effect of artemisinin, chloroquine and pyrimethamine
Keywords: پیریمتیامین; Malaria; Nicotinamide; Artemisinin; Chloroquine; Pyrimethamine; Isobolographic analysis;
Evaluation of Renal Transporter Inhibition Using Creatinine as a Substrate In Vitro to Assess the Clinical Risk of Elevated Serum Creatinine
Keywords: پیریمتیامین; renal transporter; drug interactions; in vitro-in vivo correlation; renal clearance; inhibition; AUC; area under the concentration curve; CLcr; creatinine renal clearance; Cmax; maximal total plasma concentration; Cmax,u; maximal unbound plasma concen
A transgenic Neospora caninum strain based on mutations of the dihydrofolate reductase-thymidylate synthase gene
Keywords: پیریمتیامین; Neospora caninum; DHFR-TS; Transfection; Pyrimethamine; Lac-Z gene
The synthesis and biodistribution of [11C]metformin as a PET probe to study hepatobiliary transport mediated by the multi-drug and toxin extrusion transporter 1 (MATE1) in vivo
Keywords: پیریمتیامین; Positron emission tomography (PET); Metformin; Multi-drug and toxin extrusion transporter 1 (MATE1); Hepatobiliary transport; Pyrimethamine;
Effect of Nitaxozanide and Pyrimethamine on Astrocytes Infected by Toxoplasma gondii In Vitro
Keywords: پیریمتیامین; Effect; Nitazoxanide; Pyrimethamine; Toxoplasma infection; Astrocytes
Polymorphism in dhfr/dhps genes, parasite density and ex vivo response to pyrimethamine in Plasmodium falciparum malaria parasites in Thies, Senegal
Keywords: پیریمتیامین; Plasmodium falciparum; dhfr/dhps; Pyrimethamine; Resistance
Comparison of protein patterns between Plasmodium falciparum mutant clone T9/94-M1-1(b3) induced by pyrimethamine and the original parent clone T9/94
Keywords: پیریمتیامین; Plasmodium falciparum; Proteomics; Pyrimethamine; Drug resistance; Protein; Molecular target;
Capillary zone electrophoresis as a potential technique for the simultaneous determination of sulfadoxine and pyrimethamine in tablet formulations
Keywords: پیریمتیامین; Antimalarials; Sulfadoxine; Pyrimethamine; Tablets; Capillary zone electrophoresis
Antiplasmodial and antiulcer activities of Melanthera scadens
Keywords: پیریمتیامین; Melanthera scadens; Antiplasmodial activity; Antiulcer activity; Antimalarial activity; Antiulcerogenic activity; Chemical constituent; Parasitaemia; Plasmodium berghei; Artesunate; Indomethacin; Pyrimethamine;
Spectrophotometric determination of pyrimethamine (PYM) in pharmaceutical formulation using 1,2-naphthoquinone-4-sulfonate (NQS)
Keywords: پیریمتیامین; UV–visible spectrophotometry; Pyrimethamine; NQS; Pharmaceutical formulation
Long-term ocular outcome in congenital toxoplasmosis: A prospective cohort of treated children
Keywords: پیریمتیامین; Congenital toxoplasmosis; Toxoplasma gondii; Chorioretinitis; Visual impairment; Prenatal diagnosis; Pyrimethamine; Sulfadiazine; Spiramycin; Long-term care
Self-assembly of hydrogen-bonded supramolecular structures based on hexafluorosilicate anion
Keywords: پیریمتیامین; Hexafluorosilicate; Supramolecular structures; Hydrogen bonding; Crystal engineering; Thiabendazole; Pyrimethamine
Pharmacokinetic Properties and Bioequivalence of Two Sulfadoxine/Pyrimethamine Fixed-Dose Combination Tablets: A Parallel-Design Study in Healthy Chinese Male Volunteers
Keywords: پیریمتیامین; bioequivalence; LC-IDMS; parallel design; pharmacokinetic; pyrimethamine; sulfadoxine;
An open-label Phase I/II clinical trial of pyrimethamine for the treatment of patients affected with chronic GM2 gangliosidosis (Tay–Sachs or Sandhoff variants)
Keywords: پیریمتیامین; GM2 gangliosidosis; Pyrimethamine; Pharmacologic chaperone
Pyrimethamine increases β-hexosaminidase A activity in patients with Late Onset Tay Sachs
Keywords: پیریمتیامین; Late Onset Tay Sachs; Pyrimethamine; β-hexosaminidase A
Prediction of residues involved in inhibitor specificity in the dihydrofolate reductase family
Keywords: پیریمتیامین; DHFR; Dihydrofolate reductase; Hs; H. sapiens; Ec; E. coli; Mt; M. tuberculosis; Tb; T. brucei; Tg; T. gondii; Lm; L. major; Tc; T. cruzi; Pf; P. falciparum; Pv; P. vivax; Rn; R. norvegicus; Pc; P. carnii; Lc; L. casei; Ma; M. avium; MTX; Methotrexate; TM
Screening for inhibitors of the SOD1 gene promoter: Pyrimethamine does not reduce SOD1 levels in cell and animal models
Keywords: پیریمتیامین; Amyotrophic lateral sclerosis; SOD1; Superoxide dismutase; Assay; Compound screening; Pyrimethamine
Evaluation of the effect of pyrimethamine, an anti-malarial drug, on HIV-1 replication
Keywords: پیریمتیامین; Pyrimethamine; DHFR; Anti-malaria; S-phase; HIV-1 replication; Nucleoside analog
Methotrexate and aminopterin lack in vivo antimalarial activity against murine malaria species
Keywords: پیریمتیامین; Plasmodium berghei; Plasmodium yoelii yoelii; Plasmodium chabaudi and Plasmodium vinckei; Methotrexate; Aminopterin; Antifolate; Folate receptor; Pyrimethamine
Novel point mutations in sulfadoxine resistance genes of Plasmodium falciparum from India
Keywords: پیریمتیامین; Plasmodium falciparum; Sulfadoxine; Pyrimethamine; Dihydrofolate reductase (DHFR); Dihydropteroate synthase (DHPS)
Characterization, phase solubility and molecular modeling of α-cyclodextrin/pyrimethamine inclusion complex
Keywords: پیریمتیامین; α-CD; Inclusion complex; Pyrimethamine; Toxoplasmosis; Molecular modeling
Distinct haplotypes of dhfr and dhps among Plasmodium falciparum isolates in an area of high level of sulfadoxine–pyrimethamine (SP) resistance in eastern Sudan
Keywords: پیریمتیامین; dhfr; dhps haplotypes; Pyrimethamine; Sulfadoxine resistance; Plasmodium falciparum; Evolution; Sudan
Interaction of pyrimethamine and sulfadiazine with ionic and neutral micelles: Electronic absorption and fluorescence studies
Keywords: پیریمتیامین; Antitoxoplasmosis drugs; Pyrimethamine; Sulfadiazine; Surfactant; Micelles; Binding constant
Single-day, three-dose treatment with fixed dose combination artesunate/sulfamethoxypyrazine/pyrimethamine to cure Plasmodium falciparum malaria
Keywords: پیریمتیامین; Artesunate; Sulfamethoxypyrazine; Pyrimethamine; 24-hour therapy; Malaria; Plasmodium falciparum
Determination of kinetic parameters from isothermal calorimetry for interaction processes of pyrimethamine with chitosan derivatives
Keywords: پیریمتیامین; Isothermal calorimetry; Pyrimethamine; Adsorption kinetic modeling; Chitosan;
Inclusion complexes of pyrimethamine in 2-hydroxypropyl-β-cyclodextrin: Characterization, phase solubility and molecular modelling
Keywords: پیریمتیامین; 2-Hydroxypropyl-β-cyclodextrin; Pyrimethamine; Inclusion complex; Toxoplasmosis
Toxoplasma meningoencephalitis in HIV-seronegative patients: clinical patterns, imaging features and treatment outcome
Keywords: پیریمتیامین; Protozoan infection; Toxoplasma gondii; Cerebral toxoplasmosis; Encephalitis; Meningoencephalitis; Magnetic resonance imaging; Sulfadiazine; Pyrimethamine;
Validation of a liquid chromatography–mass spectrometry multi-residue method for the simultaneous determination of sulfonamides, tetracyclines, and pyrimethamine in milk
Keywords: پیریمتیامین; Sulfonamide; Tetracycline; Pyrimethamine; Milk; Antibiotics; LC-ESI-MS
Solid-phase extraction for multiresidue determination of sulfonamides, tetracyclines, and pyrimethamine in Bovine's milk
Keywords: پیریمتیامین; Sulfonamide; Tetracycline; Pyrimethamine; Solid-phase extraction; Antibiotics; Milk
Continued efficacy of sulfadoxine-pyrimethamine as second line treatment for malaria in children in Guinea-Bissau
Keywords: پیریمتیامین; Malaria; Children; Sulfadoxine; Pyrimethamine; Retreatment; Guinea-Bissau;
Plasmodium vivax dihydrofolate reductase point mutations from the Indian subcontinent
Keywords: پیریمتیامین; Malaria; Plasmodium vivax; Dihydrofolate reductase; Antifolate; Pyrimethamine; Point mutations; Drug resistance
Simultaneous quantification of α-/β-diastereomers of arteether, sulphadoxine and pyrimethamine: A promising anti-relapse antimalarial therapeutic combination, by liquid chromatography tandem mass spectrometry
Keywords: پیریمتیامین; Tandem mass spectrometry; Blood plasma; Sulphadoxine; Pyrimethamine; α-/β-Arteether
Equine Protozoal Myeloencephalitis: Treatment, Prognosis, and Prevention
Keywords: پیریمتیامین; Sarcocystis neurona; equine protozoal myeloencephalitis; treatment; nitazoxanide; ponazuril; toltrazuril; pyrimethamine; sulfonamide
Simple and cost-effective liquid chromatographic method for determination of pyrimethamine in whole blood samples dried on filter paper
Keywords: پیریمتیامین; Pyrimethamine; Sulfadoxine; Trimethoprim; Internal standard; Filter paper method;
Liquid chromatographic-mass spectrometric assay for simultaneous pyrimethamine and sulfadoxine determination in human plasma samples
Keywords: پیریمتیامین; Sulfadoxine; Pyrimethamine; Liquid chromatography; Mass spectrometry;
Simultaneous determination of pyrimethamine, sulfadiazine and N-acetyl-sulfadiazine in plasma for monitoring infants in treatment of congenital toxoplasmosis
Keywords: پیریمتیامین; Congenital toxoplasmosis; Plasma concentrations; Pyrimethamine; Sulfadiazine; N-Acetyl-sulfadiazine; LC-MS;
A validated HPLC method for determining residues of a dual active ingredient anti-malarial drug on manufacturing equipment surfaces
Keywords: پیریمتیامین; Cleaning validation; Cross-contamination; Anti-malarial drug; Pyrimethamine; Sulfadoxine; Reversed-phase liquid chromatography;