Keywords: بازدارنده انتخابی; Chitotriosidase; Chitinase; Selective inhibitor; mCHIT1; Fibrosis;
مقالات ISI بازدارنده انتخابی (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: بازدارنده انتخابی; Glycyrrhetinic acid; Structure-activity relationship; Human carboxylesterase 2; Selective inhibitor;
Keywords: بازدارنده انتخابی; Immunoproteasome; Selective inhibitor; Non-peptide scaffold; Inhibitor identification;
Keywords: بازدارنده انتخابی; Endoplasmic reticulum aminopeptidase; ERAP1; ERAP2; IRAP; Selective inhibitor; Rational design; Molecular modeling;
Bysspectin A, an unusual octaketide dimer and the precursor derivatives from the endophytic fungus Byssochlamys spectabilis IMM0002 and their biological activities
Keywords: بازدارنده انتخابی; Byssochlamys spectabilis; Polyketide-derived octaketide dimer; Human carboxylesterase 2; Selective inhibitor;
Discovery of the selective sphingomyelin synthase 2 inhibitors with the novel structure of oxazolopyridine
Keywords: بازدارنده انتخابی; SMS; sphingomyelin synthase; SM; sphingomyelin; PC; phosphatidylcholine; CHD; coronary heart disease; SMase; sphingomyelinase; SPT; serine palmitoyl transferase; AS; atherosclerosis; SMSr; SMS related protein; SAR; structure-activity relationships; IC50;
Selective inhibition of monoamine oxidase A by purpurin, an anthraquinone
Keywords: بازدارنده انتخابی; Purpurin; Monoamine oxidase A; Selective inhibitor; Competitive inhibitor; Molecular docking;
Selective inhibitors of human mPGES-1 from structure-based computational screening
Keywords: بازدارنده انتخابی; Prostaglandin; Inflammation; Selective inhibitor; Inhibitor identification;
Design and synthesis of polyhydroxy steroids as selective inhibitors against AKR1B10 and molecular docking
Keywords: بازدارنده انتخابی; Synthesis; Polyhydroxy steroids; AKR1B10; Selective inhibitor; Anti-cancer
Molecular design and structural optimization of potent peptide hydroxamate inhibitors to selectively target human ADAM metallopeptidase domain 17
Keywords: بازدارنده انتخابی; ADAM17; ADAM10; Peptide hydroxamate; Selective inhibitor; Inflammatory bowel disease
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII
Keywords: بازدارنده انتخابی; KBYGAQLHLOBGDS-CYGOZCHUSA-N; Carbonic anhydrase; Sulfonamide; Tumor-associated isoform; Selective inhibitor;
Inhibition studies of bacterial, fungal and protozoan β-class carbonic anhydrases with Schiff bases incorporating sulfonamide moieties
Keywords: بازدارنده انتخابی; Pathogenic microorganism; Anti-infective; Bacteria; Beta-carbonic anhydrase; Selective inhibitor; Fungi; Protozoa; Schiff base; Sulfonamide;
Modeling, predicting and virtual screening of selective inhibitors of MMP-3 and MMP-9 over MMP-1 using random forest classification
Keywords: بازدارنده انتخابی; Matrix metalloproteinase; Selective inhibitor; Molecular descriptor; Random forest; Modeling; Virtual screening
Identification of the 5,5-dioxo-7,8-dihydro-6H-thiopyrano[3,2-d]pyrimidine derivatives as highly selective PDE4B inhibitors
Keywords: بازدارنده انتخابی; PDE4; PDE4B; PDE4D; Selective inhibitor; Full length; COPD;
Immobilized cholinesterases capillary reactors on-flow screening of selective inhibitors
Keywords: بازدارنده انتخابی; Selective inhibitor; Screening; Statistical comparation; Butyrylcholinesterase; Acetylcholinesterase; Enzymatic inhibition assays
Synthesis of new ibuprofen derivatives with their in silico and in vitro cyclooxygenase-2 inhibitions
Keywords: بازدارنده انتخابی; Cyclooxygenase-2; Ibuprofen; Molecular docking; Molecular modeling; Selective inhibitor
Synthesis and evaluation of copper complexes of Schiff-base condensates from 5-substituted-2-hydroxybenzaldehyde and 2-substituted-benzenamine as selective inhibitors of protein tyrosine phosphatases
Keywords: بازدارنده انتخابی; Copper complexes; Protein tyrosine phosphatases; Selective inhibitor; Schiff base; CSD; Cambridge Structural Database; ESI-MS; electrospray ionization mass spectra; Hcpmp; 4-chloro-2-((phenylimino)methyl)phenol; Hnpmp; 4-bromo-2-((phenylimino)methyl)pheno
An approach for differentiating isozymes. Construction of libraries containing short aromatic peptides as part of a method to design selective inhibitors against lipases
Keywords: بازدارنده انتخابی; Lipase; Peptidyl substrate; Selective inhibitor; Fingerprint; Isozymes;
Exploration of α-aminophosphonate N-derivatives as novel, potent and selective inhibitors of protein tyrosine phosphatases
Keywords: بازدارنده انتخابی; α-Aminophosphonate; Protein tyrosine phosphatases; Competitive inhibitor; Selective inhibitor; Cell viability; ApoptosisDMEM, Dulbecco's modified Eagle's medium; EA, elemental analysis; ESI-MS, electrospray ionization mass spectrometry; FBS, fetal bovine
Synthesis of new glycyrrhetinic acid derived ring A azepanone, 29-urea and 29-hydroxamic acid derivatives as selective 11β-hydroxysteroid dehydrogenase 2 inhibitors
Keywords: بازدارنده انتخابی; 11β-Hydroxysteroid dehydrogenase; 11β-HSD1; 11β-HSD2; Selective inhibitor; Hydroxamic acid; Glycyrrhizin; Glycyrrhetinic acid; Carbenoxolone; Glucocorticoid metabolism; Cortisone metabolism; Inflammation; Chronic inflammatory disease; Cancer;
Peripheral but crucial: A hydrophobic pocket (Tyr706, Leu337, and Met336) for potent and selective inhibition of neuronal nitric oxide synthase
Keywords: بازدارنده انتخابی; Nitric oxide synthase; Selective inhibitor; Crystal structure; Peripheral hydrophobic pocket; Pi-stacking
Selective inhibition of methoxyflavonoids on human CYP1B1 activity
Keywords: بازدارنده انتخابی; CYP1; Methoxyflavonoid; Molecular docking study; Selective inhibitor; Structure–property relationship
Synthesis of novel 3-amino and 29-hydroxamic acid derivatives of glycyrrhetinic acid as selective 11β-hydroxysteroid dehydrogenase 2 inhibitors
Keywords: بازدارنده انتخابی; 11β-Hydroxysteroid dehydrogenase; 11β-HSD1; 11β-HSD2; Selective inhibitor; Hydroxamic acid; Glycyrrhizin; Glycyrrhetinic acid; Carbenoxolone; Glucocorticoid metabolism; Cortisone metabolism; Inflammation; Chronic inflammatory disease; Cancer
Carbonic anhydrase inhibitors; Fluorinated phenyl sulfamates show strong inhibitory activity and selectivity for the inhibition of the tumor-associated isozymes IX and XII over the cytosolic ones I and II
Keywords: بازدارنده انتخابی; Carbonic anhydrase; Sulfamate; Fluorophenyl; Tumor-associated isoforms; Selective inhibitor;
AKR1C3 as a potential target for the inhibitory effect of dietary flavonoids
Keywords: بازدارنده انتخابی; Aldo-keto reductases (AKRs); Flavonoids; Oracin; Inhibition; Selective inhibitor
Carbonic anhydrase inhibitors: Inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides
Keywords: بازدارنده انتخابی; Carbonic anhydrase; Sulfonamide; Tumor-associated isoform IX and XII; Selective inhibitor
Interaction mode and selectivity of the 2PU inhibitor with the CDK4 and CDK2 cyclin-dependant kinases: A molecular dynamics study
Keywords: بازدارنده انتخابی; Cyclin-dependant kinases; Selective inhibitor; Molecular dynamics;
3D QSAR studies on a series of potent and high selective inhibitors for three kinases of RTK family
Keywords: بازدارنده انتخابی; KDR; cKit; Tie-2; CoMFA; CoMSIA; Selective inhibitor
Tetrabromobenzotriazole (TBBt) and tetrabromobenzimidazole (TBBz) as selective inhibitors of protein kinase CK2: Evaluation of their effects on cells and different molecular forms of human CK2
Keywords: بازدارنده انتخابی; CK2; protein kinase CK2; TBBt; tetrabromobenzotriazole; TBBz; tetrabromobenzimidazole; DRB; 5,6-dichloro-1-(β-d-ribofuranosyl)benzimidazole; CKA1 and CKA2; the catalytic subunits of protein kinase CK2 in S. cerevisiae; FACS; fluorescence activated cell s