Keywords: کوینازولین ها; Gefitinib; Erlotinib; Resveratrol; Chalcones; Quinazolines; Cytotoxicity;
مقالات ISI کوینازولین ها (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: کوینازولین ها; Quinazolines; Alkylation; Hydrazinolysis; HeLa; MDA-MB231; Gefitinib; Cytotoxicity;
Keywords: کوینازولین ها; Quinazolines; Oxidative annulation; Metal free; Heteroaromatic;
Keywords: کوینازولین ها; Nitrotriazoles; Nitroimidazoles; Quinolines; Quinazolines; Antitubercular agents; Antitrypanosomal agents; CZJJFJQBTHKAJW-UHFFFAOYSA-N; XWENOZDPQVGKLN-UHFFFAOYSA-N; KACPFNVXZVUZTK-UHFFFAOYSA-N; DJOAKGAPTRKBQU-UHFFFAOYSA-N; VWRUWQZIUYOBDA-UHFFFAOYSA-N; GNK
Keywords: کوینازولین ها; Quinazolines; Copper; CH aminations; Methylarenes
Keywords: کوینازولین ها; PCM analysis; âGsol; Cavitation energy; Induced dipole moments; Quinazolines;
Keywords: کوینازولین ها; Quinazolines; Quinazolinones; Phenylacetylene; Asymmetric alkynylation; Propargylic alcohol; Diethylzinc and organozinc addition;
Keywords: کوینازولین ها; Heterocycles; Synthetic methods; Inhibitors; Quinazolines; Quinazolinones; Biological activities
Keywords: کوینازولین ها; Antibiotics; Staphylococcus aureus; Enterococcus faecalis; Bacteriostatic; Bactericidal; Quinoxalines; Quinazolines; 1,5-Naphthyridines;
Keywords: کوینازولین ها; Guanidines; Pyrimidines; Quinazolines; Atwal-Biginelli reaction; Screening library;
Gold(0) catalyzed dehydrogenation of N-heterocycles
Keywords: کوینازولین ها; Gold; Catalytic dehydrogenation; Indoles; Quinazolines;
Structure-activity relationships for inhibitors of Pseudomonas aeruginosa exoenzyme S ADP-ribosyltransferase activity
Keywords: کوینازولین ها; Pseudomonas aeruginosa; Type III secretion; Bacterial exotoxins; ExoS; ADP-Ribosyltransferase; 2-Aminobenzamide; Quinazolines;
N-(1H-Pyrazol-3-yl)quinazolin-4-amines as a novel class of casein kinase 1δ/ε inhibitors: Synthesis, biological evaluation and molecular modeling studies
Keywords: کوینازولین ها; Quinazolines; Protein kinases; Casein kinase 1δ/ε; MTT assay; Neurodegenerative diseases; Cancer;
Synthesis of new 3-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-benzenesulfonamides with strong inhibition properties against the tumor associated carbonic anhydrases IX and XII
Keywords: کوینازولین ها; Carbonic anhydrase inhibitors (CAIs); Quinazolines; Tumors; Imaging;
Synthesis and biological investigation of 2,4-substituted quinazolines as highly potent inhibitors of breast cancer resistance protein (ABCG2)
Keywords: کوینازولین ها; ABC transporter; Inhibitor; ABCG2; Quinazolines; BCRP;
Synthesis and antinociceptive activity of new 2-substituted 4-(trifluoromethyl)-5,6-dihydrobenzo[h]quinazolines
Keywords: کوینازولین ها; Quinazolines; Trifluoromethyl; Pyrroles; Arthritis; Anti-hyperalgesic effect;
Recent advances in 4-aminoquinazoline based scaffold derivatives targeting EGFR kinases as anticancer agents
Keywords: کوینازولین ها; Quinazolines; EGFR inhibitors; Protein kinases; Tyrosine kinase inhibitors
Toxicological studies for adults and children of insecticide residues with common mode of action (MoA) in pome, stone, berries and other small fruit
Keywords: کوینازولین ها; AC; Acetamiprid; BZLs; Benzoylureas; CARs; Carbamates; ChL; Chlorpyrifos ethyl; ChHs; Chlorinate hydrocarbons; CP; Cypermethrin; CL (λ); Lambda-cyhalothrin; DE; Deltamethrin; DI; Diazinon; DM; Dimethoate; DSFs; Disinfecants; EN; Endosulfan; ES; Esfenvale
Toward discovery of mutant EGFR inhibitors; Design, synthesis and in vitro biological evaluation of potent 4-arylamino-6-ureido and thioureido-quinazoline derivatives
Keywords: کوینازولین ها; EGFR inhibitors; Quinazolines; Urea derivatives; Synthesis; EGFR-Her2 dual inhibitors; EGFR L858R/T790 mutant; EGFR Del19/T790M mutant;
The combination of quinazoline and chalcone moieties leads to novel potent heterodimeric modulators of breast cancer resistance protein (BCRP/ABCG2)
Keywords: کوینازولین ها; ABC transporter; ABCG2; Multidrug resistance; Chalcones; Quinazolines; Quinazoline-chalcones; Pheophorbide A assay; ATPase; ABC; ATP-binding cassette; BCRP; breast cancer resistance protein;
The reaction of 2-amino-Nâ²-arylbenzamidines with tetracyanoethene reinvestigated: routes to imidazoles, quinazolines and quinolino[2â²,3â²:4,5]imidazo[1,2-c]quinazoline-8-carbonitrile
Keywords: کوینازولین ها; Heterocycles; Quinazolines; Imidazoles; Tetracyanoethylene; Amidines; Cyclization reactions;
Discovery of 4-aminoquinazoline-urea derivatives as Aurora kinase inhibitors with antiproliferative activity
Keywords: کوینازولین ها; ZM447439; Aurora kinase; Antiproliferative activity; Cancer cell; Quinazolines; Docking simulation;
Copper-catalyzed domino reaction between 1-(2-halophenyl)methanamines and amidines or imidates for the synthesis of 2-substituted quinazolines
Keywords: کوینازولین ها; Copper; Quinazolines; Domino reaction; N-Arylation;
Assembly of 4H-chromenes, imidazobenzothiazines and quinazolines via copper-catalyzed domino reactions using 2-halobenzyl tosylates as substrates
Keywords: کوینازولین ها; Copper; Chromenes; Imidazobenzothiazines; Quinazolines; Domino reaction;
Investigation of quinazolines as inhibitors of breast cancer resistance protein (ABCG2)
Keywords: کوینازولین ها; ATP binding cassette (ABC) transporter; Breast cancer resistance protein (BCRP/ABCG2); Multidrug resistance; Quinazolines; Hoechst 33342 accumulation assay;
Solvent selection in synthesis of 4-(1-arylfluoroethoxy)quinazolines and thienopyrimidines
Keywords: کوینازولین ها; Solvent selection; Quinazolines; Thienopyrimidines; 1-Aryl-2-fluoroethanols; Cs2CO3; 4-Alkoxypyrimidine
Design and synthesis of novel 4-benzothiazole amino quinazolines Dasatinib derivatives as potential anti-tumor agents
Keywords: کوینازولین ها; Dasatinib; Tyrosine kinase; Cytotoxic activity; Cancer cell; quinazolines; CML
4-Substituted-2-phenylquinazolines as inhibitors of BCRP
Keywords: کوینازولین ها; BCRP; Inhibitors; Multidrug resistance; Quinazolines; Hoechst 33342;
Novel piperidine-fused benzoxazino- and quinazolinonaphthoxazines-synthesis and conformational study
Keywords: کوینازولین ها; Quinazolines; Naphthoxazines; DFT structural study; Conformational analysis; NMR spectroscopy;
Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: Part 2
Keywords: کوینازولین ها; Melanin concentrating hormone (MCH); Quinazolines; MCHR1 antagonists; hERG; Obesity;
Design and synthesis of fluorescent 6-aryl[1,2-c]quinazolines serving as selective and sensitive 'on-off' chemosensor for Hg2+ in aqueous media
Keywords: کوینازولین ها; Synthesis; Quinazolines; Crystal structure; UV-vis; Fluorescence; Mercury selective; Quenching;
Copper-catalyzed three-component one-pot synthesis of quinazolines
Keywords: کوینازولین ها; Ammonia water; ortho-Bromo aromatic ketones; ortho-Bromo aromatic aldehydes; Aromatic aldehydes; Primary alcohols; Quinazolines;
Neuroprotective efficacy of quinazoline type phosphodiesterase 7 inhibitors in cellular cultures and experimental stroke model
Keywords: کوینازولین ها; PDE7 inhibitors; Neuroprotection; Stroke; Quinazolines
Cytotoxic potential of novel 6,7-dimethoxyquinazolines
Keywords: کوینازولین ها; Quinazolines; Quinazolinones; Colon cancer; Anticancer agents; Ovarian cancer
Sulfur and selenium derivatives of quinazoline and pyrido[2,3-d]pyrimidine: Synthesis and study of their potential cytotoxic activity in vitro
Keywords: کوینازولین ها; Cytotoxics; Antiproliferatives; Quinazolines; Pyridopyrimidines
Molecular iodine-catalyzed and air-mediated tandem synthesis of quinolines via three-component reaction of amines, aldehydes, and alkynes
Keywords: کوینازولین ها; Molecular iodine; Quinolines; Multicomponent reaction; Quinazolines;
Microwave-assisted thermal decomposition of formamide: a tool for coupling a pyrimidine ring with an aromatic partner
Keywords: کوینازولین ها; Microwave chemistry; Decomposition of formamide; Quinazolines; Dielectric properties; Niementowski reaction;
Using the TOPS-MODE approach to fit multi-target QSAR models for tyrosine kinases inhibitors
Keywords: کوینازولین ها; Tyrosine kinase inhibitors; QSAR; TOPS-MODE; Quinazolines;
Virtual screening and synthesis of quinazolines as novel JAK2 inhibitors
Keywords: کوینازولین ها; JAK2; Quinazolines; Virtual screening; SurflexDock; Apoptosis; Stem cell; AG490
Synthesis of 4-allylquinazolines from N-(2-cyanoaryl)amides via the In-mediated allylation of nitrile and dehydrative cyclization cascade
Keywords: کوینازولین ها; Quinazolines; Indium; Nitrile; Allylation; Barbier reaction;
A convenient synthesis of quinazoline derivatives via cascade imino-Diels-Alder and oxidation reaction
Keywords: کوینازولین ها; Quinazolines; α-Iminoesters; Imino-Diels-Alder reaction; CuBr2
Click chemistry: Studies on the synthesis of novel fluorous tagged triazol-4-yl substituted quinazoline derivatives and their biological evaluation – Theoretical and experimental validation
Keywords: کوینازولین ها; Quinazolines; Propargylation; Perfluoroalkyl azides; Click reaction; Selective cyclisation; Sharpless conditions
Quinazolines as novel anti-inflammatory histone deacetylase inhibitors
Keywords: کوینازولین ها; Epigenetics; Histone deacetylase inhibitor; Chronic inflammation; Quinazolines;
3D-QSAR studies on quinazoline antifolate thymidylate synthase inhibitors by CoMFA and CoMSIA models
Keywords: کوینازولین ها; CoMFA; CoMSIA; QSAR; Quinazolines; Thymidylate synthase inhibitors;
Design and synthesis of novel substituted quinazoline derivatives as antileishmanial agents
Keywords: کوینازولین ها; Quinazolines; Pyrimidines; Antileishmanial agents
Analogs of a 4-aminothieno[2,3-d]pyrimidine lead (QB13) as modulators of P-glycoprotein substrate specificity
Keywords: کوینازولین ها; ABC transporters; P-Glycoprotein; Multidrug resistance; Thienopyrimidines; Quinazolines
Promising carboranylquinazolines for boron neutron capture therapy: Synthesis, characterization, and in vitro toxicity evaluation
Keywords: کوینازولین ها; Quinazolines; NMR spectroscopy; BNCT; Carboranes; Anti-tumor agents
Synthesis of aza analogues of the anticancer agent batracylin
Keywords: کوینازولین ها; Batracylin; Quinazolines; Pyridines; Mitsunobu reaction; Quinazolinones;
Synthesis of the antitumoural agent batracylin and related isoindolo[1,2-b]quinazolin-12(10H)-ones
Keywords: کوینازولین ها; Batracylin; Quinazolines; Mitsunobu reaction; Quinazolinones;
Regioselective addition of Grignard reagents to 2,6-dicyanoanilines and cyclization to new quinazoline derivatives under thermal/microwave irradiation conditions
Keywords: کوینازولین ها; 2,6-Dicyanoanilines; Regioisomers; Quinazolines; Grignard reagents