Keywords: پیرولوبenzodiazepines; Antibody-drug conjugates; Pyrrolobenzodiazepines; Macrocycles;
مقالات ISI پیرولوبenzodiazepines (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Access to the enantiopure pyrrolobenzodiazepine (PBD) dilactam nucleus via self-disproportionation of enantiomers
Keywords: پیرولوبenzodiazepines; Self-disproportionation of enantiomers; Pyrrolobenzodiazepines; Sublimation; Cooperative catalysis; 2,3-Dihydro-1H-pyrrole;
Topical delivery of anthramycin I. Influence of neat solvents
Keywords: پیرولوبenzodiazepines; Skin cancer; Anthramycin; Pyrrolobenzodiazepines; PBDs; Solvents; Permeation; Franz diffusion cell; Topical therapy;
Synthesis of a C2-aryl-pyrrolo[2,1-c][1,4]benzodiazepine monomer enabling the convergent construction of symmetrical and non-symmetrical dimeric analogs
Keywords: پیرولوبenzodiazepines; Pyrrolobenzodiazepines; Antibody-drug conjugates; Payloads; Drug-linker; Anti-cancer;
AlCl3-NaI assisted cleavage of polymer-bound esters with concomitant amine coupling and azido-reductive cyclization: synthesis of pyrrolobenzodiazepine derivatives
Keywords: پیرولوبenzodiazepines; Pyrrolobenzodiazepines; Solid-phase synthesis; Combinatorial chemistry; AlCl3-NaI; Azido-reductive cyclization; SLE method;
Hybrids of privileged structures benzothiazoles and pyrrolo[2,1-c] [1,4]benzodiazepin-5-one, and diversity-oriented synthesis of benzothiazoles
Keywords: پیرولوبenzodiazepines; Anti-cancer drugs; Privileged structures; Benzothiazoles; Pyrrolobenzodiazepines; Diversity-oriented synthesis
Synthesis and potential cytotoxic activity of new phenanthrylphenol-pyrrolobenzodiazepines
Keywords: پیرولوبenzodiazepines; Pyrrolobenzodiazepines; Phenanthrylphenol; DNA binding affinity; Anticancer activity; G1 cell cycle arrest; Apoptosis
Fluorescent 7-diethylaminocoumarin pyrrolobenzodiazepine conjugates: Synthesis, DNA interaction, cytotoxicity and differential cellular localization
Keywords: پیرولوبenzodiazepines; Pyrrolobenzodiazepines; PBDs; DNA-binding; DNA sequence-selective; Fluorescence conjugates; Nuclear penetration; Anticancer agents; Antitumour agents
Remarkable DNA binding affinity and potential anticancer activity of pyrrolo[2,1-c][1,4]benzodiazepine–naphthalimide conjugates linked through piperazine side-armed alkane spacers
Keywords: پیرولوبenzodiazepines; Pyrrolobenzodiazepines; Naphthalimides; Piperazine ring; DNA binding affinity; Anticancer activity
1,2,4-Benzothiadiazine linked pyrrolo[2,1-c][1,4]benzodiazepine conjugates: Synthesis, DNA-binding affinity and cytotoxicity
Keywords: پیرولوبenzodiazepines; Benzothiadiazines; Pyrrolobenzodiazepines; Cytoxicity; DNA binding
Design, synthesis, and biological testing of pyrazoline derivatives of combretastatin-A4
Keywords: پیرولوبenzodiazepines; Combretastatins; Tubulin; Anti-cancer; Pyrazolines; CC-1065; Duocarmycins; Pyrrolobenzodiazepines; Achiral; seco-Amino-CBI; Dimer
Synthesis, DNA binding, and cytotoxicity studies of pyrrolo[2,1-c][1,4]benzodiazepine-anthraquinone conjugates
Keywords: پیرولوبenzodiazepines; Pyrrolobenzodiazepines; Anthraquinones; DNA binding; Anticancer activity
Binding of f-PIP, a pyrrole- and imidazole-containing triamide, to the inverted CCAAT box-2 of the topoisomerase IIα promoter and modulation of gene expression in cells
Keywords: پیرولوبenzodiazepines; CC-1065; Duocarmycins; Pyrrolobenzodiazepines; Achiral; sec-amino-CBI; Dimer; Polyamides; Sequence specificity; Footprinting; SPR; Gene control; Topoisomerase;
DNA interstrand crosslinking agents: Synthesis, DNA interactions, and cytotoxicity of dimeric achiral seco-amino-CBI and conjugates of achiral seco-amino-CBI with pyrrolobenzodiazepine (PBD)
Keywords: پیرولوبenzodiazepines; CC-1065; Duocarmycins; Pyrrolobenzodiazepines; Achiral; Seco-amino-CBI; Dimer
Voltammetric studies of the interaction of pyrrolo[2,1-c][1,4]benzodiazepine (PBD) monomers and dimers with DNA
Keywords: پیرولوبenzodiazepines; Drug–DNA interactions; Pyrrolobenzodiazepines; PBDs; Voltammetry
Synthesis and biological activity of fluoroquinolone-pyrrolo[2,1-c][1,4]benzodiazepine conjugates
Keywords: پیرولوبenzodiazepines; Pyrrolobenzodiazepines; Fluoroquinolones; DNA binding ability; Cytotoxicity;